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骆衡 封面图

骆衡 (Heng Luo)

Gannan Medical University

34H指数
130论文数
5.2K被引数
收录论文 49
发表时间
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Learning motif-based graphs for drug-drug interaction prediction via local-global self-attention通过局部全局自我注意学习基于motif的药物-药物相互作用预测图
err2024-08-27
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PREAI
errZhong, Yi; Li, Gaozheng; Yang, Ji; Zheng, Houbing; Yu, Yongqiang; Zhang, Jiheng; Luo, Heng; Wang, Biao; Weng, Zuquan
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Borane-Catalyzed Asymmetric Reduction of 2-Alkylpyridines
err2024-08-08
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errOAAI
errLuo, Heng; Yang, Zhao-Ying; Zhang, Ming; Wang, Xiao-Chen
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Novel antimicrobial peptides against Cutibacterium acnes designed by deep learning
err2024-02-24
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errOAAI
errDong, Qichang; Wang, Shaohua; Miao, Ying; Luo, Heng; Weng, Zuquan; Yu, Lun
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Dual target PARP1/EZH2 inhibitors inducing excessive autophagy and producing synthetic lethality for triple-negative breast cancer therapy
err2024-02-01
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PREAI
errLi, Xinxin; Wang, Cheng; Li, Shang; Yin, Fucheng; Luo, Heng; Zhang, Yonglei; Luo, Zhongwen; Chen, Yifan; Wan, Siyuan; Kong, Lingyi; Wang, Xiaobing
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Indirubin derivatives as bifunctional molecules inducing DNA damage and targeting PARP for the treatment of cancer
err2023-12-01
err5
PREAI
errWan, Siyuan; Chen, Xinye; Yin, Fucheng; Li, Shang; Zhang, Yonglei; Luo, Heng; Luo, Zhongwen; Cui, Ningjie; Chen, Yifan; Li, Xinxin; Kong, Lingyi; Wang, Xiaobing
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Design, synthesis and mechanism studies of dual EZH2/BRD4 inhibitors for cancer therapy
err2023-08-01
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PREAI
errChen, Xinye; Wang, Cheng; Lu, Dehua; Luo, Heng; Li, Shang; Yin, Fucheng; Luo, Zhongwen; Cui, Ningjie; Kong, Lingyi; Wang, Xiaobing
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Oxazole-4-carboxamide/butylated hydroxytoluene hybrids with GSK-3β inhibitory and neuroprotective activities against Alzheimer's disease
err2023-08-01
err9
PREAI
errLuo, Zhongwen; Li, Shang; Zhang, Yonglei; Yin, Fucheng; Luo, Heng; Chen, Xinye; Cui, Ningjie; Wan, Siyuan; Li, Xinxin; Kong, Lingyi; Wang, Xiaobing
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C3-Cyanation of Pyridines: Constraints on Electrophiles and Determinants of Regioselectivity
err2023-01-09
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PREAI
errZhang, Ming; Zhou, Qingyang; Luo, Heng; Tang, Zi-Lu; Xu, Xiufang; Wang, Xiao-Chen
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Histone Deacetylase and Enhancer of Zeste Homologue 2 Dual Inhibitors Presenting a Synergistic Effect for the Treatment of Hematological Malignancies
err2022-09-25
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PREAI
errLu, Dehua; Wang, Cheng; Qu, Lailiang; Yin, Fucheng; Li, Shang; Luo, Heng; Zhang, Yonglei; Liu, Xingchen; Chen, Xinye; Luo, Zhongwen; Cui, Ningjie; Kong, Lingyi; Wang, Xiaobing
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Discovery of precision targeting EZH2 degraders for triple-negative breast cancer发现针对三阴性乳腺癌的精确靶向EZH2降解剂
err2022-08-01
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PREAI
errWang, Cheng; Chen, Xinye; Liu, Xingchen; Lu, Dehua; Li, Shang; Qu, Lailiang; Yin, Fucheng; Luo, Heng; Zhang, Yonglei; Luo, Zhongwen; Cui, Ningjie; Kong, Lingyi; Wang, Xiaobing
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Discovery of PT-65 as a highly potent and selective Proteolysis-targeting chimera degrader of GSK3 for treating Alzheimer's disease
err2021-12-01
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PREAI
errQu, Lailiang; Li, Shang; Ji, Limei; Luo, Si; Ding, Ming; Yin, Fucheng; Wang, Cheng; Luo, Heng; Lu, Dehua; Liu, Xingchen; Peng, Wan; Kong, Lingyi; Wang, Xiaobing
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Parthenolide Derivatives as PKM2 Activators Showing Potential in Colorectal Cancer
err2021-12-01
err19
PREAI
errLiu, Xingchen; Wang, Cheng; Li, Shang; Qu, Lailiang; Yin, Fucheng; Lu, Dehua; Luo, Heng; Chen, Xinye; Luo, Zhongwen; Cui, Ningjie; Wang, Xiaobing; Kong, Lingyi
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Borane-Catalyzed Reduction of Pyridines via a Hydroboration/Hydrogenation Cascade
err2021-08-17
err18
PREAI
errYang, Zhao-Ying; Luo, Heng; Zhang, Ming; Wang, Xiao-Chen
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研究方向

DNA-bindingDNA unwindingATPase activitiesBloom helicase分子机制Bloom解旋酶催化核心与双链DNA相互作用新型N,N-二取代席夫碱的合成及其体外抗菌和抗肿瘤活性评价药物化学抗菌抗肿瘤活性苯甲醛席夫碱的抗菌活性及其构效关系bacteria inhibitors齐墩果酸衍生物微生物活性构效关系鞣花烷型三萜类化合物的提取与细胞毒性miR-34b通过调控TGF-β通路抑制前列腺癌细胞迁移与侵袭miR-17-92基因簇在肿瘤细胞中的表达、调控和作用机制黄酮类醚类化合物抗癌活性新型L型邻苯醌类似物的细胞毒性机制研究通过靶向启动子活性调控Fli-1激活抑制前列腺癌细胞生长和转移的新型3',5'-二异戊烯基查尔酮研究丹参酮类似物抗癌机制前列腺癌细胞凋亡焦亡机制PKCδ/JNK信号通路基于天然产物库的筛选靶向HIV-1衣壳C端结构域2的抑制剂含硒药物ebselen靶向LEDGF/p75破坏其与HIV-1整合酶的相互作用reproductive toxicity in zebrafish紫穗槐中atisine型二萜生物碱的抗TMV活性G4DNA structureProstate cancer cells抗癌药物设计IL-24在肿瘤发生发展中的作用静电纺丝制备PBAT空心多孔微纤维及其功能化用于多肽释放超分子化学发光材料葫芦[8]脲超分子组装室温磷光体系L-苯丙氨酸二肽通过靶向TNFSF9、CYR61和c-Jun抑制前列腺癌细胞增殖antitumor drug development微核糖核酸-451肾脏功能前列腺癌细胞生长抑制