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收藏Novel triazole-tethered thiazol-4(5H)-one hybrids as potential therapeutics for obesity and type 2 diabetes: in vitro, in vivo, and in silico evaluations新型三唑连接的噻唑-4(5H)-酮杂化物作为肥胖和2型糖尿病潜在治疗药物:体外、体内及计算机模拟评价
El-Sofany, Walaa I.; Toumi, Amani; Daoud, Ismail; Haddad, Saoussen; Latif, Salman; Alshammari, Ahlam F.; Alshammari, Mona Zaheed; Alshammari, Hissah Khashman; Alshammari, Nawal S.; Boudriga, Sarra; Hamden, Khaled
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收藏Antiobesity and antidiabetes effects of Cyperus rotundus rhizomes presenting protein tyrosine phosphatase, dipeptidyl peptidase 4, metabolic enzymes, stress oxidant and inflammation inhibitory potential
Abdella, Faiza I. A.; Toumi, Amani; Boudriga, Sarra; Alanazi, Tahani Y. A.; Alshamari, Asma K.; Alrashdi, Ahlam Abdulrahman; Hamden, Khaled
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收藏Design, synthesis and biological evaluation of new 1,ω-Bis-(5-alkyl-3-tosyl-1,3,4,2-triazaphospholino)alkanes as in vitro α-amylase and lipase inhibitors新型1,ω-双-(5-烷基-3-甲苯磺酰基-1,3,4,2-三唑磷杂) 烷烃作为体外 α-淀粉酶和脂肪酶抑制剂的设计,合成和生物学评价
Hamzaoui, Salwa; Ben Salah, Bochra; Bouguerra, Soumaya; Hamden, Khaled; Alghamdi, Othman A.; Miled, Nabil; Kossentini, Mohamed
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收藏Synthesis of Tetracyclic Spirooxindolepyrrolidine-Engrafted Hydantoin Scaffolds: Crystallographic Analysis, Molecular Docking Studies and Evaluation of Their Antimicrobial, Anti-Inflammatory and Analgesic Activities
Toumi, Amani; Abdella, Faiza I. A.; Boudriga, Sarra; Alanazi, Tahani Y. A.; Alshamari, Asma K.; Alrashdi, Ahlam Abdulrahman; Dbeibia, Amal; Hamden, Khaled; Daoud, Ismail; Knorr, Michael; Kirchhoff, Jan-Lukas; Strohmann, Carsten
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收藏New spiropyrrolothiazole derivatives bearing an oxazolone moiety as potential antidiabetic agent: Design, synthesis, crystal structure, Hirshfeld surface analysis, ADME and molecular docking studies
Ben Hammouda, Manel; Boudriga, Sarra; Hamden, Khaled; Askri, Moheddine; Knorr, Michael; Strohmann, Carsten; Brieger, Lukas; Krupp, Anna; Anouar, El Hassane; Snoussi, Mejdi; Aouadi, Kaiss; Kadri, Adel
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收藏Diversity-Oriented Synthesis of Spiropyrrolo[1,2-a]isoquinoline Derivatives via Diastereoselective and Regiodivergent Three-Component 1,3-Dipolar Cycloaddition Reactions: In Vitro and in Vivo Evaluation of the Antidiabetic Activity of Rhodanine Analogues
Toumi, Amani; Boudriga, Sarra; Hamden, Khaled; Daoud, Ismail; Askri, Moheddine; Soldera, Armand; Lohier, Jean-Francois; Strohmann, Carsten; Brieger, Lukas; Knorr, Michael
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收藏Antihyperlipidemic, Antihyperglycemic, and Liver Function Protection of Olea europaea var. Meski Stone and Seed Extracts: LC-ESI-HRMS-Based Composition Analysis
Ben Saad, Amina; Tiss, Mohamed; Keskes, Henda; Chaari, Anisa; Sakavitsi, Maria Eleni; Hamden, Khaled; Halabalaki, Maria; Allouche, Noureddine
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收藏Protective and curative effects of Bacillus subtilis SPB1 biosurfactant on high-fat-high-fructose diet induced hyperlipidemia, hypertriglyceridemia and deterioration of liver function in rats
Zouari, Raida; Hamden, Khaled; El Feki, Abdelfattah; Chaabouni, Khansa; Makni-Ayadi, Fatma; Kallel, Choumous; Sallemi, Fahima; Ellouze-Chaabouni, Semia; Ghribi-Aydi, Dhouha
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