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A*Star - Experimental Drug Development Centre (Eddc)

学者数141
论文数79
被引数0
关联论文 (79)
发表时间
Discovery of a potent anti-Zika virus benzamide series targeting the viral protein NS4B发现一种靶向病毒蛋白NS4B的强效抗寨卡病毒苯甲酰胺系列
err2026-04-01
err0
PREAI
errChung, Donghoon; Otsuka, Yuka; Kim, Eunjung; Ullah, Sultan; Kennedy, Nicole M.; Ngo, Khac Huy; Kang, Jinjoo; Tomlinson, Reece; Alejandro, Brian; Barnaby, Koji; Miller, Jeffrey; Shumate, Justin; Teo, Chwee Fang; Tan, Yaw Bia; Chew, Che Shin; Kang, CongBao; Luo, Dahai; Scampavia, Louis; Spicer, Timothy P.; Bannister, Thomas D.
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A Series of Pyrazolo-Quinazoline Amines Inhibits the Cytochrome bd Oxidase in Mycobacterium tuberculosis
err2026-01-01
err0
PREAI
errSingh, Samsher; Ng, Pearly Shuyi; Lakshmanan, Umayal; Mathiyazakan, Vikneswaran; Wiggins, Thomas; Lee, Bei Shi; Ang, Shi Hua; Lin Sim, Sandra Wei; Santos, May Delos; Moraski, Garrett; Miller, Marvin; Berney, Michael; Gruber, Gerhard; Pethe, Kevin
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Reverse phase, ion exchange, HILIC and mix-mode chromatography for the determination of metformin and evogliptin in human plasma and pharmaceutical formulations
err2024-08-01
err1
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errKharabe, Pankaj M.; Jumade, Prasad P.; Khatale, Pravin N.; Katolkar, Parimal P.; Butle, Santosh R.; Kshirsagar, Mahendra D.; Pendharkar, Vishal V.; Sawale, Amol V.; Choudhari, Kalyani S.
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Single-cell landscape of functionally cured chronic hepatitis B patients reveals activation of innate and altered CD4-CTL driven adaptive immunity-功能性治愈的慢性乙型肝炎患者的单细胞景观揭示了先天和改变的CD4-CTL驱动的适应性免疫的激活-
err2024-07-01
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errOAAI
errNarmada, Balakrishnan Chakrapani; Khakpoor, Atefeh; Shirgaonkar, Niranjan; Narayanan, Sriram; Aw, Pauline Poh Kim; Singh, Malay; Ong, Kok Haur; Owino, Collins Oduor; Ng, Jane Wei Ting; Yew, Hui Chuing; Nasir, Nu Soibah Binte Mohamed; Au, Veonice Bijin; Sng, Reina; Kaliaperumal, Nivashini; Khine, Htet Htet Toe Wai; di Tocco, Francesca Casuscelli; Masayuki, Otsuka; Naikar, Shamita; Ng, Hui Xin; Chia, Su Li; Seah, Cindy Xin Yi; Alnawaz, Myra H. J.; Wai, Chris Lee Yoon; Tay, Amy Yuh Ling; Mangat, Kamarjit Singh; Chew, Valerie; Yu, Weimiao; Connolly, John Edward; Periyasamy, Giridharan; Plissonnier, Marie-Laure; Levrero, Massimo; Lim, Seng Gee; DasGupta, Ramanuj
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Cytotoxic activity and cell specificity of a novel LHRH peptide drug conjugate, D-Cys6-LHRH vedotin, against ovarian cancer cell lines
err2024-04-15
err1
PREAI
errVankadara, Subramanyam; Ke, Zhiyuan; Wang, Sifang; Foo, Sin Yun; Gunaratne, Jayantha; Lee, May Ann; Koh, Xiaoying; Chia, C. S. Brian
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GaMF1.39's antibiotic efficacy and its enhanced antitubercular activity in combination with clofazimine, Telacebec, ND-011992, or TBAJ-876
err2023-12-12
err3
errOAAI
errRagunathan, Priya; Shuyi Ng, Pearly; Singh, Samsher; Poh, Wee Han; Litty, Dennis; Kalia, Nitin Pal; Larsson, Simon; Harikishore, Amaravadhi; Rice, Scott A.; Ingham, Philip W.; Mueller, Volker; Moraski, Garrett; Miller, Marvin J.; Dick, Thomas; Pethe, Kevin; Gruber, Gerhard
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RAF1 deficiency causes a lethal syndrome that underscores RTK signaling during embryogenesis
err2023-04-17
err3
errOAAI
errWong, Samantha; Tan, Yu Xuan; Loh, Abigail Yi Ting; Tan, Kiat Yi; Lee, Hane; Aziz, Zainab; Nelson, Stanley F.; Ozkan, Engin; Kayserili, Hülya; Escande-Beillard, Nathalie; Reversade, Bruno
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Trans-interaction of risk loci 6p24.1 and 10q11.21 is associated with endothelial damage in coronary artery disease
err2022-12-01
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errTay, Kai Yi; Wu, Kan Xing; Chioh, Florence Wen Jing; Autio, Matias Ilmari; Pek, Nicole Min Qian; Narmada, Balakrishnan Chakrapani; Tan, Sock-Hwee; Low, Adrian Fatt-Hoe; Lian, Michelle Mulan; Chew, Elaine Guo Yan; Lau, Hwee Hui; Kao, Shih Ling; Teo, Adrian Kee Keong; Foo, Jia Nee; Foo, Roger Sik Yin; Heng, Chew Kiat; Chan, Mark Yan Yee; Cheung, Christine
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Elucidating host cell response pathways and repurposing therapeutics for SARS-CoV-2 and other coronaviruses
err2022-11-05
err3
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errShen, Zhewei; Halberg, Anna; Fong, Jia Yi; Guo, Jingyu; Song, Gavin; Louie, Brent; Luedtke, Gregory R.; Visuthikraisee, Viwat; Protter, Andrew A.; Koh, Xiaoying; Baik, Taegon; Lum, Pek Yee
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Haploinsufficiency of CYP8B1 associates with increased insulin sensitivity in humansCYP8B1的单倍不足与人类胰岛素敏感性增加有关
err2022-11-01
err12
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errZhong, Shiqi; Chevre, Raphael; Mayan, David Castano; Corliano, Maria; Cochran, Blake J.; Sem, Kai Ping; van Dijk, Theo H.; Peng, Jianhe; Tan, Liang Juin; Hartimath, Siddesh V.; Ramasamy, Boominathan; Cheng, Peter; Groen, Albert K.; Kuipers, Folkert; Goggi, Julian L.; Drum, Chester; van Dam, Rob M.; Tan, Ru San; Rye, Kerry-Anne; Hayden, Michael R.; Cheng, Ching-Yu; Chacko, Shaji; Flannick, Jason; Sim, Xueling; Tan, Hong Chang; Singaraja, Roshni R.
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Variable-heavy (VH) families influencing IgA1&2 engagement to the antigen, FcαRI and superantigen proteins G, A, and L
err2022-04-20
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errLing, Wei-Li; Su, Chinh Tran-To; Lua, Wai-Heng; Yeo, Joshua Yi; Poh, Jun-Jie; Ng, Yuen-Ling; Wipat, Anil; Gan, Samuel Ken-En
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More Than Meets the Kappa for Antibody Superantigen Protein L (PpL)
err2022-02-11
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errOAAI
errLing, Wei-Li; Yeo, Joshua Yi; Ng, Yuen-Ling; Wipat, Anil; Gan, Samuel Ken-En
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Structural model of human PORCN illuminates disease-associated variants and drug-binding sites
err2021-12-20
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errYu, Jia; Liao, Pei-Ju; Xu, Weijun; Jones, Julie R.; Everman, David B.; Flanagan-Steet, Heather; Keller, Thomas H.; Virshup, David M.
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Update on the Development of MNK Inhibitors as Therapeutic Agents
err2021-09-17
err33
PREAI
errXu, Weijun; Kannan, Srinivasaraghavan; Verma, Chandra S.; Nacro, Kassoum
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Spectrophotometer on-the-go: The development of a 2-in-1 UV-Vis portable Arduino-based spectrophotometer
err2021-07-01
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PREAI
errPoh, Jun-Jie; Wu, Wei-Ling; Goh, Nicholas Wei-Jie; Tan, Samuel Ming-Xuan; Gan, Samuel Ken-En
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Strategic Design of Catalytic Lysine-Targeting Reversible Covalent BCR-ABL Inhibitors催化赖氨酸靶向可逆共价bcr-abl抑制剂的策略设计
err2021-06-24
err56
PREAI
errQuach, David; Tang, Guanghui; Anantharajan, Jothi; Baburajendran, Nithya; Poulsen, Anders; Wee, John L. K.; Retna, Priya; Li, Rong; Liu, Boping; Tee, Doris H. Y.; Kwek, Perlyn Z.; Joy, Joma K.; Yang, Wan-Qi; Zhang, Chong-Jing; Foo, Klement; Keller, Thomas H.; Yao, Shao Q.
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Design and Development of a Low Cost, Non-Contact Infrared Thermometer with Range Compensation
errSENSORS
IF3.5
err2021-05-31
err15
errOAAI
errGoh, Nicholas Wei-Jie; Poh, Jun-Jie; Yeo, Joshua Yi; Aw, Benjamin Jun-Jie; Lai, Szu Cheng; Cheng, Jayce Jian Wei; Tan, Christina Yuan Ling; Gan, Samuel Ken-En
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Engineered NS1 for Sensitive, Specific Zika Virus Diagnosis from Patient Serology
err2021-05-01
err8
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errYap, Thai Leong; Hong, Shin Yee; Soh, Jun Hui; Ravichandraprabhu, Lekha; Lim, Vanessa W. X.; Chan, Hsi-Min; Ong, Tommy Z. X.; Chua, Ying Ping; Koh, Shi En; Wang, Huajing; Leo, Yee Sin; Ying, Jackie Y.; Sun, William
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