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Oleg Ursu

merck & company

30H指数
139论文数
7.3K被引数
收录论文 35
发表时间
PepSeA: Peptide Sequence Alignment and Visualization Tools to Enable Lead Optimization
err2022-02-22
err3
errOAAI
errBaylon, Javier L.; Ursu, Oleg; Muzdalo, Anja; Wassermann, Anne Mai; Adams, Gregory L.; Spale, Martin; Mejzlik, Petr; Gromek, Anna; Pisarenko, Viktor; Hancharyk, Dzianis; Jenkins, Esteban; Bednar, David; Chang, Charlie; Clarova, Kamila; Glick, Meir; Bitton, Danny A.
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Machine learning prediction and tau-based screening identifies potential Alzheimer's disease genes relevant to immunity机器学习预测和基于tau的筛选确定与免疫相关的潜在阿尔茨海默病基因
err2022-02-11
err27
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errBinder, Jessica; Ursu, Oleg; Bologa, Cristian; Jiang, Shanya; Maphis, Nicole; Dadras, Somayeh; Chisholm, Devon; Weick, Jason; Myers, Orrin; Kumar, Praveen; Yang, Jeremy J.; Bhaskar, Kiran; Oprea, Tudor, I
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Identification of new GLUT2-selective inhibitors through in silico ligand screening and validation in eukaryotic expression systems
err2021-07-02
err16
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errSchmidl, Sina; Ursu, Oleg; Iancu, Cristina V.; Oreb, Mislav; Oprea, Tudor I.; Choe, Jun-yong
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DrugCentral 2021 supports drug discovery and repositioning
err2020-11-05
err109
errOAAI
errAvram, Sorin; Bologa, Cristian G.; Holmes, Jayme; Bocci, Giovanni; Wilson, Thomas B.; Dac-Trung Nguyen; Curpan, Ramona; Halip, Liliana; Bora, Alina; Yang, Jeremy J.; Knockel, Jeffrey; Sirimulla, Suman; Ursu, Oleg; Oprea, Tudor, I
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A mass spectrometry-based proteome map of drug action in lung cancer cell lines (Jul, 10.1038/s41589-020-0572-3, 2020)
err2020-08-11
err0
errOAAI
errRuprecht, Benjamin; Di Bernardo, Julie; Wang, Zhao; Mo, Xuan; Ursu, Oleg; Christopher, Matthew; Fernandez, Rafael B.; Zheng, Li; Dill, Brian D.; Wang, Huijun; Xu, Yuting; Liaw, Andy; Mortison, Jonathan D.; Siriwardana, Nirodhini; Andresen, Brian; Glick, Meir; Tata, James R.; Kutilek, Victoria; Cornella-Taracido, Ivan; Chi, An
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A mass spectrometry-based proteome map of drug action in lung cancer cell lines
err2020-07-20
err41
PREAI
errRuprecht, Benjamin; Di Bernardo, Julie; Wang, Zhao; Mo, Xuan; Ursu, Oleg; Christopher, Matthew; Fernandez, Rafael B.; Zheng, Li; Dill, Brian D.; Wang, Huijun; Xu, Yuting; Liaw, Andy; Mortison, Jonathan D.; Siriwardana, Nirodhini; Andresen, Brian; Glick, Meir; Tata, James R.; Kutilek, Victoria; Cornella-Taracido, Ivan; Chi, An
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DrugCentral 2018: an update药物中心2018: 更新
err2018-10-29
err95
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errUrsu, Oleg; Holmes, Jayme; Bologa, Cristian G.; Yang, Jeremy J.; Mathias, Stephen L.; Stathias, Vasileios; Dac-Trung Nguyen; Schurer, Stephan; Oprea, Tudor
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Activation of Rho Family GTPases by Small Molecules
err2018-05-10
err16
errOAAI
errPalsuledesai, Charuta C.; Suryiladze, Zurab; Waller, Anna; Miscioscia, T. Fabiola; Guo, Yuna; Wu, Yang; Strouse, Jake; Romero, Elsa; Salas, Virginia M.; Curpan, Ramona; Young, Susan; Carter, Mark; Foutz, Terry; Galochkina, Zhanna; Ames, Harold; Haynes, Mark K.; Edwards, Bruce S.; Nicolotti, Orazio; Luo, Li; Ursu, Oleg; Bologa, Cristian G.; Oprea, Tudor, I; Wandinger-Ness, Angela; Sklar, Larry A.
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Unexplored therapeutic opportunities in the human genome (vol 17, pg 317, 2018)人类基因组中未开发的治疗机会 (第17卷,317页,2018页)
err2018-03-23
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errOprea, Tudor I.; Bologa, Cristian G.; Brunak, Soren; Campbell, Allen; Gan, Gregory N.; Gaulton, Anna; Gomez, Shawn M.; Guha, Rajarshi; Hersey, Anne; Holmes, Jayme; Jadhav, Ajit; Jensen, Lars Juhl; Johnson, Gary L.; Karlson, Anneli; Leach, Andrew R.; Ma'ayan, Avi; Malovannaya, Anna; Mani, Subramani; Mathias, Steven L.; McManus, Michael T.; Meehan, Terrence F.; von Mering, Christian; Muthas, Daniel; Dac-Trung Nguyen; Overington, John P.; Papadatos, George; Qin, Jun; Reich, Christian; Roth, Bryan L.; Schurer, Stephan C.; Simeonov, Anton; Sklar, Larry A.; Southall, Noel; Tomita, Susumu; Tudose, Ilinca; Ursu, Oleg; Vidovic, Dusica; Waller, Anna; Westergaard, David; Yang, Jeremy J.; Zahoranszky-Kohalmi, Gergely
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Unexplored therapeutic opportunities in the human genome人类基因组中未开发的治疗机会
err2018-03-23
err278
errOAAI
errOprea, Tudor I.; Bologa, Cristian G.; Brunak, Soren; Campbell, Allen; Gan, Gregory N.; Gaulton, Anna; Gomez, Shawn M.; Guha, Rajarshi; Hersey, Anne; Holmes, Jayme; Jadhav, Ajit; Jensen, Lars Juhl; Johnson, Gary L.; Karlson, Anneli; Leach, Andrew R.; Ma'ayan, Avi; Malovannaya, Anna; Mani, Subramani; Mathias, Stephen L.; McManus, Michael T.; Meehan, Terrence F.; von Mering, Christian; Muthas, Daniel; Dac-Trung Nguyen; Overington, John P.; Papadatos, George; Qin, Jun; Reich, Christian; Roth, Bryan L.; Schurer, Stephan C.; Simeonov, Anton; Sklar, Larry A.; Southall, Noel; Tomita, Susumu; Tudose, Ilinca; Ursu, Oleg; Vidovic, Dusica; Waller, Anna; Westergaard, David; Yang, Jeremy J.; Zahoranszky-Kohalmi, Gergely
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Protein biomarker druggability profiling蛋白质生物标志物药力分析
err2017-02-01
err2
errOAAI
errMani, Subramani; Cannon, Daniel; Ohls, Robin; Oprea, Tudor; Mathias, Stephen; Ballard, Karri; Ursu, Oleg; Bologa, Cristian
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A comprehensive map of molecular drug targets分子药物靶点的综合图谱
err2016-12-02
err1.7K
errOAAI
errSantos, Rita; Ursu, Oleg; Gaulton, Anna; Bento, A. Patricia; Donadi, Ramesh S.; Bologa, Cristian G.; Karlsson, Anneli; Al-Lazikani, Bissan; Hersey, Anne; Oprea, Tudor I.; Overington, John P.
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Pharos: Collating protein information to shed light on the druggable genomePharos: 整理蛋白质信息以阐明可药用基因组
err2016-11-29
err189
errOAAI
errDac-Trung Nguyen; Mathias, Stephen; Bologa, Cristian; Brunak, Soren; Fernandez, Nicolas; Gaulton, Anna; Hersey, Anne; Holmes, Jayme; Jensen, Lars Juhl; Karlsson, Anneli; Liu, Guixia; Ma'ayan, Avi; Mandava, Geetha; Mani, Subramani; Mehta, Saurabh; Overington, John; Patel, Juhee; Rouillard, Andrew D.; Schurer, Stephan; Sheils, Timothy; Simeonov, Anton; Sklar, Larry A.; Southall, Noel; Ursu, Oleg; Vidovic, Dusica; Waller, Anna; Yang, Jeremy; Jadhav, Ajit; Oprea, Tudor I.; Guha, Rajarshi
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DrugCentral: online drug compendium药物中心: 在线药物概要
err2016-10-26
err194
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errUrsu, Oleg; Holmes, Jayme; Knockel, Jeffrey; Bologa, Cristian G.; Yang, Jeremy J.; Mathias, Stephen L.; Nelson, Stuart J.; Oprea, Tudor I.
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BDDCS, the Rule of 5 and drugabilityBDDCS、5法则与可药性
err2016-06-01
err567
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errBenet, Leslie Z.; Hosey, Chelsea M.; Ursu, Oleg; Oprea, Tudor I.
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Badapple: promiscuity patterns from noisy evidenceBadaple: 来自嘈杂证据的滥交模式
err2016-05-28
err86
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errYang, Jeremy J.; Ursu, Oleg; Lipinski, Christopher A.; Sklar, Larry A.; Oprea, Tudor I.; Bologa, Cristian G.
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Discovery of a specific inhibitor of human GLUT5 by virtual screening and in vitro transport evaluation通过虚拟筛选和体外转运评估发现人GLUT5的特异性抑制剂
err2016-04-14
err57
errOAAI
errThompson, Alayna M. George; Ursu, Oleg; Babkin, Petr; Iancu, Cristina V.; Whang, Alex; Oprea, Tudor I.; Choe, Jun-yong
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R-ketorolac targets Cdc42 and Rac1 GTPases and alters ovarian tumor cell behaviors critical for invasion and metastasis
err2015-08-01
err3
PREAI
errGuo, Yuna; Kenney, S. Ray; Sklar, Larry A.; Buranda, Tione; Oprea, Tudor I.; Ursu, Oleg; Adams, Sarah F.; Rutledge, Teresa; Muller, Carolyn; Lomo, Lesley; Hudson, Laurie G.; Wandinger-Ness, Angela
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