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Compound PZ-1262, a 4-isoquinoline-sulfonamide analog of Brexpiprazole, produces potential antidepressant, anxiolytic and procognitive effects in rodent models Partyka, Anna; Golebiowska, Joanna; Marciniec, Krzysztof; Canale, Vittorio; Trybala, Wojciech; Satala, Grzegorza; Grychowska, Katarzyna; Jastrzebska-Wiesek, Magdalena; Bojarski, Andrzej J.; Nikiforuk, Agnieszka; Daniel, Wladyslawa A.; Wesolowska, Anna; Zajdel, Pawel; Popik, Piotr 分享 收藏
Simultaneous 5-HT1BR agonist/5-HT6R antagonist action as a potential treatment of Parkinson's disease and its comorbidities Zajdel, Pawe l; Matloka, Mikolaj; Konieczny, Jolanta; Kos, Tomasz; Lammers, Josie C.; Cavalco, Natalie G.; Clark, Allison A.; Lenda, Tomasz; Satala, Grzegorz; Canale, Vittorio; Grychowska, Katarzyna; Krawczyk, Martyna; Nikiforuk, Agnieszka; Partyka, Anna; Jastrzebska-Wiesek, Magdalena; Berghauzen-Maciejewska, Klemencja; Biala, Dominika; Janicka, Monika; Janusz, Artur; Piast, Radoslaw; Mulewski, Krzysztof; Smuga, Damian; Pieczykolan, Jerzy; Wieczorek, Maciej; Moszczynski-Petkowski, Rafal; Dubiel, Krzysztof; Ossowska, Krystyna; Bojarski, Andrzej J.; Kaminski, Krzysztof; Mccorvy, John D.; Popik, Piotr 分享 收藏
Unraveling psilocybin's therapeutic potential: behavioral and neuroplasticity insights in Wistar-Kyoto and Wistar male rat models of treatment-resistant depression (Jul, 10.1007/s00213-024-06644-3, 2024) Kolasa, Magdalena; Nikiforuk, Agnieszka; Korlatowicz, Agata; Solich, Joanna; Potasiewicz, Agnieszka; Dziedzicka-Wasylewska, Marta; Bugno, Ryszard; Hogendorf, Adam; Bojarski, Andrzej; Faron-Gorecka, Agata 分享 收藏
Unraveling psilocybin's therapeutic potential: behavioral and neuroplasticity insights in Wistar-Kyoto and Wistar male rat models of treatment-resistant depression Magdalena, Kolasa; Agnieszka, Nikiforuk; Agata, Korlatowicz; Joanna, Solich; Agnieszka, Potasiewicz; Dziedzicka-Wasylewska, Marta; Ryszard, Bugno; Adam, Hogendorf; Andrzej, Bojarski; Agata, Faron-Gorecka 分享 收藏
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Impact of the Substitution Pattern at the Basic Center and Geometry of the Amine Fragment on 5-HT6 and D3R Affinity in the 1H-Pyrrolo[3,2-c]quinoline Series Grychowska, Katarzyna; Pietrus, Wojciech; Kulawik, Ludmila; Bento, Ophelie; Satala, Grzegorz; Bantreil, Xavier; Lamaty, Frederic; Bojarski, Andrzej J.; Golebiowska, Joanna; Nikiforuk, Agnieszka; Marin, Philippe; Chaumont-Dubel, Severine; Kurczab, Rafal; Zajdel, Pawel 分享 收藏
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Effects of ketamine optical isomers, psilocybin, psilocin and norpsilocin on time estimation and cognition in rats Popik, Piotr; Hogendorf, Adam; Bugno, Ryszard; Khoo, Shaun Yon-Seng; Zajdel, Pawel; Malikowska-Racia, Natalia; Nikiforuk, Agnieszka; Golebiowska, Joanna 分享 收藏
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Structure-Based Design and Optimization of FPPQ, a Dual-Acting 5-HT3 and 5-HT6 Receptor Antagonist with Antipsychotic and Procognitive Properties Zajdel, Pawel; Grychowska, Katarzyna; Mogilski, Szczepan; Kurczab, Rafal; Satala, Grzegorz; Bugno, Ryszard; Kos, Tomasz; Golebiowska, Joanna; Malikowska-Racia, Natalia; Nikiforuk, Agnieszka; Chaumont-Dubel, Severine; Bantreil, Xavier; Pawlowski, Maciej; Martinez, Jean; Subra, Gilles; Lamaty, Frederic; Marin, Philippe; Bojarski, Andrzej J.; Popik, Piotr 分享 收藏
2-Phenyl-1H-pyrrole-3-carboxamide as a New Scaffold for Developing 5-HT6 Receptor Inverse Agonists with Cognition-Enhancing Activity 2-苯基-1h-吡咯-3-甲酰胺作为开发具有认知增强活性的5-HT6受体反向激动剂的新支架 Drop, Marcin; Canale, Vittorio; Chaumont-Dubel, Severine; Kurczab, Rafal; Satala, Grzegorz; Bantreil, Xavier; Walczak, Maria; Koczurkiewicz-Adamczyk, Paulina; Latacz, Gniewomir; Gwizdak, Anna; Krawczyk, Martyna; Golebiowska, Joanna; Grychowska, Katarzyna; Bojarski, Andrzej J.; Nikiforuk, Agnieszka; Subra, Gilles; Martinez, Jean; Pawlowski, Maciej; Popik, Piotr; Marin, Philippe; Lamaty, Frederic; Zajdel, Pawel 分享 收藏
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