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Geoffrey I. Shapiro

dana-farber cancer institute

115H-index
2.0KPaper Count
5.7WCitation Count
Published Papers 303
Publication Date
AI-enhanced adaptive virtual screening of large libraries for ligand discovery
err2026-09-01
err0
errOAAI
errDomiziana Cecchini; AkshatKumar Nigam; Ming Tang; Joana Reis; Matt Koop; Andrea Gottinger; Callum Robert Nicoll; Yao Wang; Abhilash Jayaraj; Süleyman Selim Çınaroglu˘; Ricarda Törner; Yehor Malets; Minko Gehev; Krishna M. Padmanabha Das; Kelly Churion; Jongwan Kim; Nidhin Thomas; Yong Li; Hyuk-Soo Seo; Sirano Dhe-Paganon; Christopher Secker; Mohammad Haddadnia; Alexander Hasson; Minkai Li; Abhishek Kumar; Roni Levin-Konigsberg; Eun-Bee Choi; Geoffrey I. Shapiro; Huel Cox; Luke Sebastian; Chelsea Braithwaite; Puspalata Bashyal; Dmytro S. Radchenko; Aditya Kumar; Lei Yang; Pierre-Yves Aquilanti; Henry Gabb; Amr Alhossary; Eric O’Neill; Gerhard Wagner; Alán Aspuru-Guzik; Yurii S. Moroz; Charalampos G. Kalodimos; Konstantin Fackeldey; John D. Schuetz; Andrea Mattevi; Haribabu Arthanari; Christoph Gorgulla
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Disruption of microhomology-mediated end joining in Ewing sarcoma
err2026-07-21
err0
errOAAI
errShuhei Asada; Guangli Zhu; Jithma Prasad Abeykoon; Yutaro Tanaka; Huy Nguyen; Yuna Hirohashi; Divya R. Iyer; Nicholas William Ashton; Sirisha Mukkavalli; Martha Velazquez; Lige Jiang; Miles Del Busso; Judith Jebastin Thangaiah; Steven I. Robinson; Kalindi Parmar; Eliezer M. Van Allen; Riaz Gillani; Geoffrey I. Shapiro; Alan D. D’Andrea
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Fibroblast growth factor receptor inhibition for succinate dehydrogenase-deficient gastrointestinal stromal tumors: a phase 2 trial
err2026-05-26
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errOAAI
errPriscilla Merriam; James J. Morrow; Emanuele Mazzola; Nicole L. Solimini; Prafulla C. Gokhale; Ping Chi; Alice P. Chen; Mark Agulnik; Melissa Burgess; Scott M. Schuetze; Neeta Somaiah; Brian A. Van Tine; Seth M. Pollack; Gabriel Tinoco; Jonathan Trent; Breelyn A. Wilky; Nicola Bothwick; Benjamin K. Eschle; Vivian Nguyen; Jan H. Beumer; Noushin Rastkari; Shahanawaz Jiwani; Peter I-Fan Wu; Lorraine Pelosof; Matthew L. Hemming; Geoffrey I. Shapiro; George Demetri; Bradley Bernstein; Suzanne George
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Targeting FGFR signaling overcomes therapeutic resistance and immune evasion in oncogenic PIK3CA-driven serous-like endometrial cancer
err2026-05-04
err0
errOAAI
errXin Cheng; Yadong Zhang; Changli Qian; Erica Holdridge; Guruprasad Ananda; Tao Jiang; Jing Ni; Shaozhen Xie; Hao Gu; Renlei Ji; Elena V. Ivanova; Marisa R. Nucci; Zhe Wang; Kaifu Chen; Bose Kochupurakkal; Gordon J. Freeman; Geoffrey I. Shapiro; Joyce Liu; Panagiotis A. Konstantinopoulos; Ursula Matulonis; Jean J. Zhao
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Phase 1 clinical trial of the ataxia telangiectasia and Rad3-related inhibitor berzosertib with irinotecan in patients with advanced solid tumors (ETCTN 9938)
errCancer
IF5.1
err2025-10-29
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PREAI
errLiza C. Villaruz MD; Jingxiao Jin MD; Hong Wang PhD; James J. Lee MD, PhD; Jason J. Luke MD; John C. Rhee MD; Saiama N. Waqar MD; Geoffrey I. Shapiro MD, PhD; James Cleary MD, PhD; Diwakar Davar MD; Timothy F. Burns MD, PhD; Rashmi Verma MD; Manik Amin MD; Leonard Appleman MD, PhD; Kristen K. Ciombor MD; Elizabeth J. Davis MD; Jonathan W. Riess MD; E. Claire Dees MD; Edward J. Kim MD, PhD; Dana Cardin MD; Jianxia Guo PhD; Susan M. Christner BS; Joshua Deppas MS; Angelina M. Parise BS; John C. Schmitz PhD; Bella S. Guerrouahen PhD; Michael Suchko BS; Alejandro Contreras MD, PhD; Li Li PhD; Katherine V. Ferry-Galow PhD; Ting-Chia Chang MS; Shahanawaz Jiwani MD, PhD; Christopher J. Bakkenist PhD; Edward Chu MD; Steven D. Gore MD; Jan H. Beumer PharmD, PhD
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Efficacy of neratinib-based therapy in ERBB2-mutant lung adenocarcinomas: findings from 2 international phase 2 studies
err2025-10-01
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PREAI
errBob T. Li; Leena Gandhi; Vignesh Ravichandran; Benjamin Besse; Julien Mazières; Geoffrey I. Shapiro; Valentina Boni; Saiama N. Waqar; Haeseong Park; David I. Quinn; Alejandro Martinez; Salomon M. Stemmer; Alexis B. Cortot; Fabrice Barlesi; Elisabeth Quoix; Mark E. Burkard; S. Duygu Selcuklu; Casey Hunt; Mark T.A. Donoghue; Mark G. Kris; Judith Bebchuk; Lisa D. Eli; Leanne McCulloch; David B. Solit; Pasi A. Jänne
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International guidelines on the diagnosis and treatment of NUT carcinoma
err2025-07-31
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errOAAI
errYu Zhang; Qi Zhang; Yue Hao; Jia Luo; Yingshi Piao; Wenxian Wang; Zhengbo Song; Ziming Li; Luka Brcic; Aijun Liu; Jinpu Yu; Yasuhiro Tsutani; Wenzhao Zhong; Wenfeng Fang; Zhijie Wang; Shengxiang Ren; Athanasios G. Papavassiliou; Yongchang Zhang; Jingjing Liu; Shirong Zhang; Xiuyu Cai; Ayten Kayi Cangir; Anwen Liu; Wen Li; Filippo Lococo; Ping Zhan; Hongbing Liu; Tangfeng Lv; Liyun Miao; Lingfeng Min; Helmut Popper; Yu Chen; Jingping Yuan; Feng Wang; Zhansheng Jiang; Gen Lin; Long Huang; Xingxiang Pu; Rongbo Lin; Kalevi Kairemo; Weifeng Liu; Chuangzhou Rao; Dongqing Lv; Zongyang Yu; Ashrafian Leanne; Xiaoyan Li; Chuanhao Tang; Hifzur R. Siddique; Chengzhi Zhou; Junping Zhang; Junli Xue; Vishal Shelat; Hui Guo; Qian Chu; Rui Meng; Fatemeh Ardeshir; Jingxun Wu; Rui Zhang; Jin Zhou; Robert A. Kratzke; Zhengfei Zhu; Yongheng Li; Hong Qiu; Fan Xia; Fiorella Calabrese; Yang Xia; Alessandro Wasum Mariani; Yuanyuan Lu; Xiaofeng Chen; Mark A. Klein; Rui Ge; Enyong Dai; Axel H. Schönthal; Yu Han; Zhenying Guo; Jian Zhang; Yinghua Ji; Xianbin Liang; Hongmei Zhang; Xuelei Ma; Marco Chiappetta; Xuewen Liu; Francoise Galateau Salle; Yu Yao; Malgorzata Szolkowska; Weiwei Pan; Fei Pang; Fan Wu; Stefan B. Watzka; Liping Wang; Youcai Zhu; Li Lin; Aparna Sharma; Jianfei Tu; Xinqing Lin; Jing Cai; Ling Xu; Jisheng Li; Xiaodong Jiao; Kainan Li; Marjorie G. Zauderer; Jia Wei; Huijing Feng; Lin Wang; Yingying Du; Wang Yao; Elizabeth Dudnik; Xuefei Shi; Xiaomin Niu; Dongmei Yuan; Yanwen Yao; Jianhui Huang; Yue Feng; Yinbin Zhang; Binbin Song; Wenfeng Li; Jianfei Fu; Marina K. Baine; Pingli Sun; Hong Wang; Mingxiang Ye; Dong Wang; Zhaofeng Wang; Jing Wu; Yunyun Yang; Yuan Fang; Zhen Wang; Bin Wan; Donglai Lv; Huafei Chen; Shengjie Yang; Jing Kang; Jiatao Zhang; Chao Zhang; Lin Shi; Yina Wang; Mohamed Emam Sobeih; Bihui Li; Bin Lian; Lili Mao; Zhang Zhang; Ke Wang; Zhongwu Li; Zhefeng Liu; Nong Yang; Lin Wu; Xiaobing Chen; Gu Jin; Miao Li; Guansong Wang; Thomas U. Marron; Jiandong Wang; Sanjay Popat; Meiyu Fang; Yong Fang; Daniel Mansilla; Yuan Li; Xiaojia Wang; Jing Chen; Yiping Zhang; Xixu Zhu; Yi Shen; Shenglin Ma; Aaron S. Mansfield; Biyun Wang; Lu Si; Anja C. Roden; Bjørn H. Grønberg; Yong Song; Geoffrey I. Shapiro; Christopher A. French; Yuanzhi Lu; Qian Wang; Chunwei Xu
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The RAS-MEK-ERK pathway in low-grade serous ovarian cancer
err2025-07-17
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PREAI
errElizabeth H. Stover; Elizabeth K. Lee; Geoffrey I. Shapiro; Joan S. Brugge; Ursula A. Matulonis; Joyce F. Liu
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Final results from the phase Ia/Ib study of the novel bromodomain and extra-terminal domain inhibitor, BI 894999, in patients with advanced solid tumors or diffuse large B-cell lymphoma
err2025-05-01
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PREAI
errLauer, U. M.; Awada, A.; Postel-Vinay, S.; Shapiro, G. I.; Thieblemont, C.; Piha-Paul, S. A.; Paik, P. K.; Shepard, D. R.; Docampo, L. I.; Galot, R.; Rottey, S.; Sadrolhefazi, B.; Marzin, K.; Musa, H.; Schoffski, P.
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MUC1-C dependency in drug resistant HR+/HER2- breast cancer identifies a new target for antibody-drug conjugate treatment
err2025-04-26
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errOAAI
errNakashoji, Ayako; Bhattacharya, Atrayee; Ozawa, Hiroki; Haratake, Naoki; Shigeta, Keisuke; Fushimi, Atsushi; Yamashita, Nami; Matsui, Akira; Kure, Shoko; Kameyama, Tomoe; Takeuchi, Makoto; Fukuda, Kazumasa; Yokoe, Takamichi; Nagayama, Aiko; Hayahsida, Tetsu; Kitagawa, Yuko; Liu, Renyan; Giordano, Antonio; Jeselsohn, Rinath; Shapiro, Geoffrey I.; Kufe, Donald
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Olaparib in treatment-refractory isocitrate dehydrogenase 1 (IDH1)- and IDH2-mutant cholangiocarcinoma: Safety and antitumor activity from the phase 2 National Cancer Institute 10129 trial
errCANCER
IF5.1
err2025-02-07
err0
PREAI
errCecchini, Michael; Pilat, Mary Jo; Uboha, Nataliya; Azad, Nilofer S.; Cho, May; Davis, Elizabeth J.; Ahnert, Jordi Rodon; Tinoco, Gabriel; Shapiro, Geoffrey I.; Khagi, Simon; Powers, Benjamin; Spencer, Kristen; Groisberg, Roman; Drappatz, Jan; Chen, Li; Das, Biswajit; Bao, Xun; Li, Jing; Narayan, Azeet; Vu, Dennis; Patel, Abhijit; Niger, Monica; Doroshow, Deborah; Durecki, Diane; Boerner, Scott A.; Bindra, Ranjit; Ivy, Percy; Shyr, Derek; Shyr, Yu; Lorusso, Patricia M.
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Hiding in plain sight: NUT carcinoma is an unrecognized subtype of squamous cell carcinoma of the lungs and head and neck
err2025-02-03
err1
PREAI
errLuo, Jia; Bishop, Justin A.; Dubois, Steven G.; Hanna, Glenn J.; Sholl, Lynette M.; Stelow, Edward B.; Thompson, Lester D. R.; Shapiro, Geoffrey I.; French, Christopher A.
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First Results of Migoprotafib, a Potent and Highly Selective Src Homology-2 Domain-Containing Phosphatase 2 Inhibitor in Patients with Advanced Solid Tumors
err2024-12-31
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errOAAI
errJohnson, Melissa L.; Wolf, Beni B.; Wang, Judy S.; Philipovskiy, Alexander; Shapiro, Geoffrey I.; Bockorny, Bruno; Guo, Wei; Shen, Jinshan; Jen, Kai Yu; Lerose, Marybeth; Hunter, Tamieka Lauz; Padval, Mahesh; Schmidt-Kittler, Oleg; Bhatia, Namrata; Dubey, Sarita; Suchomel, Julia; Bendell, Johanna C.; Jauhari, Shekeab; Eng-Wong, Jennifer; Lin, Jessica J.
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PARG inhibitor sensitivity correlates with accumulation of single- stranded DNA gaps in preclinical models of ovarian cancer
err2024-11-15
err0
PREAI
errRavindranathan, Ramya; Somuncu, Ozge; da Costa, Alexandre Andre B. A.; Mukkavalli, Sirisha; Lamarre, Benjamin P.; Nguyen, Huy; Grochala, Carter; Jiao, Yuqing; Liu, Joyce; Kochupurakkal, Bose; Parmar, Kalindi; Shapiro, Geoffrey I.; D'Andrea, Alan D.
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Cyclin D1 Overexpression in Mantle Cell Lymphoma Causes Cellular Dependence on Microhomology-Mediated End-Joining
errBLOOD
IF23.1
err2024-11-05
err0
PREAI
errAbeykoon, Jithma P.; Asada, Shuhei; Zu, Guangli; Hirohashi, Yuna; Iyer, Divya; Parmar, Kalindi; Jiang, Lige; Mukkavalli, Sirisha; Yi, Dongni; Manske, Michelle; Wu, Xiaosheng; Gwin, Kimberly; Witzig, Thomas E.; Shapiro, Geoffrey, I; D'Andrea, Alan D.
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Phase 2 Trial Testing The PARP Inhibitor Niraparib In Patients With Advanced Pancreatic Cancer with Pathogenic Variants In BRCA 1, BRCA2, PALB2, ATM and CHEK2
err2024-09-15
err0
PREAI
errHuffman, Brandon M.; Crowdis, Jett; Yurgelun, Matthew B.; Horick, Nora; Li, Yvonne; Huy Nguyen; Parmar, Kalindi; Kochupurakkal, Bose S.; Enzinger, Andrea; Giannakis, Marios; McCleary, Nadine; Ng, Kimmie; Patel, Anuj K.; Perez, Kimberly J.; Rubinson, Douglas A.; Schlechter, Benjamin L.; Singh, Harshabad; Lam, Helen; Ramsey, Kaitlyn; Andrews, Elizabeth; Culnane, Leigh; Bullock, Andrea; Rattani, Ahmed; Clark, Jeffrey; Peters, Mary Linton; Wolpin, Brian M.; D'Andrea, Alan D.; Shapiro, Geoffrey I.; Aguirre, Andrew J.; Cleary, James M.
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Pre-clinical evaluation of cyclin-dependent kinase 2 and 1 inhibition in anti-estrogen-sensitive and resistant breast cancer cells
err2024-08-19
err0
errOAAI
errJohnson, N.; Bentley, J.; Wang, L-Z; Newell, D. R.; Robson, C. N.; Shapiro, G. I.; Curtin, N. J.
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Single-Stranded DNA Gap Accumulation Is a Functional Biomarker for USP1 Inhibitor Sensitivity
err2024-06-17
err2
errOAAI
errda Costa, Alexandre A.; Somuncu, Ozge; Ravindranathan, Ramya; Mukkavalli, Sirisha; Martignetti, David B.; Nguyen, Huy; Jiao, Yuqing; Lamarre, Benjamin P.; Sadatrezaei, Golbahar; Moreau, Lisa; Liu, Joyce; Iyer, Divya R.; Lazaro, Jean-Bernard; Shapiro, Geoffrey I.; Parmar, Kalindi; D'Andrea, Alan D.
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MUC1-C INTEGRATES CHRONIC ACTIVATION OF INTERFERON PATHWAYS WITH CHROMATIN REMODELING IN TREATMENT RESISTANCE OF TRIPLE-NEGATIVE BREAST CANCER
err2024-05-02
err0
PREAI
errYamashita, Nami; Morimoto, Yoshihiro; Fushimi, Atsushi; Ahmad, Rehan; Bhattacharya, Atrayee; Inoue, Yuka; Withers, Henry; Shapiro, Geoffrey; Yoshizumi, Tomoharu; Ueno, Takayuki; Ohno, Shinji; Long, Mark; Kufe, Donald
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Assessment of Patient-Derived Xenograft Growth and Antitumor Activity: The NCI PDXNet Consensus Recommendations
err2024-04-19
err3
errOAAI
errMeric-Bernstam, Funda; Lloyd, Michael W.; Koc, Soner; Evrard, Yvonne A.; McShane, Lisa M.; Lewis, Michael T.; Evans, Kurt W.; Li, Dali; Rubinstein, Lawrence; Welm, Alana; Dean II, Dennis A.; Srivastava, Anuj; Grover, Jeffrey W.; Ha, Min J.; Chen, Huiqin; Huang, Xuelin; Varadarajan, Kaushik; Wang, Jing; Roth, Jack A.; Welm, Bryan; Govinden, Ramaswamy; Ding, Li; Kaochar, Salma; Mitsiades, Nicholas; Carvajal-Carmona, Luis; Herylyn, Meenhard; Davies, Michael A.; Shapiro, Geoffrey I.; Fields, Ryan; Trevino, Jose G.; Harrell, Joshua C.; Doroshow, James H.; Chuang, Jeffrey H.; Moscow, Jeffrey A.
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