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Adam McCluskey

the university of newcastle

54H指数
365论文数
9.9K被引数
收录论文 132
发表时间
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From indole to pyrrole-based inhibitors of the large GTPase, dynamin and the in-cell inhibition of clathrin mediated endocytosis从吲哚到基于吡咯的大GTP酶、dynamin及其对网格蛋白介导的内吞作用的细胞内抑制剂的抑制
errEuropean Journal of Medicinal Chemistry
IF5.9
err2026-09-01
err0
PREAI
errBeatrice Chiew; Nicholas S. O’Brien; Kate Prichard; Michael P. Hamilton; Mohammed K. Amin; Bryony Munro; Jakobi Stegh; Jing Xue; Phillip J. Robinson; Adam McCluskey
err分享
err收藏
Sulfonadyn Compounds: A Class of Aryl Sulfonamides That Inhibit Dynamin GTPase and Clathrin-Mediated Endocytosis and Are Antiepileptic in Animal Models磺胺达尼化合物：一类抑制Dynamin GTPase和笼蛋白介导的内吞作用且在动物模型中具有抗癫痫活性的芳基磺酰胺类化合物
errACS Chemical Biology
IF3.8
err2026-06-18
err0
PREAI
errNigel C. Jones; Mark J. Robertson; Luke R. Odell; Ngoc Chau; Jing Xue; Joseph I. Ambrus; Fiona M. Deane; Nicholas S. O’Brien; Kelly A. Young; Anna Mariana; Nick N. Gorgani; Peter G. Hains; Terence J. O’Brien; Phillip J. Robinson; Adam McCluskey
err分享
err收藏
In vitro activity of robenidine analogue NCL195 against methicillin-resistant Staphylococcus pseudintermedius罗贝尼定类似物NCL195在体外对耐甲氧西林中间型金黄色葡萄球菌的活性
errMicrobiology Spectrum
IF3.8
err2026-06-02
err0
PREAI
errBista, Sayara; Nguyen, Hang Thi; Soares da Costa, Tatiana P.; Woolford, Lucy; Blaskovich, Mark A. T.; Veltman, Tania; Young, Kelly A.; McCluskey, Adam; Siak, Meng; Page, Stephen W.; Venter, Henrietta; Trott, Darren J.; Ogunniyi, Abiodun D.
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DFT guided design of novel quinone bioisosteres as inhibitors of the clathrin N-terminal domain-amphiphysin protein-protein interaction. Dihydroquinazolin-4(1H)-ones and quinazolin-3(4H)-ones.DFT指导的新型喹诺酮生物电子等排体的设计，作为网格蛋白N端域-突触体蛋白蛋白间相互作用的抑制剂。二氢喹唑啉-4(1H)-酮和喹唑啉-3(4H)-酮。
errEuropean Journal of Medicinal Chemistry
IF5.9
err2026-03-02
err0
PREAI
errNicholas S. O’Brien; Jing Xue; Claudia Bahnik; Martin Neuenschwander; Michael Kraub; Phillip J. Robinson; Volker Haucke; Adam McCluskey
err分享
err收藏
Substituted Benzylidene-3-Oxo-3,4-Dihydro-2H-Benzo[b][1,4]thiazine-6-Carboxylic Acid Analogs as Dynamin GTPase Inhibitors取代的Benzylidene-3-Oxo-3,4-Dihydro-2H-Benzo[b][1,4]thiazine-6-羧酸类似物作为Dynamin GTPase抑制剂
errCHEMMEDCHEM
IF3.4
err2025-11-01
err0
PREAI
errLin, Andrew J. S.; O'Brien, Nicholas S.; Florence, Abigail; Killen, Matthew; Frailey, Shelby L.; Gilbert, Jayne; Sakoff, Jennette A.; Amin, Mohammed K.; Castelloe, Emily E.; Chau, Ngoc; Xue, Jing; Robinson, Phillip J.; McCluskey, Adam
err分享
err收藏
Exploration of hydrazine-based small molecules as metal chelators for KDM4 inhibition肼基小分子作为KDM4抑制剂的金属螯合剂研究
errRSC Med. Chem.
IF3.6
err2025-08-22
err0
PREAI
errAngus J. Saxton; Jayden Sterling; Michael P. Hamilton; Ramzi H. Abbassi; Adam McCluskey; Lenka Munoz; Jennifer R. Baker
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err收藏
Front Cover: Inhibition of the Clathrin Terminal Domain—Amphiphysin Protein–Protein Interaction. Probing the Pitstop 2 Aromatic Moiety (ChemMedChem 16/2025)封面: 抑制网格蛋白末端结构域—突触小泡蛋白的蛋白质-蛋白质相互作用。探查 Pitstop 2 芳香基团 (ChemMedChem 16/2025)
errChemMedChem
IF3.4
err2025-08-21
err0
PREAI
errKate Prichard; Mark J Robertson; Ngoc Chau; Jing Xue; Martin Neuenschwander; Uwe Fink; Andre Horatscheck; Marc Nazare; Phillip J Robinson; Volker Haucke; Adam McCluskey
err分享
err收藏
Inhibition of the Clathrin Terminal Domain—Amphiphysin Protein–Protein Interaction. Probing the Pitstop 2 Aromatic Moiety抑制网格蛋白末端结构域—突触小泡蛋白的蛋白质-蛋白质相互作用。探查Pitstop 2的芳香基团
errChemMedChem
IF3.4
err2025-07-11
err0
PREAI
errKate Prichard; Mark J Robertson; Ngoc Chau; Jing Xue; Martin Neuenschwander; Uwe Fink; Andre Horatscheck; Marc Nazare; Phillip J Robinson; Volker Haucke; Adam McCluskey
err分享
err收藏
Next-generation small molecule inhibitors of clathrin function acutely inhibit endocytosis下一代小分子抑制剂的笼形蛋白功能急性抑制内吞作用
errSTRUCTURE
IF4.3
err2025-05-01
err1
errOAAI
errHoratscheck, Andre; Krauss, Michael; Bulut, Haydar; Chambon, Valerie; Zadah, Massilullah Shafaq; Dransart, Estelle; Peloza, Kimberly; Santos, Karine F.; Robertson, Mark J.; Prichard, Kate; Miksche, Sandra; Radetzki, Silke; von Kries, Jens-Peter; Wahl, Markus C.; McCluskey, Adam; Johannes, Ludger
err分享
err收藏
Quinoline- and Pyrimidine-based Allosteric Modulators of the Sarco/Endoplasmic Reticulum Calcium ATPase
errCHEMMEDCHEM
IF3.4
err2024-11-21
err0
errOAAI
errPaula, Stefan; Jahani, Farnaz; Almahmodi, Dina; Sobota, Sydni; Devaraja, Shiffany; O'Brien, Nicholas S.; Young, Kelly A.; Prichard, Kate; McCluskey, Adam
err分享
err收藏
Inhibition Clathrin Mediated Endocytosis: Pitstop 1 and Pitstop 2 Chimeras
errCHEMMEDCHEM
IF3.4
err2024-09-29
err0
errOAAI
errPrichard, Kate; Chau, Ngoc; Xue, Jing; Krauss, Michael; Sakoff, Jennette A.; Gilbert, Jayne; Bahnik, Claudia; Muehlbauer, Maria; Radetzki, Silke; Robinson, Phillip J.; Haucke, Volker; McCluskey, Adam
err分享
err收藏
Next-generation of BBQ analogues that selectively target breast cancer
errFRONTIERS IN CHEMISTRY
IF4.2
err2024-06-21
err0
errOAAI
errBaker, Jennifer R.; Gilbert, Jayne; O'Brien, Nicholas S.; Russell, Cecilia C.; Mccluskey, Adam; Sakoff, Jennette A.
err分享
err收藏
2,3-Dihydroquinazolin-4(1H)-ones and quinazolin-4(3H)-ones as broad-spectrum cytotoxic agents and their impact on tubulin polymerisation
errRSC MEDICINAL CHEMISTRY
IF3.6
err2024-01-01
err3
PREAI
errO'Brien, Nicholas S.; Gilbert, Jayne; McCluskey, Adam; Sakoff, Jennette A.
err分享
err收藏
Oral administration of a 2-aminopyrimidine robenidine analogue (NCL1 95) significantly reduces Staphylococcus aureus infection and reduces Escherichia coli infection in combination with sub -inhibitory colistin concentrations in a bioluminescent mouse model
errANTIMICROBIAL AGENTS AND CHEMOTHERAPY
IF4.5
err2023-10-18
err0
errOAAI
errNguyen, Hang Thi; Venter, Henrietta; Woolford, Lucy; Young, Kelly A.; Mccluskey, Adam; Garg, Sanjay; Sapula, Sylvia S.; Page, Stephen W.; Ogunniyi, Abiodun David; Trott, Darren J.
err分享
err收藏
Expansion of a Synthesized Library of N-Benzyl Sulfonamides Derived from an Indole Core to Target Pancreatic Cancer
errCHEMMEDCHEM
IF3.4
err2023-07-20
err2
PREAI
errHopkins, Megan D.; Costello, Ian J.; Brandeburg, Zachary C.; Slay, Emily L.; Zanders, Levi A.; Dunn, Caroline E.; Derewonko, Carina A.; Davitt, Colin L.; Reeder, Madison A.; Prichard, Kate; Chiew, Beatrice; McCluskey, Adam; Sheaff, Robert J.; Lamar, Angus A.
err分享
err收藏
Systematic literature review reveals suboptimal use of chemical probes in cell-based biomedical research
errNATURE COMMUNICATIONS
IF15.7
err2023-06-03
err9
errOAAI
errSterling, Jayden; Baker, Jennifer R. R.; McCluskey, Adam; Munoz, Lenka
err分享
err收藏
Wiskostatin and other carbazole scaffolds as off target inhibitors of dynamin I GTPase activity and endocytosis
errEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
IF5.9
err2023-02-01
err4
PREAI
errCossar, Peter J.; Cardoso, David; Mathwin, Daniel; Russell, Cecilia C.; Chiew, Beatrice; Hamilton, Michael P.; Baker, Jennifer R.; Young, Kelly A.; Chau, Ngoc; Robinson, Phillip J.; McCluskey, Adam
err分享
err收藏
The sulfonadyns: a class of aryl sulfonamides inhibiting dynamin I GTPase and clathrin mediated endocytosis are anti-seizure in animal models
errRSC MEDICINAL CHEMISTRY
IF3.6
err2023-01-01
err3
errOAAI
errOdell, Luke R. R.; Jones, Nigel C. C.; Chau, Ngoc; Robertson, Mark J. J.; Ambrus, Joseph I. I.; Deane, Fiona M. M.; Young, Kelly A. A.; Whiting, Ainslie; Xue, Jing; Prichard, Kate; Daniel, James A. A.; Gorgani, Nick N. N.; O'Brien, Terence J. J.; Robinson, Phillip J. J.; McCluskey, Adam
err分享
err收藏
Novel piperazine-1,2,3-triazole leads for the potential treatment of pancreatic cancer
errRSC MEDICINAL CHEMISTRY
IF3.6
err2023-01-01
err1
errOAAI
errSun, Jufeng; Baker, Jennifer R.; Russell, Cecilia C.; Pham, Hong N. T.; Goldsmith, Chloe D.; Cossar, Peter J.; Sakoff, Jennette A.; Scarlett, Christopher J.; Mccluskey, Adam
err分享
err收藏
Prodrugs of the Archetypal Dynamin Inhibitor Bis-T-22
errCHEMMEDCHEM
IF3.4
err2022-11-09
err2
errOAAI
errOdell, Luke R.; Robertson, Mark J.; Young, Kelly A.; McGeachie, Andrew B.; Quan, Annie; Robinson, Phillip J.; McCluskey, Adam
err分享
err收藏

研究方向

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