未登录Discovery of a potent anti-Zika virus benzamide series targeting the viral protein NS4B发现一种靶向病毒蛋白NS4B的强效抗寨卡病毒苯甲酰胺系列
Chung, Donghoon; Otsuka, Yuka; Kim, Eunjung; Ullah, Sultan; Kennedy, Nicole M.; Ngo, Khac Huy; Kang, Jinjoo; Tomlinson, Reece; Alejandro, Brian; Barnaby, Koji; Miller, Jeffrey; Shumate, Justin; Teo, Chwee Fang; Tan, Yaw Bia; Chew, Che Shin; Kang, CongBao; Luo, Dahai; Scampavia, Louis; Spicer, Timothy P.; Bannister, Thomas D.
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收藏A Series of Pyrazolo-Quinazoline Amines Inhibits the Cytochrome bd Oxidase in Mycobacterium tuberculosis
Singh, Samsher; Ng, Pearly Shuyi; Lakshmanan, Umayal; Mathiyazakan, Vikneswaran; Wiggins, Thomas; Lee, Bei Shi; Ang, Shi Hua; Lin Sim, Sandra Wei; Santos, May Delos; Moraski, Garrett; Miller, Marvin; Berney, Michael; Gruber, Gerhard; Pethe, Kevin
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收藏Reverse phase, ion exchange, HILIC and mix-mode chromatography for the determination of metformin and evogliptin in human plasma and pharmaceutical formulations
Kharabe, Pankaj M.; Jumade, Prasad P.; Khatale, Pravin N.; Katolkar, Parimal P.; Butle, Santosh R.; Kshirsagar, Mahendra D.; Pendharkar, Vishal V.; Sawale, Amol V.; Choudhari, Kalyani S.
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收藏Single-cell landscape of functionally cured chronic hepatitis B patients reveals activation of innate and altered CD4-CTL driven adaptive immunity-功能性治愈的慢性乙型肝炎患者的单细胞景观揭示了先天和改变的CD4-CTL驱动的适应性免疫的激活-
Narmada, Balakrishnan Chakrapani; Khakpoor, Atefeh; Shirgaonkar, Niranjan; Narayanan, Sriram; Aw, Pauline Poh Kim; Singh, Malay; Ong, Kok Haur; Owino, Collins Oduor; Ng, Jane Wei Ting; Yew, Hui Chuing; Nasir, Nu Soibah Binte Mohamed; Au, Veonice Bijin; Sng, Reina; Kaliaperumal, Nivashini; Khine, Htet Htet Toe Wai; di Tocco, Francesca Casuscelli; Masayuki, Otsuka; Naikar, Shamita; Ng, Hui Xin; Chia, Su Li; Seah, Cindy Xin Yi; Alnawaz, Myra H. J.; Wai, Chris Lee Yoon; Tay, Amy Yuh Ling; Mangat, Kamarjit Singh; Chew, Valerie; Yu, Weimiao; Connolly, John Edward; Periyasamy, Giridharan; Plissonnier, Marie-Laure; Levrero, Massimo; Lim, Seng Gee; DasGupta, Ramanuj
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收藏Cytotoxic activity and cell specificity of a novel LHRH peptide drug conjugate, D-Cys6-LHRH vedotin, against ovarian cancer cell lines
Vankadara, Subramanyam; Ke, Zhiyuan; Wang, Sifang; Foo, Sin Yun; Gunaratne, Jayantha; Lee, May Ann; Koh, Xiaoying; Chia, C. S. Brian
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收藏Regio-MPNN: predicting regioselectivity for general metal-catalyzed cross-coupling reactions using a chemical knowledge informed message passing neural networkRegio-mpnn: 使用化学知识信息传递神经网络预测一般金属催化交叉偶联反应的区域选择性
Li, Baochen; Liu, Yuru; Sun, Haibin; Zhang, Rentao; Xie, Yongli; Foo, Klement; Mak, Frankie S.; Zhang, Ruimao; Yu, Tianshu; Lin, Sen; Wang, Peng; Wang, Xiaoxue
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收藏GaMF1.39's antibiotic efficacy and its enhanced antitubercular activity in combination with clofazimine, Telacebec, ND-011992, or TBAJ-876
Ragunathan, Priya; Shuyi Ng, Pearly; Singh, Samsher; Poh, Wee Han; Litty, Dennis; Kalia, Nitin Pal; Larsson, Simon; Harikishore, Amaravadhi; Rice, Scott A.; Ingham, Philip W.; Mueller, Volker; Moraski, Garrett; Miller, Marvin J.; Dick, Thomas; Pethe, Kevin; Gruber, Gerhard
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收藏RAF1 deficiency causes a lethal syndrome that underscores RTK signaling during embryogenesis
Wong, Samantha; Tan, Yu Xuan; Loh, Abigail Yi Ting; Tan, Kiat Yi; Lee, Hane; Aziz, Zainab; Nelson, Stanley F.; Ozkan, Engin; Kayserili, Hülya; Escande-Beillard, Nathalie; Reversade, Bruno
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收藏Trans-interaction of risk loci 6p24.1 and 10q11.21 is associated with endothelial damage in coronary artery disease
Tay, Kai Yi; Wu, Kan Xing; Chioh, Florence Wen Jing; Autio, Matias Ilmari; Pek, Nicole Min Qian; Narmada, Balakrishnan Chakrapani; Tan, Sock-Hwee; Low, Adrian Fatt-Hoe; Lian, Michelle Mulan; Chew, Elaine Guo Yan; Lau, Hwee Hui; Kao, Shih Ling; Teo, Adrian Kee Keong; Foo, Jia Nee; Foo, Roger Sik Yin; Heng, Chew Kiat; Chan, Mark Yan Yee; Cheung, Christine
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收藏Elucidating host cell response pathways and repurposing therapeutics for SARS-CoV-2 and other coronaviruses
Shen, Zhewei; Halberg, Anna; Fong, Jia Yi; Guo, Jingyu; Song, Gavin; Louie, Brent; Luedtke, Gregory R.; Visuthikraisee, Viwat; Protter, Andrew A.; Koh, Xiaoying; Baik, Taegon; Lum, Pek Yee
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收藏Haploinsufficiency of CYP8B1 associates with increased insulin sensitivity in humansCYP8B1的单倍不足与人类胰岛素敏感性增加有关
Zhong, Shiqi; Chevre, Raphael; Mayan, David Castano; Corliano, Maria; Cochran, Blake J.; Sem, Kai Ping; van Dijk, Theo H.; Peng, Jianhe; Tan, Liang Juin; Hartimath, Siddesh V.; Ramasamy, Boominathan; Cheng, Peter; Groen, Albert K.; Kuipers, Folkert; Goggi, Julian L.; Drum, Chester; van Dam, Rob M.; Tan, Ru San; Rye, Kerry-Anne; Hayden, Michael R.; Cheng, Ching-Yu; Chacko, Shaji; Flannick, Jason; Sim, Xueling; Tan, Hong Chang; Singaraja, Roshni R.
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收藏Variable-heavy (VH) families influencing IgA1&2 engagement to the antigen, FcαRI and superantigen proteins G, A, and L
Ling, Wei-Li; Su, Chinh Tran-To; Lua, Wai-Heng; Yeo, Joshua Yi; Poh, Jun-Jie; Ng, Yuen-Ling; Wipat, Anil; Gan, Samuel Ken-En
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收藏Strategic Design of Catalytic Lysine-Targeting Reversible Covalent BCR-ABL Inhibitors催化赖氨酸靶向可逆共价bcr-abl抑制剂的策略设计
Quach, David; Tang, Guanghui; Anantharajan, Jothi; Baburajendran, Nithya; Poulsen, Anders; Wee, John L. K.; Retna, Priya; Li, Rong; Liu, Boping; Tee, Doris H. Y.; Kwek, Perlyn Z.; Joy, Joma K.; Yang, Wan-Qi; Zhang, Chong-Jing; Foo, Klement; Keller, Thomas H.; Yao, Shao Q.
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收藏Engineered NS1 for Sensitive, Specific Zika Virus Diagnosis from Patient Serology
Yap, Thai Leong; Hong, Shin Yee; Soh, Jun Hui; Ravichandraprabhu, Lekha; Lim, Vanessa W. X.; Chan, Hsi-Min; Ong, Tommy Z. X.; Chua, Ying Ping; Koh, Shi En; Wang, Huajing; Leo, Yee Sin; Ying, Jackie Y.; Sun, William
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