未登录Ifinatamab deruxtecan (I-DXd), a novel B7-H3-targeting antibody-drug conjugate, demonstrates efficient payload delivery into tumor through target-dependent internalization
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收藏Epigenetic programming underpins B cell dysfunction in human SLE
Scharer, Christopher D.; Blalock, Emily L.; Mi, Tian; Barwick, Benjamin G.; Jenks, Scott A.; Deguchi, Tsuneo; Cashman, Kevin S.; Neary, Bridget E.; Patterson, Dillon G.; Hicks, Sakeenah L.; Khosroshahi, Arezou; Lee, F. Eun-Hyung; Wei, Chungwen; Sanz, Inaki; Boss, Jeremy M.
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收藏Humanized UGT2 and CYP3A transchromosomic rats for improved prediction of human drug metabolism人源化UGT2和CYP3A转染色体大鼠用于改善人类药物代谢的预测
Kazuki, Yasuhiro; Kobayashi, Kaoru; Hirabayashi, Masumi; Abe, Satoshi; Kajitani, Naoyo; Kazuki, Kanako; Takehara, Shoko; Takiguchi, Masato; Satoh, Daisuke; Kuze, Jiro; Sakuma, Tetsushi; Kaneko, Takehito; Mashimo, Tomoji; Osamura, Minori; Hashimoto, Mari; Wakatsuki, Riko; Hirashima, Rika; Fujiwara, Ryoichi; Deguchi, Tsuneo; Kurihara, Atsushi; Tsukazaki, Yasuko; Senda, Naoto; Yamamoto, Takashi; Scheer, Nico; Oshimura, Mitsuo
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收藏Synthesis and evaluation of novel stearoyl-CoA desaturase 1 inhibitors: 1′-{6-[5-(pyridin-3-ylmethyl)-1,3,4-oxadiazol-2-yl]pyridazin-3-yl}-3,4-dihydrospiro[chromene-2,4′-piperidine] analogs
Uto, Yoshikazu; Ueno, Yuko; Kiyotsuka, Yohei; Miyazawa, Yuriko; Kurata, Hitoshi; Ogata, Tsuneaki; Yamada, Makiko; Deguchi, Tsuneo; Konishi, Masahiro; Takagi, Toshiyuki; Wakimoto, Satoko; Ohsumi, Jun
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