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收藏Exploration of (R)-[11C]YH168 as a PET tracer for imaging monoacylglycerol lipase in the brain: from mice to non-human primates
He, Yingfang; Zheng, Mingqiang; Gu, Jiwei; Reichert, Lisa; Trimborn, Johannes; Zhang, Hui; Keller, Claudia; Crosby, Mallory; Collin, Ludovic; Heer, Dominik; Pavlovic, Anto; Topp, Andreas; Wittwer, Matthias Beat; Grether, Uwe; Gobbi, Luca; Schibli, Roger; Huang, Yiyun; Mu, Linjing
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收藏Preclinical evaluation and pilot clinical study of [68Ga]Ga-NOTA-H006 for non-invasive PET imaging of 5T4 oncofetal antigen
He, Yingfang; Tian, Ruhua; Xu, Dong; Wu, Yanfei; Rina, Sa; Chen, Tengxiang; Guan, Yihui; Xie, Tianwu; Ying, Tianlei; Xie, Fang; Han, Junbin
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收藏Development of radiofluorinated MLN-4760 derivatives for PET imaging of the SARS-CoV-2 entry receptor ACE2
Wang, Jinling; Beyer, Darja; Vaccarin, Christian; He, Yingfang; Tanriver, Matthias; Benoit, Roger; Deupi, Xavier; Mu, Linjing; Bode, Jeffrey W.; Schibli, Roger; Mueller, Cristina
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收藏Metabotropic glutamate receptor 5 (mGluR5) is associated with neurodegeneration and amyloid deposition in Alzheimer's disease: A [18F]PSS232 PET/MRI study
Wang, Jie; He, Yingfang; Chen, Xing; Huang, Lin; Li, Junpeng; You, Zhiwen; Huang, Qi; Ren, Shuhua; He, Kun; Schibli, Roger; Mu, Linjing; Guan, Yihui; Guo, Qihao; Zhao, Jun; Xie, Fang
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收藏Identification of (R)-[18F]YH134 for Monoacylglycerol Lipase Neuroimaging and Exploration of Its Use for Central Nervous System and Peripheral Drug Development
He, Yingfang; Kramer, Stefanie D.; Grether, Uwe; Wittwer, Matthias B.; Collin, Ludovic; Kuhn, Bernd; Topp, Andreas; Heer, Dominik; O'Hara, Fionn; Honer, Michael; Pavlovic, Anto; Richter, Hans; Ritter, Martin; Rombach, Didier; Keller, Claudia; Gobbi, Luca; Mu, Linjing
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收藏Multi-parameter optimization: Development of a morpholin-3-one derivative with an improved kinetic profile for imaging monoacylglycerol lipase in the brain
He, Yingfang; Grether, Uwe; Taddio, Marco F.; Meier, Carla; Keller, Claudia; Edelmann, Martin R.; Honer, Michael; Huber, Sylwia; Wittwer, Matthias B.; Heer, Dominik; Richter, Hans; Collin, Ludovic; Hug, Melanie N.; Hilbert, Manuel; Postmus, Annemarieke G. J.; Stevens, Anna Floor; Van der Stelt, Mario; Kramer, Stefanie D.; Schibli, Roger; Mu, Linjing; Gobbi, Luca C.
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收藏Discovery, synthesis and evaluation of novel reversible monoacylglycerol lipase radioligands bearing a morpholine-3-one scaffold
He, Yingfang; Gobbi, Luca C.; Herde, Adrienne Mueller; Rombach, Didier; Ritter, Martin; Kuhn, Bernd; Wittwer, Matthias B.; Heer, Dominik; Hornsperger, Benoit; Bell, Charles; O'Hara, Fionn; Benz, Jorg; Honer, Michael; Keller, Claudia; Collin, Ludovic; Richter, Hans; Schibli, Roger; Grether, Uwe; Mu, Linjing
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收藏Development of High Brain-Penetrant and Reversible Monoacylglycerol Lipase PET Tracers for Neuroimaging
He, Yingfang; Schild, Matthias; Grether, Uwe; Benz, Jorg; Leibrock, Lea; Heer, Dominik; Topp, Andreas; Collin, Ludovic; Kuhn, Bernd; Wittwer, Matthias; Keller, Claudia; Gobbi, Luca C.; Schibli, Roger; Mu, Linjing
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收藏Synthesis and evaluation of new 1-oxa-8-azaspiro [4.5] decane derivatives as candidate radioligands for sigma-1 receptors
Tian, Jiale; He, Yingfang; Deuther-Conrad, Winnie; Fu, Hualong; Xie, Fang; Zhang, Ying; Wang, Tao; Zhang, Xiaojun; Zhang, Jinming; Brust, Peter; Huang, Yiyun; Jia, Hongmei
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收藏Positron Emission Tomography Imaging Evaluation of a Novel 18F-Labeled Sigma-1 Receptor Radioligand in Cynomolgus Monkeys食蟹猴中新型18f标记的Sigma-1受体放射性配体的正电子发射断层扫描成像评估
Jia, Hongmei; Cai, Zhengxin; Holden, Daniel; He, Yingfang; Lin, Shu-fei; Li, Songye; Baum, Evan; Shirali, Anupama; Kapinos, Michael; Gao, Hong; Ropchan, Jim; Huang, Yiyun
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收藏18F-Labeled indole-based analogs as highly selective radioligands for imaging sigma-2 receptors in the brain
Wang, Liang; Ye, Jiajun; He, Yingfang; Deuther-Conrad, Winnie; Zhang, Jinming; Zhang, Xiaojun; Cui, Mengchao; Steinbach, Joerg; Huang, Yiyun; Brust, Peter; Jia, Hongmei
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收藏1-(4-[18F]Fluorobenzyl)-4-[(tetrahydrofuran-2-yl)methyl]piperazine: A Novel Suitable Radioligand with Low Lipophilicity for Imaging σ1 Receptors in the Brain
He, Yingfang; Xie, Fang; Ye, Jiajun; Deuther-Conrad, Winnie; Cui, Bixiao; Wang, Liang; Lu, Jie; Steinbach, Jorg; Brust, Peter; Huang, Yiyun; Lu, Jie; Jia, Hongmei
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