Not logged in The Concise Guide to PHARMACOLOGY 2025/26: Ion channels Alexander, Stephen P. H.; Striessnig, Jorg; Gibb, Alasdair J.; Mathie, Alistair A.; Veale, Emma L.; Kelly, Eamonn; Peach, Chloe J.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Southan, Christopher; Davies, Jamie A.; Aldrich, Richard W.; Attali, Bernard; Baggetta, Austin M.; Becirovic, Elvir; Beech, David J.; Biel, Martin; Bill, Roslyn M.; Caceres, Ana I.; Catterall, William A.; Chua, Han Chow; Conner, Alex C.; Danahay, Henry; Davies, Paul; De Clerq, Katrien; Delling, Markus; Di Virgilio, Francesco; Falzoni, Simonetta; Fang, Wei; Fenske, Stefanie; Fortuny-gomez, Anna; Fountain, Samuel; Chandy, George K.; Ghovanloo, Mohammad-reza; Goldstein, Steve A. N.; Gosling, Martin; Grimm, Christian; Grissmer, Stephan; Ha, Kotdaji; Hales, Tim G.; Hammelmann, Verena; Hanukoglu, Israel; Hu, Meiqin; Ijzerman, Ad P.; Jabba, Sairam V.; Jarvis, Mike; Jensen, Anders A.; Jordt, Sven E.; Kaczmarek, Leonard K.; Kellenberger, Stephan; Kennedy, Charles; King, Brian; Kitchen, Philip; Liu, Qiang; Lynch, Joseph W.; Manville, Rian W.; Meades, Jessica; Mehlfeld, Verena; Nicke, Annette; Offermanns, Stefan; Perez-reyes, Edward; Plant, Leigh D.; Pless, Stephan A.; Rash, Lachlan D.; Ren, Dejian; Rubaiy, Hussein N.; Salman, Mootaz M.; Sieghart, Werner; Sivilotti, Lucia G.; Smart, Trevor G.; Snutch, Terrance P.; Tammaro, Paolo; Tian, Jinbin; Trimmer, James S.; Van Den Eynde, Charlotte; Vergani, Paola; Vriens, Joris; Waxman, Stephen G.; Wei, Aguan D.; Winn, Brenda T.; Wulff, Heike; Xu, Haoxing; Yang, Fan; Yue, Lixia; Zhang, Xiaoli; Zhu, Michael Share Save
The Concise Guide to PHARMACOLOGY 2025/26: G protein-coupled receptors Alexander, Stephen P. H.; Davenport, Anthony P.; Kelly, Eamonn; Gibb, Alasdair J.; Mathie, Alistair A.; Peach, Chloe J.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Southan, Christopher; Davies, Jamie A.; Abbracchio, Maria Pia; Abraham, George R.; Agoulnik, Alexander; Alexander, Wayne; Al-hosaini, Khaled; Back, Magnus; Baker, Jillian G.; Barnes, Nicholas M.; Bathgate, Ross; Beaulieu, Jean-Martin; Beck-Sickinger, Annette G.; Behrens, Maik; Bennett, Kirstie A.; Bernstein, Kenneth E.; Bettler, Bernhard; Birdsall, Nigel J. M.; Blaho, Victoria A.; Bonaventure, Pascal; Boulay, Francois; Bousquet, Corinne; Brauner-Osborne, Hans; Brown, Andrew J.; Burnstock, Geoffrey; Busnelli, Marta; Calo, Girolamo; Caruso, Vanni; Castano, Justo P.; Catt, Kevin J.; Ceruti, Stefania; Chazot, Paul; Chiang, Nan; Chini, Bice; Christopoulos, Arthur; Chun, Jerold; Cianciulli, Antonia; Civelli, Olivier; Clapp, Lucie H.; Couture, Rejean; Cox, Helen M.; Csaba, Zsolt; Dahlgren, Claes; Dautzenberg, Frank M.; Dent, Gordon; Douglas, Steven D.; Dournaud, Pascal; Dubocovich, Margarita L.; Eguchi, Satoru; Escher, Emanuel; Filardo, Edward J.; Fong, Tung; Forsman, Huamei Fu; Fumagalli, Marta; Gainetdinov, Raul R.; Garelja, Michael L.; de Gasparo, Marc; Gbahou, Florence; Gerard, Craig; Gershengorn, Marvin; Glass, Michelle; Gloriam, David E.; Gobeil, Fernand; Goodfriend, Theodore L.; Goudet, Cyril; Gratz, Lukas; Gregory, Karen J.; Gruber, Christian; Gundlach, Andrew L.; Hamann, Jorg; Hanson, Julien; Hartman, Deborah S.; Hauger, Richard L.; Hay, Debbie L.; Heinemann, Akos; Heitman, Laura; Herr, Deron R.; Hollenberg, Morley D.; Holliday, Nicholas D.; Holst, Birgitte; Horiuchi, Mastgugu; Hoyer, Daniel; Hunyady, Laszlo; Husain, Ahsan; IJzerman, Adriaan P.; Inagami, Tadashi; Insel, Paul A.; Jacobson, Kenneth A.; Jacobson, Laura H.; Jensen, Robert T.; Jockers, Ralf; Jonnalagadda, Deepa; Karnik, Sadashiva; Kaupmann, Klemens; Kemp, Jacqueline; Kennedy, Charles; Kihara, Yasuyuki; Kinsolving, Julia; Kitazawa, Takio; Kozielewicz, Pawel; Kreienkamp, Hans-Juergen; Kukkonen, Jyrki P.; Laishram, Luxmichan; Langenhan, Tobias; Langmead, Christopher J.; Larhammar, Dan; Leach, Katie; Lecca, Davide; Lee, John D.; Leeman, Susan E.; Leprince, Jerome; Leurs, Rob; Li, Xaria X.; Liebscher, Ines; Lolait, Stephen J.; Lupp, Amelie; Macrae, Robyn; Maguire, Janet J.; Malfacini, Davide; Manning, Maurice; Marangon, Davide; Martemyanov, Kirill; Mazella, Jean; McArdle, Craig A.; Melmed, Shlomo; Michel, Martin C.; Miller, Laurence J.; Mitolo, Vincenzo; Mouillac, Bernard; Mueller, Christa E.; Murphy, Philip M.; Nahon, Jean-Louis; Neubig, Richard R.; Ngo, Tony; Norel, Xavier; Nyimanu, Duuamene; O'Carroll, Anne-Marie; Offermanns, Stefan; Panaro, Maria Antonietta; Parmentier, Marc; Perry-Hauser, Nicole; Pertwee, Roger G.; Pin, Jean-Philippe; Prossnitz, Eric R.; Qin, Helena Chengxue; Quinn, Mark; Raffaele, Stefano; Ramachandran, Rithwik; Ray, Manisha; Reinscheid, Rainer K.; Buzon, Alejandro Romeral; Rondard, Philippe; Rosenkilde, Mette M.; Rovati, G. Enrico; Ruzza, Chiara; Sanger, Gareth J.; Scholz, Nicole; Schoeneberg, Torsten; Schulte, Gunnar; Schulz, Stefan; Segaloff, Deborah L.; Serhan, Charles N.; Shukla, Arun K.; Singh, Khuraijam Dhanachandra; Smith, Craig M.; Smith, Nicola J.; Staeubert, Claudia; Stoddart, Leigh A.; Sugimoto, Yukihiko; Summers, Roger; Tan, Valerie P.; Thal, David M.; Thomas, Walter (Wally); Timmermans, Pieter B. M. W. M.; Tirupula, Kalyan; Toll, Lawrence; Tulipano, Giovanni; Unal, Hamiyet; Unger, Thomas; Valant, Celine; Vanderheyden, Patrick; Vaudry, David; Vaudry, Hubert; Verbalis, Joseph G.; Vilardaga, Jean-Pierre; Walker, Christopher S.; Wang, Ji Ming; Ward, Donald T.; Wester, Hans-Juergen; Willars, Gary B.; Williams, Tom Lloyd; Woodruff, Trent M.; Wu, Huixian; Yang, Cheng; Yao, Chengcan; Ye, Richard D.; Zaidman, Nathan Share Save
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The solute carrier superfamily interactome Frommelt, Fabian; Ladurner, Rene; Goldmann, Ulrich; Wolf, Gernot; Ingles-Prieto, Alvaro; Lineiro-Retes, Eva; Gelova, Zuzana; Hopp, Ann-Katrin; Christodoulaki, Eirini; Teoh, Shao Thing; Leippe, Philipp; Santini, Brianda L.; Rebsamen, Manuele; Lindinger, Sabrina; Serrano, Iciar; Onstein, Svenja; Klimek, Christoph; Barbosa, Barbara; Pantielieieva, Anastasiia; Dvorak, Vojtech; Hannich, Thomas J.; Schoenbett, Julian; Sansig, Gilles; Mocking, Tamara A. M.; Ooms, Jasper F.; Ijzerman, Adriaan P.; Heitman, Laura H.; Sykacek, Peter; Reinhardt, Juergen; Mueller, Andre C.; Wiedmer, Tabea Share Save
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CC chemokine receptor 2 is allosterically modulated by sodium ions and amiloride derivatives through a distinct sodium ion binding site den Hollander, Lisa S.; Zweemer, Annelien J. M.; Bequignon, Olivier J. M.; Hammerl, Dora M.; Bleijs, Bente T. M.; Veenhuizen, Margo; Lantsheer, Wernard J. F.; Chau, Bobby; van Westen, Gerard J. P.; IJzerman, Adriaan P.; Heitman, Laura H. Share Save
Labeling of CC Chemokine Receptor 2 with a Versatile Intracellular Allosteric Probe den Hollander, Lisa S.; Beerkens, Bert L. H.; Dekkers, Sebastian; van Veldhoven, Jacobus P. D.; Zacarias, Natalia V. Ortiz; van der Horst, Cas; Sieders, Elisabeth G.; de Valk, Bert; Wang, Jianhui; Ijzerman, Adriaan P.; van der Es, Daan; Heitman, Laura H. Share Save
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Exploring novel dilazep derivatives as hENT1 inhibitors and potentially covalent molecular tools Dilweg, Majlen A.; Gorostiola Gonzalez, Marina; de Ruiter, Martijn D.; Meijboom, Nadine J.; van Veldhoven, Jacobus P. D.; Liu, Rongfang; Jespers, Willem; van Westen, Gerard J. P.; Heitman, Laura H.; Ijzerman, Adriaan P.; van der Es, Daan Share Save
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Multitarget Thiol-Activated Tetrapyridyl Gold(III) Complexes for Hypoxic Cancer Therapy Zhou, Xue-Quan; Abyar, Selda; Carbo-Bague, Imma; Wang, Lan; Turck, Sebastian; Siegler, Maxime A.; Basu, Uttara; Ott, Ingo; Liu, Rongfang; Ijzerman, Adriaan P.; Bonnet, Sylvestre Share Save
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The Concise Guide to PHARMACOLOGY 2023/24: G protein-coupled receptors Alexander, Stephen P. H.; Christopoulos, Arthur; Davenport, Anthony P.; Kelly, Eamonn; Mathie, Alistair A.; Peters, John A.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Davies, Jamie A.; Abbracchio, Maria Pia; Abraham, George; Agoulnik, Alexander; Alexander, Wayne; Al-hosaini, Khaled; Back, Magnus; Baker, Jillian G.; Barnes, Nicholas M.; Bathgate, Ross; Beaulieu, Jean-Martin; Beck-Sickinger, Annette G.; Behrens, Maik; Bernstein, Kenneth E.; Bettler, Bernhard; Birdsall, Nigel J. M.; Blaho, Victoria; Boulay, Francois; Bousquet, Corinne; Brauner-Osborne, Hans; Burnstock, Geoffrey; Calo, Girolamo; Castano, Justo P.; Catt, Kevin J.; Ceruti, Stefania; Chazot, Paul; Chiang, Nan; Chini, Bice; Chun, Jerold; Cianciulli, Antonia; Civelli, Olivier; Clapp, Lucie H.; Couture, Rejean; Cox, Helen M.; Csaba, Zsolt; Dahlgren, Claes; Dent, Gordon; Douglas, Steven D.; Dournaud, Pascal; Eguchi, Satoru; Escher, Emanuel; Filardo, Edward J.; Fong, Tung; Fumagalli, Marta; Gainetdinov, Raul R.; Garelja, Michael L.; de Gasparo, Marc; Gerard, Craig; Gershengorn, Marvin; Gobeil, Fernand; Goodfriend, Theodore L.; Goudet, Cyril; Gratz, Lukas; Gregory, Karen J.; Gundlach, Andrew L.; Hamann, Jorg; Hanson, Julien; Hauger, Richard L.; Hay, Debbie L.; Heinemann, Akos; Herr, Deron; Hollenberg, Morley D.; Holliday, Nicholas D.; Horiuchi, Mastgugu; Hoyer, Daniel; Hunyady, Laszlo; Husain, Ahsan; Ijzerman, Adriaan P.; Inagami, Tadashi; Jacobson, Kenneth A.; Jensen, Robert T.; Jockers, Ralf; Jonnalagadda, Deepa; Karnik, Sadashiva; Kaupmann, Klemens; Kemp, Jacqueline; Kennedy, Charles; Kihara, Yasuyuki; Kitazawa, Takio; Kozielewicz, Pawel; Kreienkamp, Hans-Juergen; Kukkonen, Jyrki P.; Langenhan, Tobias; Larhammar, Dan; Leach, Katie; Lecca, Davide; Lee, John D.; Leeman, Susan E.; Leprince, Jerome; Li, Xaria X.; Lolait, Stephen J.; Lupp, Amelie; Macrae, Robyn; Maguire, Janet; Malfacini, Davide; Mazella, Jean; McArdle, Craig A.; Melmed, Shlomo; Michel, Martin C.; Miller, Laurence J.; Mitolo, Vincenzo; Mouillac, Bernard; Mueller, Christa E.; Murphy, Philip M.; Nahon, Jean-Louis; Ngo, Tony; Norel, Xavier; Nyimanu, Duuamene; O'Carroll, Anne-Marie; Offermanns, Stefan; Panaro, Maria Antonietta; Parmentier, Marc; Pertwee, Roger G.; Pin, Jean-Philippe; Prossnitz, Eric R.; Quinn, Mark; Ramachandran, Rithwik; Ray, Manisha; Reinscheid, Rainer K.; Rondard, Philippe; Rovati, G. Enrico; Ruzza, Chiara; Sanger, Gareth J.; Schoeneberg, Torsten; Schulte, Gunnar; Schulz, Stefan; Segaloff, Deborah L.; Serhan, Charles N.; Singh, Khuraijam Dhanachandra; Smith, Craig M.; Stoddart, Leigh A.; Sugimoto, Yukihiko; Summers, Roger; Tan, Valerie P.; Thal, David; Thomas, Walter (Wally); Timmermans, Pieter B. M. W. M.; Tirupula, Kalyan; Toll, Lawrence; Tulipano, Giovanni; Unal, Hamiyet; Unger, Thomas; Valant, Celine; Vanderheyden, Patrick; Vaudry, David; Vaudry, Hubert; Vilardaga, Jean-Pierre; Walker, Christopher S.; Wang, Ji Ming; Ward, Donald T.; Wester, Hans-Juergen; Willars, Gary B.; Williams, Tom Lloyd; Woodruff, Trent M.; Yao, Chengcan; Ye, Richard D. Share Save
The Concise Guide to PHARMACOLOGY 2023/24: Ion channels Alexander, Stephen P. H.; Mathie, Alistair A.; Peters, John A.; Veale, Emma L.; Striessnig, Joerg; Kelly, Eamonn; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Davies, Jamie A.; Aldrich, Richard W.; Attali, Bernard; Baggetta, Austin M.; Becirovic, Elvir; Biel, Martin; Bill, Roslyn M.; Caceres, Ana I.; Catterall, William A.; Conner, Alex C.; Davies, Paul; De Clerq, Katrien; Delling, Markus; Di Virgilio, Francesco; Falzoni, Simonetta; Fenske, Stefanie; Fortuny-Gomez, Anna; Fountain, Samuel; George, Chandy; Goldstein, Steve A. N.; Grimm, Christian; Grissmer, Stephan; Ha, Kotdaji; Hammelmann, Verena; Hanukoglu, Israel; Hu, Meiqin; Ijzerman, Ad P.; Jabba, Sairam V.; Jarvis, Mike; Jensen, Anders A.; Jordt, Sven E.; Kaczmarek, Leonard K.; Kellenberger, Stephan; Kennedy, Charles; King, Brian; Kitchen, Philip; Liu, Qiang; Lynch, Joseph W.; Meades, Jessica; Mehlfeld, Verena; Nicke, Annette; Offermanns, Stefan; Perez-Reyes, Edward; Plant, Leigh D.; Rash, Lachlan; Ren, Dejian; Salman, Mootaz M.; Sieghart, Werner; Sivilotti, Lucia G.; Smart, Trevor G.; Snutch, Terrance P.; Tian, Jinbin; Trimmer, James S.; Van den Eynde, Charlotte; Vriens, Joris; Wei, Aguan D.; Winn, Brenda T.; Wulff, Heike; Xu, Haoxing; Yang, Fan; Fang, Wei; Yue, Lixia; Zhang, Xiaoli; Zhu, Michael Share Save
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Development of an Affinity-Based Probe to Profile Endogenous Human Adenosine A3 Receptor Expression Beerkens, Bert L. H.; Snijders, Inge M.; Snoeck, Joep; Liu, Rongfang; Tool, Anton T. J.; Le Devedec, Sylvia E.; Jespers, Willem; Kuijpers, Taco W.; van Westen, Gerard J. P.; Heitman, Laura H.; IJzerman, Adriaan P.; van der Es, Daan Share Save
Kinetic profiling of novel spirobenzo-oxazinepiperidinone derivatives as equilibrative nucleoside transporter 1 inhibitors Vlachodimou, Anna; Bouma, Jara; De Cleyn, Michel; Berthelot, Didier; Pype, Stefan; Bosmans, Jean-Paul; van Vlijmen, Herman; Wroblowski, Berthold; Heitman, Laura H.; IJzerman, Adriaan P. Share Save