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SaveStructure-Based Design and Optimization of FPPQ, a Dual-Acting 5-HT3 and 5-HT6 Receptor Antagonist with Antipsychotic and Procognitive Properties
Zajdel, Pawel; Grychowska, Katarzyna; Mogilski, Szczepan; Kurczab, Rafal; Satala, Grzegorz; Bugno, Ryszard; Kos, Tomasz; Golebiowska, Joanna; Malikowska-Racia, Natalia; Nikiforuk, Agnieszka; Chaumont-Dubel, Severine; Bantreil, Xavier; Pawlowski, Maciej; Martinez, Jean; Subra, Gilles; Lamaty, Frederic; Marin, Philippe; Bojarski, Andrzej J.; Popik, Piotr
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SavePotent Lys Patch-Containing Stapled Peptides Targeting PCSK9
Bourbiaux, Kevin; Legrand, Baptiste; Verdie, Pascal; Mallart, Sergio; Manette, Geraldine; Minoletti, Claire; Stepp, J. David; Prigent, Philippe; Le Bail, Jean-Christophe; Gauzy-Lazo, Laurence; Duclos, Olivier; Martinez, Jean; Amblard, Muriel
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Save2-Phenyl-1H-pyrrole-3-carboxamide as a New Scaffold for Developing 5-HT6 Receptor Inverse Agonists with Cognition-Enhancing Activity
Drop, Marcin; Canale, Vittorio; Chaumont-Dubel, Severine; Kurczab, Rafal; Satala, Grzegorz; Bantreil, Xavier; Walczak, Maria; Koczurkiewicz-Adamczyk, Paulina; Latacz, Gniewomir; Gwizdak, Anna; Krawczyk, Martyna; Golebiowska, Joanna; Grychowska, Katarzyna; Bojarski, Andrzej J.; Nikiforuk, Agnieszka; Subra, Gilles; Martinez, Jean; Pawlowski, Maciej; Popik, Piotr; Marin, Philippe; Lamaty, Frederic; Zajdel, Pawel
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SaveDirect Synthesis of Peptide-Containing Silicones: A New Way to Bioactive Materials
Martin, Julie; Wehbi, Mohammad; Echalier, Cecile; Hunger, Sylvie; Bethry, Audrey; Garric, Xavier; Pinese, Coline; Martinez, Jean; Vezenkov, Lubomir; Subra, Gilles; Mehdi, Ahmad
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SavePain relief devoid of opioid side effects following central action of a silylated neurotensin analog
Tetreault, Pascal; Besserer-Offroy, Elie; Brouillette, Rebecca L.; Rene, Adeline; Murza, Alexandre; Fanelli, Roberto; Kirby, Karyn; Parent, Alexandre J.; Dubuc, Isabelle; Beaudet, Nicolas; Cote, Jerome; Longpre, Jean-Michel; Martinez, Jean; Cavelier, Florine; Sarret, Philippe
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SaveTurning peptides into bioactive nylons
Jebors, Said; Pinese, Coline; Montheil, Titouan; Bethry, Audrey; Verquin, Simon; Plais, Louise; Moulin, Marie; Dupont, Chloe; Garric, Xavier; Mehdi, Ahmad; Martinez, Jean; Subra, Gilles
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SaveSolid-Phase Synthesis of Substrate-Based Dipeptides and Heterocyclic Pseudo-dipeptides as Potential NO Synthase Inhibitors
Touati-Jallabe, Youness; Tintillier, Thibault; Mauchauffee, Elodie; Boucher, Jean-Luc; Leroy, Jeremy; Ramassamy, Booma; Hamze, Abdallah; Mezghenna, Karima; Bouzekrini, Amine; Verna, Claudia; Martinez, Jean; Lajoix, Anne-Dominique; Hernandez, Jean-Francois
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SaveSelf-mineralization and assembly of a bis-silylated Phe-Phe pseudodipeptide to a structured bioorganic-inorganic material
Jebors, Said; Valot, Laurine; Echalier, Cecile; Legrand, Baptiste; Mikhaleff, Remi; Van der Lee, Arie; Arenal, Raul; Dumy, Pascal; Amblard, Muriel; Martinez, Jean; Mehdi, Ahmad; Subra, Gilles
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Save12/10-Helix in Mixed β-Peptides Alternating Bicyclic and Acyclic β-Amino Acids: Probing the Relationship between Bicyclic Side Chain and Helix Stability
Simon, Matthieu; Milbeo, Pierre; Liu, Hongtao; Andre, Christophe; Wenger, Emmanuel; Martinez, Jean; Amblard, Muriel; Aubert, Emmanuel; Legrand, Baptiste; Calmes, Monique
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