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Safety, tolerability, pharmacokinetics, and pharmacodynamics of a novel kappa opioid receptor agonist ZYKR1: a randomized double-blind placebo-control phase 1 study in healthy adult human participants Kansagra, Kevinkumar A.; Momin, Taufik; Patel, Hardik B.; Shah, Chintan; Parmar, Gordhan; Ghoghari, Ashok; Patel, Harilal V.; Parmar, Deven V. 分享 收藏
Discovery of a potent G-protein-coupled receptor 119 agonist for the treatment of type 2 diabetes Pola, Suresh; Shah, Shailesh R.; Pingali, Harikishore; Zaware, Pandurang; Thube, Baban; Makadia, Pankaj; Patel, Hoshang; Bandyopadhyay, Debdutta; Rath, Akshyaya; Giri, Suresh; Patel, Jitendra H.; Ranvir, R. K.; Sundar, S. R.; Patel, Harilal; Kumar, Jeevan; Jain, Mukul R. 分享 收藏
A Phase 3, Randomized, Open-label, Noninferiority Trial Evaluating Anti-rabies Monoclonal Antibody Cocktail (Twinrab™) Against Human Rabies Immunoglobulin Reply Kansagra, Kevinkumar; Parmar, Deven; Mendiratta, Sanjeev Kumar; Patel, Jatin; Joshi, Shuchi; Sharma, Nitin; Parihar, Anurag; Bhoge, Swapnil; Patel, Harilal; Kalita, Pankaj; Munshi, Renuka; Kurmi, Prakash; Shah, Ruchir; Gupta, Abhishek; Bhalla, Hira Lal; Bekkalele, Harish; Verma, Rajendra Kumar; Agarwal, Dinesh; Sharma, Shrikant; Gawande, Avinash; Chhaya, Gaurav 分享 收藏
Outcomes of Desidustat Treatment in People with Anemia and Chronic Kidney Disease: A Phase 2 Study Desidustat治疗贫血和慢性肾脏疾病患者的结果: 一项2期研究 Parmar, Deven V.; Kansagra, Kevinkumar A.; Patel, Jatin C.; Joshi, Shuchi N.; Sharma, Nitin S.; Shelat, Apeksha D.; Patel, Nirav B.; Nakrani, Vishal B.; Shaikh, Farheen A.; Patel, Harilal V.; Sharma, Raj Kumar; Gupta, Krishan Lal; Devaraju, Sree Bhushan Raju; Koradia, Parshottam; Agrawal, Dhananjai; Sahay, Manisha; Sajgure, Atul; Srinivasa, Sanjay; Singhal, Saurabh; Redewad, Nagnath K.; Varade, Deepak 分享 收藏
Identification and preclinical characterization of a novel and potent poly (ADP-ribose) polymerase (PARP) inhibitor ZYTP1 Jain, Mukul R.; Mohapatra, Jogeswar; Bandhyopadhyay, Debdutta; Chatterjee, Abhijit; Ghoshdastidar, Krishnarup; Patel, Dinesh; Patel, Ankit; Bhayani, Hitesh; Srivastava, Brijesh Kumar; Shedage, Sandeep A.; Kadam, Pravin; Sundar, Rajesh; Patel, Harilal; Giri, Poonam; Patel, Prakash; Gupta, Laxmikant; Srinivas, Nuggehally R.; Patel, Pankaj R.; Desai, Ranjit C. 分享 收藏
One should avoid retro-orbital pharmacokinetic sample collections for intranasal dosing in rats: Illustration of spurious pharmacokinetics generated for anti-migraine drugs zolmitriptan and eletriptan Patel, Harilal; Patel, Prakash; Modi, Nirav; Shah, Shaival; Ghoghari, Ashok; Variya, Bhavesh; Laddha, Ritu; Baradia, Dipesh; Dobaria, Nitin; Mehta, Pavak; Srinivas, Nuggehally R. 分享 收藏
ZY15557, a novel, long acting inhibitor of dipeptidyl peptidase-4, for the treatment of Type 2 diabetes mellitus Jain, Mukul R.; Joharapurkar, Amit A.; Kshirsagar, Samadhan G.; Patel, Vishal J.; Bahekar, Rajesh H.; Patel, Harilal V.; Jadav, Pradip A.; Patel, Pankaj R.; Desai, Ranjit C. 分享 收藏
Discovery of a Potent and Orally Efficacious TGR5 Receptor Agonist 发现一种有效且口服有效的TGR5受体激动剂 Agarwal, Sameer; Patil, Amit; Aware, Umesh; Deshmukh, Prashant; Darji, Brijesh; Sasane, Santosh; Sairam, Kalapatapu V. V. M.; Priyadarsiny, Priyanka; Giri, Poonam; Patel, Harilal; Giri, Suresh; Jain, Mukul; Desai, Ranjit C. 分享 收藏
Pharmacological characterization of ZYDPLA1, a novel long-acting dipeptidyl peptidase-4 inhibitor Jain, Mukul R.; Joharapurkar, Amit A.; Bahekar, Rajesh H.; Patel, Harilal; Jadav, Pradip; Kshirsagar, Samadhan G.; Patel, Vishal J.; Patel, Kartikkumar N.; Ramanathan, Vikram K.; Patel, Pankaj R.; Desai, Ranjit C. 分享 收藏
Synthesis and structure-activity relationship of potent, selective and orally active anthranilamide-based factor Xa inhibitors: Application of weakly basic sulfoximine group as novel S4 binding element Pandya, Vrajesh; Jain, Mukul; Chakrabarti, Ganes; Soni, Hitesh; Parmar, Bhavesh; Chaugule, Balaji; Patel, Jigar; Jarag, Tushar; Joshi, Jignesh; Joshi, Nirav; Rath, Akshyaya; Unadkat, Vishal; Sharma, Bhavesh; Ajani, Haresh; Kumar, Jeevan; Sairam, Kalapatapu V. V. M.; Patel, Harilal; Patel, Pankaj 分享 收藏
Discovery of Orally Active, Potent, and Selective Benzotriazole-Based PTP1B Inhibitors 口服活性,强效和选择性的基于苯并三唑的PTP1B抑制剂的发现 Patel, Dipam; Jain, Mukul; Shah, Shailesh R.; Bahekar, Rajesh; Jadav, Pradip; Darji, Brijesh; Siriki, Yernaidu; Bandyopadhyay, Debdutta; Joharapurkar, Amit; Kshirsagar, Samadhan; Patel, Harilal; Shaikh, Mubeen; Sairam, Kalapatapu V. V. M.; Patel, Pankaj 分享 收藏
Design and synthesis of novel oxazole containing 1,3-Dioxane-2-carboxylic acid derivatives as PPAR α/γ dual agonists Pingali, Harikishore; Jain, Mukul; Shah, Shailesh; Makadia, Pankaj; Zaware, Pandurang; Goel, Ashish; Patel, Megha; Giri, Suresh; Patel, Harilal; Patel, Pankaj 分享 收藏