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Virtual screening-guided repurposing of fluorescent probes to detect EGFR expression in renal cells 虚拟筛选指导的荧光探针再利用以检测肾细胞中EGFR表达 Graziano, Giovanni; Trisciuzzi, Daniela; Contino, Marialessandra; Stasi, Alessandra; Laghezza, Antonio; Cimmarusti, Maria Teresa; Campioni, Monica; Mammone, Mariachiara; Fanizzi, Annalisa; Degennaro, Pasquale; Mastrofilippo, Nicola; Fiorentino, Marco; Pontrelli, Paola; Stefanachi, Angela; Colabufo, Nicola Antonio; Gesualdo, Loreto; Nicolotti, Orazio 分享 收藏
First-In-Class Thiosemicarbazone Metal Complexes Targeting the Sigma-2 Receptor (S2R) as an Innovative Strategy against Pancreatic Cancer (vol 67, pg 20118, 2024) 靶向Sigma-2受体(S2R)的第一类硫代半卡巴腙金属配合物作为对抗胰腺癌的创新策略(vol 67, pg 20118, 2024) Barbanente, Alessandra; Kopecka, Joanna; Vitone, Daniele; Niso, Mauro; Rizzi, Rosanna; Cuocci, Corrado; Abatematteo, Francesca Serena; Mastropasqua, Francesco; Colabufo, Nicola Antonio; Margiotta, Nicola; Arnesano, Fabio; Riganti, Chiara; Abate, Carmen 分享 收藏
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First-In-Class Thiosemicarbazone Metal Complexes Targeting the Sigma-2 Receptor (S2R) as an Innovative Strategy against Pancreatic Cancer Barbanente, Alessandra; Kopecka, Joanna; Vitone, Daniele; Niso, Mauro; Rizzi, Rosanna; Cuocci, Corrado; Abatematteo, Francesca Serena; Mastropasqua, Francesco; Colabufo, Nicola Antonio; Margiotta, Nicola; Arnesano, Fabio; Riganti, Chiara; Abate, Carmen 分享 收藏
Dual Inhibitors of P-gp and Carbonic Anhydrase XII (hCA XII) against Tumor Multidrug Resistance with Piperazine Scaffold Braconi, Laura; Riganti, Chiara; Parenti, Astrid; Cecchi, Marta; Nocentini, Alessio; Bartolucci, Gianluca; Menicatti, Marta; Contino, Marialessandra; Colabufo, Nicola Antonio; Manetti, Dina; Romanelli, Maria Novella; Supuran, Claudiu T.; Teodori, Elisabetta 分享 收藏
N-Adamantyl-1-alkyl-4-oxo-1,4-dihydroquinoline-3-carboxamide Derivatives as Fluorescent Probes to Detect Microglia Activation through the Imaging of Cannabinoid Receptor Subtype 2 (CB2R) Intranuovo, Francesca; Majellaro, Maria; Mastropasqua, Francesco; Delre, Pietro; Abatematteo, Francesca Serena; Mangiatordi, Giuseppe Felice; Stefanachi, Angela; Brea, Jose; Loza, Maria Isabel; Riganti, Chiara; Ligresti, Alessia; Kumar, Poulami; Esposito, Daniela; Cristino, Luigia; Nicois, Alessandro; Gonzalez, Lucia; Perrone, Maria Grazia; Colabufo, Nicola Antonio; Sotelo, Eddy; Abate, Carmen; Contino, Marialessandra 分享 收藏
Nature-Inspired 1-Phenylpyrrolo[2,1-a]isoquinoline Scaffold for Novel Antiproliferative Agents Circumventing P-Glycoprotein-Dependent Multidrug Resistance Nevskaya, Alisa A.; Purgatorio, Rosa; Borisova, Tatiana N.; Varlamov, Alexey V.; Anikina, Lada V.; Obydennik, Arina Yu.; Nevskaya, Elena Yu.; Niso, Mauro; Colabufo, Nicola A.; Carrieri, Antonio; Catto, Marco; de Candia, Modesto; Voskressensky, Leonid G.; Altomare, Cosimo D. 分享 收藏
A scalable route to quaternary ammonium-functionalized AgCl colloidal antimicrobials inhibiting food pathogenic bacteria and biofilms Bajrami, Diellza; Hossain, Syed Imdadul; Barbarossa, Alexia; Sportelli, Maria Chiara; Picca, Rosaria Anna; Gentile, Luigi; Mastrolonardo, Francesco; Rosato, Antonio; Carocci, Alessia; Colabufo, Nicola Antonio; Mizaikoff, Boris; Cioffi, Nicola 分享 收藏
Tetrazole and oxadiazole derivatives as bioisosteres of tariquidar and elacridar: New potent P-gp modulators acting as MDR reversers Braconi, Laura; Dei, Silvia; Contino, Marialessandra; Riganti, Chiara; Bartolucci, Gianluca; Manetti, Dina; Romanelli, Maria Novella; Perrone, Maria Grazia; Colabufo, Nicola Antonio; Guglielmo, Stefano; Teodori, Elisabetta 分享 收藏
A conformational rearrangement of the SARS-CoV-2 host protein sigma-1 is required for antiviral activity: insights from a combined in-silico/in-vitro approach Abatematteo, Francesca Serena; Delre, Pietro; Mercurio, Ivan; Rezelj, Veronica V. V.; Siliqi, Dritan; Beaucourt, Stephanie; Lattanzi, Gianluca; Colabufo, Nicola Antonio; Leopoldo, Marcello; Saviano, Michele; Vignuzzi, Marco; Mangiatordi, Giuseppe Felice; Abate, Carmen 分享 收藏
N-adamantyl-anthranil amide derivatives: New selective ligands for the cannabinoid receptor subtype 2 (CB2R) N-金刚烷基-邻氨基苯甲酰胺衍生物: 大麻素受体亚型2 (CB2R) 的新选择性配体 Graziano, Giovanni; Delre, Pietro; Carofiglio, Francesca; Brea, Jose; Ligresti, Alessia; Kostrzewa, Magdalena; Riganti, Chiara; Gioe-Gallo, Claudia; Majellaro, Maria; Nicolotti, Orazio; Colabufo, Nicola Antonio; Abate, Carmen; Loza, Maria Isabel; Sotelo, Eddy; Mangiatordi, Giuseppe Felice; Contino, Marialessandra; Stefanachi, Angela; Leonetti, Francesco 分享 收藏
Exploring Mannosylpurines as Copper Chelators and Cholinesterase Inhibitors with Potential for Alzheimer's Disease Schino, Ignazio; Cantore, Mariangela; de Candia, Modesto; Altomare, Cosimo D.; Maria, Catarina; Barros, Joao; Cachatra, Vasco; Calado, Patricia; Shimizu, Karina; Freitas, Adilson A.; Oliveira, Maria C.; Ferreira, Maria J.; Lopes, Jose N. C.; Colabufo, Nicola A.; Rauter, Amelia P. 分享 收藏
Development of N-(1-Adamantyl)benzamides as Novel Anti-Inflammatory Multitarget Agents Acting as Dual Modulators of the Cannabinoid CB2 Receptor and Fatty Acid Amide Hydrolase Intranuovo, Francesca; Brunetti, Leonardo; DelRe, Pietro; Mangiatordi, Giuseppe Felice; Stefanachi, Angela; Laghezza, Antonio; Niso, Mauro; Leonetti, Francesco; Loiodice, Fulvio; Ligresti, Alessia; Kostrzewa, Magdalena; Brea, Jose; Loza, Maria Isabel; Sotelo, Eddy; Saviano, Michele; Colabufo, Nicola Antonio; Riganti, Chiara; Abate, Carmen; Contino, Marialessandra 分享 收藏
Extra virgin olive oil extract rich in secoiridoids induces an anti-inflammatory profile in peripheral blood mononuclear cells from obese children De Santis, Stefania; Crupi, Pasquale; Piacente, Laura; Mestice, Anna; Colabufo, Nicola Antonio; Amodio, Loredana; Pontrelli, Paola; Gesualdo, Loreto; Moschetta, Antonio; Clodoveo, Maria Lisa; Faienza, Maria Felicia; Corbo, Filomena 分享 收藏
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Liquid Biopsy beyond Cancer: A miRNA Detection in Serum with Electrochemical Chip for Non-Invasive Coeliac Disease Diagnosis Caratelli, Veronica; Moccia, Maria; Paggioro, Francesca R.; Fiore, Luca; Avitabile, Concetta; Saviano, Michele; Imbriani, Anna Lisa; Dardano, Principia; De Stefano, Luca; Moscone, Danila; Colabufo, Nicola A.; El Idrissi, Imane Ghafir; Russo, Francesco; Riezzo, Giuseppe; Giannelli, Gianluigi; Arduini, Fabiana 分享 收藏
Overcoming Multidrug Resistance (MDR): Design, Biological Evaluation and Molecular Modelling Studies of 2,4-Substituted Quinazoline Derivatives Braconi, Laura; Teodori, Elisabetta; Contino, Marialessandra; Riganti, Chiara; Bartolucci, Gianluca; Manetti, Dina; Romanelli, Maria Novella; Perrone, Maria Grazia; Colabufo, Nicola Antonio; Guglielmo, Stefano; Dei, Silvia 分享 收藏