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Jens Meiler

institute for drug discovery

78H-index
872Paper Count
3.2WCitation Count
Published Papers 279
Publication Date
Rapid and energy-efficient ultra-large library screening for drug discovery on a SpiNNaker2 neuromorphic chip
err2026-07-21
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errJohnny Alexander Jimenez Siegert; Florian Kelber; Bernhard Vogginger; Paul Eisenhuth; Max Beining; Vivian Ehrlich; Johannes Partzsch; Christian Mayr; Jens Meiler
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The pathway-independent positive allosteric modulator C1 allows for the identification of active Y4 receptor relevant positions
err2026-01-13
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errCorinna Schüß; Oanh Vu; Tim Pelczyk; Mario Schubert; Yu Du; Jan Stichel; C. David Weaver; Jens Meiler; Annette G. Beck-Sickinger
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Superwater as a generative AI framework to predict water molecule positions on protein structures
err2025-12-18
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errXiaohan Kuang; Yunchao Lance Liu; Xiaobo Lin; Jesse Spencer-Smith; Tyler Derr; Yinghao Wu; Hans Bitter; Yongbo Hu; Jens Meiler; Zhaoqian Su
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Phenotypic Variability and Paternal Inheritance of a CHD8 Variant Causing Intellectual Developmental Disorder With Autism and Macrocephaly Confirmed by Epigenetic and Structural Analyses
err2025-12-17
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errFuruta, Yutaka; Ezell, Kimberly M.; Hamid, Rizwan; Cogan, Joy D.; Cassini, Thomas A.; Rives, Lynette; McMinn, Ashley; Shah, Shailee; Peltier, Amanda C.; Layfield, Stephen; Fletcher, Robin S.; Tedder, Matthew L.; Louie, Raymond J.; Lee, Jennifer A.; Kerkhof, Jennifer; Rzasa, Jessica; Sadikovic, Bekim; Al Mamun, Abdullah; Sheehan, Jonathan H.; Moth, Christopher W.; Meiler, Jens; Vawter-lee, Marissa; Mendoza-sengco, Paola Maria; Holzen, Jennifer B.; Pruthi, Sumit; Phillips III, John A.; Tinker, Rory J.
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General trends in the calnexin-dependent expression and pharmacological rescue of clinical CFTR variants
err2025-12-11
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PREAI
errTedman, Austin; Olson, John A.; Kim, Minsoo; Foye, Catherine; Jackson, Janise J.; McDonald, Eli F.; McKee, Andrew G.; Noguera, Karen; Kuntz, Charles P.; Meiler, Jens; Oliver, Kathryn E.; Plate, Lars; Schlebach, Jonathan P.
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Investigating the neuronal role of the proteasomal ATPase subunit gene PSMC5 in neurodevelopmental proteasomopathies
err2025-11-26
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errSébastien Küry; Janelle E. Stanton; Geeske M. van Woerden; Amélie Bosc-Rosati; Tzung-Chien Hsieh; Lise Bray; Marielle Oloudé; Cory Rosenfelt; Marie Pier Scott-Boyer; Victoria Most; Tianyun Wang; Jonas J. Papendorf; Charlotte de Konink; Wallid Deb; Virginie Vignard; Maja Studencka-Turski; Thomas Besnard; Anna M. Hajdukowicz; Franziska G. Thiel; Sophie Wolfgramm; Laëtitia Florenceau; Silvestre Cuinat; Sylvain Marsac; Yann Verrès; Audrey Dangoumau; Léa Poirier; Ingrid M. Wentzensen; Annabelle Tuttle; Cara Forster; Johanna Striesow; Richard Golnik; Damara Ortiz; Laura Jenkins; Jill A. Rosenfeld; Alban Ziegler; Clara Houdayer; Dominique Bonneau; Erin Torti; Amber Begtrup; Kristin G. Monaghan; Sureni V. Mullegama; Catharina M. L. Nienke Volker-Touw; Koen L. I. van Gassen; Renske Oegema; Mirjam S. de Pagter; Katharina Steindl; Anita Rauch; Ivan Ivanovski; Kimberly McDonald; Emily Boothe; Andrew Dauber; Janice Baker; Noelle Andrea V. Fabie; Raphael A. Bernier; Tychele N. Turner; Siddharth Srivastava; Kira A. Dies; Lindsay C. Swanson; Carrie Costin; Alali Abdulrazak; Rebekah K. Jobling; John Pappas; Rachel Rabin; Dmitriy Niyazov; Anne Chun-Hui Tsai; Karen Kovak; David B. Beck; May Christine V. Malicdan; David R. Adams; Lynne Wolfe; Rebecca D. Ganetzky; Colleen C. Muraresku; Davit Babikyan; Zdeněk Sedláček; Miroslava Hančárová; Andrew T. Timberlake; Hind Al Saif; Berkley Nestler; Kayla King; MJ Hajianpour; Gregory Costain; D’Arcy Prendergast; Chumei Li; David Geneviève; Antonio Vitobello; Arthur Sorlin; Christophe Philippe; Tamar Harel; Ori Toker; Ataf Sabir; Derek Lim; Mark J. Hamilton; Lisa J. Bryson; Elaine Cleary; Sacha Weber; Trevor L. Hoffman; Anna M. Cueto-González; Eduardo F. Tizzano; David Gómez-Andrés; Marta Codina-Solà; Athina Ververi; Efterpi Pavlidou; Alexandros Lambropoulos; Kyriakos Garganis; Marlène Rio; Jonathan Levy; Sarah J. Langas; Anne M. McRae; Mathieu K. Lessard; Maria Daniela D’Agostino; Isabelle De Bie; Meret Wegler; Rami Abou Jamra; Susanne B. Kamphausen; Viktoria Bothe; Lorraine Potocki; Eric Olinger; Yves Sznajer; Elsa Wiame; Michelle L. Thompson; Molly C. Schroeder; Catherine Gooch; Raphael A. Smith; Arti Pandya; Larissa M. Busch; Uwe Völker; Elke Hammer; Kristian Wende; Benjamin Cogné; Bertrand Isidor; Jens Meiler; Clémentine Ripoll; Stéphanie Bigou; Frédéric Laumonnier; Peter W. Hildebrand; Evan E. Eichler; Kirsty McWalter; Peter M. Krawitz; Florence Roux-Dalvai; Ype Elgersma; Julien Marcoux; Marie-Pierre Bousquet; Arnaud Droit; Jeremie Poschmann; Andreas M. Grabrucker; Francois V. Bolduc; Stéphane Bézieau; Frédéric Ebstein; Elke Krüger
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Ultra-large library screening with an evolutionary algorithm in Rosetta (REvoLd)
err2025-11-07
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errOAAI
errPaul Eisenhuth; Fabian Liessmann; Rocco Moretti; Jens Meiler
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Glutamine synthetase deficiency enhances CD8 T cell survival and stress resilience in the tumor microenvironment
err2025-10-01
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PREAI
errFisher-Gupta, Emilie L.; Hathaway, Emma S.; Perera, Jeffrey M.; Jennings, Erin Q.; Chi, Channing; Sewell, Allison E.; Stone, Spenser H.; Muka, Jason E.; Sinard, Rachael C.; Decorte, Joseph A.; Chen, Heidi; Wilson, John T.; Meiler, Jens; Rathmell, Jeffrey C.
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Transient ligand contacts of the intrinsically disordered N-terminus of neuropeptide Y2 receptor regulate arrestin-3 recruitment
err2025-09-19
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errOAAI
errAnette Kaiser; Juan C. Rojas Echeverri; Asat Baischew; Maik Pankonin; Karl D. Leitner; Claudio Iacobucci; Davide Sala; Christian Ihling; Ronny Müller; Rok Ferenc; Annette G. Beck-Sickinger; Peter Schmidt; Jens Meiler; Peter W. Hildebrand; Andrea Sinz
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Genomics-informed drug-repurposing strategy identifies two therapeutic targets for preventing liver disease associated with metabolic dysfunction
err2025-08-07
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errOAAI
errHannah M. Seagle; Alexis T. Akerele; Joseph A. DeCorte; Jacklyn N. Hellwege; Joseph H. Breeyear; Jeewoo Kim; Michael G. Levin; Samuel Khodursky; Adam Bress; Kyung Min Lee; Jens Meiler; Dipender Gill; Jennifer S. Lee; Kent Heberer; Donald R. Miller; Peter D. Reaven; Kyong-Mi Chang; Julie A. Lynch; Nikhil K. Khankari; Megan M. Shuey; Todd L. Edwards; Marijana Vujkovic
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Structural insights into the binding modes of Arrestin-3 finger loop to the neuropeptide Y1 and Y2 receptors
err2025-08-07
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errOAAI
errVarsha Gupta; Jeannette M. Laugwitz; Mateusz Sklodowski; Matthias Voitel; Davide Sala; Anette Kaiser; Matthias Elgeti; Jens Meiler; Daniel Huster; Annette G. Beck-Sickinger; Peter Schmidt; Anja Penk
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Notch activity is modulated by the aGPCR Latrophilin binding the DSL ligand in C. elegans
err2025-07-12
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errWillem Berend Post; Victoria Elisabeth Groß; Daniel Matúš; Iannis Charnay; Fabian Liessmann; Florian Seufert; Peter Hildebrand; Jens Meiler; Anette Kaiser; Torsten Schöneberg; Simone Prömel
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CACHE Challenge #2: Targeting the RNA Site of the SARS-CoV-2 Helicase Nsp13
err2025-06-20
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PREAI
errOleksandra Herasymenko; Madhushika Silva; Abd Al-Aziz A. Abu-Saleh; Ayaz Ahmad; Jesus Alvarado-Huayhuaz; Oscar E. A. Arce; Roly J. Armstrong; Cheryl Arrowsmith; Kelly E. Bachta; Hartmut Beck; Denes Berta; Mateusz K. Bieniek; Vincent Blay; Albina Bolotokova; Philip E. Bourne; Marko Breznik; Peter J. Brown; Aaron D. G. Campbell; Emanuele Carosati; Irene Chau; Daniel J. Cole; Ben Cree; Wim Dehaen; Katrin Denzinger; Karina dos Santos Machado; Ian Dunn; Prasannavenkatesh Durai; Kristina Edfeldt; Aled Edwards; Darren Fayne; Daniel Felfoldi; Kallie Friston; Pegah Ghiabi; Elisa Gibson; Judith Günther; Anders Gunnarsson; Alexander Hillisch; Douglas R. Houston; Jan Halborg Jensen; Rachel J. Harding; Kate S. Harris; Laurent Hoffer; Anders Hogner; Joshua T. Horton; Scott Houliston; Judd F. Hultquist; Ashley Hutchinson; John J. Irwin; Marko Jukič; Shubhangi Kandwal; Andrea Karlova; Vittorio L. Katis; Ryan P. Kich; Dmitri Kireev; David Koes; Nicole L. Inniss; Uta Lessel; Sijie Liu; Peter Loppnau; Wei Lu; Sam Martino; Miles McGibbon; Jens Meiler; Akhila Mettu; Sam Money-Kyrle; Rocco Moretti; Yurii S. Moroz; Charuvaka Muvva; Joseph A. Newman; Leon Obendorf; Brooks Paige; Amit Pandit; Keunwan Park; Sumera Perveen; Rachael Pirie; Gennady Poda; Mykola Protopopov; Vera Pütter; Federico Ricci; Natalie J. Roper; Edina Rosta; Margarita Rzhetskaya; Yogesh Sabnis; Karla J. F. Satchell; Frederico Schmitt Kremer; Thomas Scott; Almagul Seitova; Casper Steinmann; Valerij Talagayev; Olga O. Tarkhanova; Natalie J. Tatum; Dakota Treleaven; Adriano Velasque Werhli; W. Patrick Walters; Xiaowen Wang; Jude Wells; Geoffrey Wells; Yvonne Westermaier; Gerhard Wolber; Lars Wortmann; Jixian Zhang; Zheng Zhao; Shuangjia Zheng; Matthieu Schapira
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Molecular basis for Gβγ-SNARE-mediated inhibition of synaptic vesicle fusion
err2025-06-14
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errOAAI
errAnna R. Eitel; Benjamin K. Mueller; Ali I. Kaya; Montana Young; Jackson B. Cassada; Eric W. Bell; Lauren Schnitkey; Zack Zurawski; Yun Y. Yim; Qiangjun Zhou; Jens Meiler; Heidi E. Hamm
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Similar Binding Mode of a 5-Sulfonylthiouracil Derivative Antagonist at Chemerin Receptors CMKLR1 and GPR1
err2025-05-16
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errSchermeng, Tina; Furll, Alexander; Liessmann, Fabian; von Bredow, Lukas; Stichel, Jan; Weaver, C. David; Tretbar, Maik; Meiler, Jens
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Advancements in Ligand-Based Virtual Screening through the Synergistic Integration of Graph Neural Networks and Expert-Crafted Descriptors
err2025-05-14
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errOAAI
errLiu, Yunchao; Moretti, Rocco; Wang, Yu; Dong, Ha; Yan, Bailu; Bodenheimer, Bobby; Derr, Tyler; Meiler, Jens
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Identification and optimization of a small molecule inhibitor of the ovarian tumor protease of the Crimean-Congo hemorrhagic fever virus
err2025-04-01
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PREAI
errBeckmann, Lorenz; Liessmann, Fabian; Icker, Maik; Rieger, Dominic; Schlegel, Phillip; Urban, Nicole; Schaefer, Michael; Meiler, Jens; Schoeder, Clara T.; Tretbar, Maik
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RosettaHDX: Predicting antibody-antigen interaction from hydrogen-deuterium exchange mass spectrometry data
err2025-03-01
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PREAI
errTran, Minh H.; Martina, Cristina E.; Moretti, Rocco; Nagel, Marcus; Schey, Kevin L.; Meiler, Jens
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