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Marc Nazaré

leibniz-forschungsinstitut für molekulare pharmakologie (fmp)

34H-index
182Paper Count
3.6KCitation Count
Published Papers 80
Publication Date
Probing 3-Amino-2H-Azaindazoles as Allosteric Inhibitors of the Protein Tyrosine Phosphatase SHP2
err2026-06-14
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errMachoud Amoussa; Nina-Louisa Efrém; Feng Li; Ziqiong Guo; Yvette Roske; Katrin Jana Frank; Szymon Pach; Clemens Alexander Wolf; Feng Bo; Marina Lesina; Mika Kintzel; Rana Alsalim; Victoria Zeitz; Noémi Csorba; Silke Radetzki; György M. Keserű; Oliver Daumke; Hana Algül; Gerhard Wolber; Jia Li; Marc Nazaré
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Mapping the SHP2 Allosteric Pocket With Target-Biased Covalent Fragments
err2026-04-24
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errOAAI
errNina-Louisa Efrém; Noémi Csorba; Machoud Amoussa; Péter Ábrányi-Balogh; Ziqiong Guo; László Petri; Feng Bo; Vincenzo Di Lorenzo; Yvette Roske; Tibor Viktor Szalai; Levente Mihalovits; József Simon; Jia Li; Oliver Daumke; György M. Keserű; Marc Nazaré
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Mechanistic Insights into G Protein-Biased κ-Opioid Receptor Signaling Using Dual-Charged Naltrexamine Amides
err2026-02-05
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errNiklas Piet Doering; Kristina Puls; Marta Diceglie; Anja Meraner; Axel Hentsch; Siriwat Hongnak; Armin Wurzer; Helmut Schmidhammer; Mariana Spetea; Marc Nazare; Gerhard Wolber
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Calcium Competitive Inhibition of Langerin by Thiazolopyrimidinones
err2025-11-01
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PREAI
errNing, Yunzhan; Efrem, Nina-Louisa; Amoussa, Machoud; Turhan, Ertan; Zheng, Dazhong; Lefebre, Jonathan; Ruwolt, Max; Neu, Ursula; Besch, Maurice; Loll, Bernhard; Kurzbach, Dennis; Kohnke, Jesko; Nazare, Marc; Rademacher, Christoph
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Front Cover: Inhibition of the Clathrin Terminal Domain—Amphiphysin Protein–Protein Interaction. Probing the Pitstop 2 Aromatic Moiety (ChemMedChem 16/2025)
err2025-08-21
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PREAI
errKate Prichard; Mark J Robertson; Ngoc Chau; Jing Xue; Martin Neuenschwander; Uwe Fink; Andre Horatscheck; Marc Nazare; Phillip J Robinson; Volker Haucke; Adam McCluskey
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Generation of Regulatory T Cells From Human Memory CD4+T Cells by Upregulation of Naked Cuticle Homolog 2
err2025-08-05
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errOAAI
errJiajun He; Kristy Ou; Michael Schmueck-Henneresse; Edgar Specker; Jérôme Paul; Marc Nazare; Jens Peter von Kries; Julia K. Polansky; Alf Hamann; Stefan Frischbutter
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Inhibition of the Clathrin Terminal Domain—Amphiphysin Protein–Protein Interaction. Probing the Pitstop 2 Aromatic Moiety
err2025-07-11
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PREAI
errKate Prichard; Mark J Robertson; Ngoc Chau; Jing Xue; Martin Neuenschwander; Uwe Fink; Andre Horatscheck; Marc Nazare; Phillip J Robinson; Volker Haucke; Adam McCluskey
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A universal cannabinoid CB1 and CB2 receptor TR-FRET kinetic ligand-binding assay
err2025-04-09
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errOAAI
errBorrega-Roman, Leire; Hoare, Bradley L.; Kosar, Miroslav; Sarott, Roman C.; Patej, Kacper J.; Bouma, Jara; Scott-Dennis, Morgan; Koers, Eline J.; Gazzi, Thais; Mach, Leonard; Barrondo, Sergio; Salles, Joan; Guba, Wolfgang; Kusznir, Eric; Nazare, Marc; Rufer, Arne C.; Grether, Uwe; Heitman, Laura H.; Sykes, David A.; Veprintsev, Dmitry B.
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Aminopeptidase-Responsive NIR Photosensitizer for Precision Targeting and Eradication of Pseudomonas aeruginosa Biofilms
err2024-12-23
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PREAI
errLiu, Yang; Liu, Kaixuan; Lei, Ling; Wang, Qinghua; Wang, Xiang; Meng, Xiangchuan; Liu, Qian; Du, Jiacheng; Zhang, Leilei; Nazare, Marc; Hu, Hai-Yu
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Benzo-Crown-Ether Functionalized O-BODIPY Probes for Cations - A Selective Fluorescent Probe for Ba2+
err2024-07-25
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errSprenger, Tobias; Schwarze, Thomas; Holdt, Hans-Juergen; Hentsch, Axel; Nazare, Marc
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Highly Selective Drug-Derived Fluorescent Probes for the Cannabinoid Receptor Type 1 (CB1R)
err2024-07-11
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errOAAI
errMach, Leonard; Omran, Anahid; Bouma, Jara; Radetzki, Silke; Sykes, David A.; Guba, Wolfgang; Li, Xiaoting; Hoeffelmeyer, Calvin; Hentsch, Axel; Gazzi, Thais; Mostinski, Yelena; Wasinska-Kalwa, Malgorzata; de Molnier, Fabio; van der Horst, Cas; von Kries, Jens Peter; Vendrell, Marc; Hua, Tian; Veprintsev, Dmitry B.; Heitman, Laura H.; Grether, Uwe; Nazare, Marc
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Patent review of cannabinoid receptor type 2 (CB2R) modulators (2016-present)
err2024-07-02
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PREAI
errKosar, Miroslav; Mach, Leonard; Carreira, Erick M.; Nazare, Marc; Pacher, Pal; Grether, Uwe
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Novel Tryptophan Hydroxylase Inhibitor TPT-001 Reverses PAH, Vascular Remodeling, and Proliferative-Proinflammatory Gene Expression
err2024-07-01
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errLegchenko, Ekaterina; Chouvarine, Philippe; Qadri, Fatimunnisa; Specker, Edgar; Nazare, Marc; Wesolowski, Radoslaw; Matthes, Susann; Bader, Michael; Hansmann, Georg
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DOTA-Based Plectin-1 Targeted Contrast Agent Enables Detection of Pancreatic Cancer in Human Tissue
err2024-05-24
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errOAAI
errGazzi, Thais; Lesina, Marina; Wang, Qinghua; Berninger, Alexandra; Radetzki, Silke; Demir, Ihsan Ekin; Kohlmann, Larissa; Meiser, Waldemar; Wilke, Sebastian; von Kries, Jens Peter; Alguel, Hana; Hu, Hai-Yu; Nazare, Marc
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Visualization of membrane localization and the functional state of CB2R pools using matched agonist and inverse agonist probe pairs
err2024-01-01
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errOAAI
errWasinska-Kalwa, M.; Omran, A.; Mach, L.; Scipioni, L.; Bouma, J.; Li, X.; Radetzki, S.; Mostinski, Y.; Schippers, M.; Gazzi, T.; van der Horst, C.; Brennecke, B.; Hanske, A.; Kolomeets, Y.; Guba, W.; Sykes, D.; von Kries, J. P.; Broichhagen, J.; Hua, T.; Veprintsev, D.; Heitman, L. H.; Oddi, S.; MacCarrone, M.; Grether, U.; Nazare, M.
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Discovery of tetrazolo-pyridazine-based small molecules as inhibitors of MACC1-driven cancer metastasis
err2023-12-01
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errYan, Shixian; Schoepe, Paul Curtis; Lewis, Joe; Putzker, Kerstin; Uhrig, Ulrike; Specker, Edgar; von Kries, Jens Peter; Lindemann, Peter; Omran, Anahid; Sanchez-Ibarra, Hector E.; Unger, Anke; Zischinsky, Mia-Lisa; Klebl, Bert; Walther, Wolfgang; Nazare, Marc; Kobelt, Dennis; Stein, Ulrike
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Structure-Based Design of Xanthine-Imidazopyridines and -Imidazothiazoles as Highly Potent and In Vivo Efficacious Tryptophan Hydroxylase Inhibitors
err2023-10-31
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PREAI
errSpecker, Edgar; Wesolowski, Radoslaw; Schuetz, Anja; Matthes, Susann; Mallow, Keven; Wasinska-Kalwa, Malgorzata; Winkler, Lars; Oder, Andreas; Alenina, Natalia; Pleimes, Dirk; von Kries, Jens Peter; Heinemann, Udo; Bader, Michael; Nazare, Marc
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Structural Basis for Highly Selective Class II Alpha Phosphoinositide-3-Kinase Inhibition
err2023-10-11
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errKuecuekdisli, Murat; Bel-Abed, Hassen; Cirillo, Davide; Lo, Wen-Ting; Efrem, Nina-Louisa; Horatscheck, Andre; Perepelittchenko, Liudmila; Prokofeva, Polina; Ehret, Theresa A. L.; Radetzki, Silke; Neuenschwander, Martin; Specker, Edgar; Medard, Guillaume; Mueller, Susanne; Wilhelm, Stephanie; Kuster, Bernhard; von Kries, Jens Peter; Haucke, Volker; Nazare, Marc
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CLK2 and CLK4 are regulators of DNA damage-induced NF-kB targeted by novel small molecule inhibitors
err2023-10-01
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errOAAI
errMucka, Patrick; Lindemann, Peter; Bosco, Bartolomeo; Willenbrock, Michael; Radetzki, Silke; Neuenschwander, Martin; Brischetto, Cristina; Kries, Jens Peter von; Nazare, Marc; Scheidereit, Claus
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