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Sandra Kovachka

university cote d'azur, cnrs and icn

9H指数
26论文数
297被引数
收录论文 10
发表时间
Inhibition of PTCH1 drug efflux activity enhances chemotherapy efficacy against triple negative breast cancers抑制PTCH1药物外排活性增强三阴性乳腺癌的化疗效果
err2026-04-18
err0
errOAAI
errSarah Cogoluegnes; Sandra Kovachka; Thierry Dubois; Roberto Würth; Elisa Donato; Andreas Trumpp; Michel Franco; Frédéric Luton; Stéphane Azoulay; Isabelle Mus-Veteau
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Transcriptome-Wide, Unbiased Profiling of Ribonuclease Targeting Chimeras
err2024-07-24
err0
PREAI
errTong, Yuquan; Su, Xiaoxuan; Rouse, Warren; Childs-Disney, Jessica L.; Taghavi, Amirhossein; Zanon, Patrick R. A.; Kovachka, Sandra; Wang, Tenghui; Moss, Walter N.; Disney, Matthew D.
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Heterobifunctional small molecules to modulate RNA function
err2024-05-01
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PREAI
errKovachka, Sandra; Tong, Yuquan; Childs-Disney, Jessica L.; Disney, Matthew D.
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Identification of small molecules affecting the interaction between human hemoglobin and Staphylococcus aureus IsdB hemophore
err2024-04-09
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errOAAI
errCozzi, Monica; Failla, Mariacristina; Gianquinto, Eleonora; Kovachka, Sandra; Comani, Valeria Buoli; Compari, Carlotta; De Bei, Omar; Giaccari, Roberta; Marchesani, Francesco; Marchetti, Marialaura; Ronda, Luca; Rolando, Barbara; Baroni, Massimo; Cruciani, Gabriele; Campanini, Barbara; Bettati, Stefano; Faggiano, Serena; Lazzarato, Loretta; Spyrakis, Francesca
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Structure-guided optimization of 3-hydroxybenzoisoxazole derivatives as inhibitors of Aldo-keto reductase 1C3 (AKR1C3) to target prostate cancer3-羟基苯并异恶唑衍生物作为醛酮还原酶1C3 (AKR1C3) 抑制剂靶向前列腺癌的结构指导优化
err2024-03-01
err4
errOAAI
errPippione, Agnese Chiara; Kovachka, Sandra; Vigato, Chiara; Bertarini, Laura; Mannella, Iole; Sainas, Stefano; Rolando, Barbara; Denasio, Enrica; Piercy-Mycock, Helen; Romalho, Linda; Salladini, Edoardo; Adinolfi, Salvatore; Zonari, Daniele; Peraldo-Neia, Caterina; Chiorino, Giovanna; Passoni, Alice; Mirza, Osman Asghar; Frydenvang, Karla; Pors, Klaus; Lolli, Marco Lucio; Spyrakis, Francesca; Oliaro-Bosso, Simonetta; Boschi, Donatella
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Small molecule approaches to targeting RNA靶向RNA的小分子方法
err2024-01-26
err14
errOAAI
errKovachka, Sandra; Panosetti, Marc; Grimaldi, Benedetto; Azoulay, Stephane; Di Giorgio, Audrey; Duca, Maria
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Investigation into the Use of Encorafenib to Develop Potential PROTACs Directed against BRAFV600E Protein
err2022-12-03
err8
errOAAI
errMarini, Elisabetta; Marino, Marco; Gionfriddo, Giulia; Maione, Federica; Pandini, Marta; Oddo, Daniele; Giorgis, Marta; Rolando, Barbara; Blua, Federica; Gastaldi, Simone; Marchio, Serena; Kovachka, Sandra; Spyrakis, Francesca; Gianquinto, Eleonora; Di Nicolantonio, Federica; Bertinaria, Massimo
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New aldo-keto reductase 1C3 (AKR1C3) inhibitors based on the hydroxytriazole scaffold
err2022-07-01
err12
PREAI
errPippione, Agnese Chiara; Kilic-Kurt, Zuhal; Kovachka, Sandra; Sainas, Stefano; Rolando, Barbara; Denasio, Enrica; Pors, Klaus; Adinolfi, Salvatore; Zonari, Daniele; Bagnati, Renzo; Lolli, Marco Lucio; Spyrakis, Francesca; Oliaro-Bosso, Simonetta; Boschi, Donatella
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Covalent Probes Reveal Small-Molecule Binding Pockets in Structured RNA and Enable Bioactive Compound Design共价探针揭示结构化RNA中的小分子结合口袋,并实现生物活性化合物设计
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errSandra Kovachka; Jielei Wang; Amirhossein Taghavi; Yilin Jia; Taro Asaba; Karen C. Wolff; Mason Martin; Xueyi Yang; Samantha M. Meyer; Sabine Ottilie; Mina Heacock; Zhong Cheng; Case W. McNamara; Gurudutt Dubey; Arnab K. Chatterjee; Sumit Chanda; José Gallego; Jessica L. Childs-Disney; Matthew D. Disney
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