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Andrew M. Petros

AbbVie

40H指数
102论文数
1.0W被引数
收录论文 35
发表时间
Beyond Isotopic Labeling: Expanding the Reach of Protein-Detect NMR in Lead Discovery
err2025-03-01
err0
PREAI
errFrederick, Thomas E.; Namanja, Andrew T.; Wu, Haihong; Sun, Chaohong; Petros, Andrew M.
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Identification and structure-based drug design of cell-active inhibitors of interleukin 17A at a novel C-terminal site
err2022-08-26
err8
errOAAI
errGoedken, Eric R.; Argiriadi, Maria A.; Dietrich, Justin D.; Petros, Andrew M.; Krishnan, Navasona; Panchal, Sanjay C.; Qiu, Wei; Wu, Haihong; Zhu, Haizhong; Adams, Ashley M.; Bodelle, Pierre M.; Goguen, Lucas; Richardson, Paul L.; Slivka, Peter F.; Srikumaran, Myron; Upadhyay, Anup K.; Wu, Bainan; Judge, Russell A.; Vasudevan, Anil; Gopalakrishnan, Sujatha M.; Cox, Philip B.; Stoll, Vincent S.; Sun, Chaohong
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Insights into the Conformation and Self-Association of a Concentrated Monoclonal Antibody using Isothermal Chemical Denaturation and Nuclear Magnetic Resonance
err2021-12-01
err1
errOAAI
errXu, Jianwen; Namanja, Andrew; Chan, Siew Leong; Son, Chelsea; Petros, Andrew M.; Sun, Chaohong; Radziejewski, Czeslaw; Ihnat, Peter M.
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Development of Orally Efficacious Allosteric Inhibitors of TNFα via Fragment-Based Drug Design
err2020-12-30
err21
PREAI
errDietrich, Justin D.; Longenecker, Kenton L.; Wilson, Noel S.; Goess, Christian; Panchal, Sanjay C.; Swann, Steven L.; Petros, Andrew M.; Hobson, Adrian D.; Ihle, David; Song, Danying; Richardson, Paul; Comess, Kenneth M.; Cox, Philip B.; Dombrowski, Amanda; Sarris, Kathy; Donnelly-Roberts, Diana L.; Duignan, David B.; Gomtsyan, Arthur; Jung, Paul; Krueger, A. Chris; Mathieu, Suzanne; McClure, Andrea; Stoll, Vincent S.; Wetter, Jill; Mankovich, John A.; Hajduk, Philip J.; Vasudevan, Anil; Stoffel, Robert H.; Sun, Chaohong
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Fragment-Based Discovery of an Apolipoprotein E4 (apoE4) Stabilizer
err2019-04-01
err21
PREAI
errPetros, Andrew M.; Korepanova, Alla; Jakob, Clarissa G.; Qiu, Wei; Panchal, Sanjay C.; Wang, Jie; Dietrich, Justin D.; Brewer, Jason T.; Pohlki, Frauke; Kling, Andreas; Wilcox, Kyle; Lakics, Viktor; Bahnassawy, Lamiaa; Reinhardt, Peter; Partha, Sarathy Karunan; Bodelle, Pierre M.; Lake, Marc; Charych, Erik I.; Stoll, Vincent S.; Sun, Chaohong; Mohler, Eric G.
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The EED protein-protein interaction inhibitor A-395 inactivates the PRC2 complex (vol 13, pg 389, 2017)
err2017-08-01
err7
errOAAI
errHe, Yupeng; Selvaraju, Sujatha; Curtin, Michael L.; Jakob, Clarissa G.; Zhu, Haizhong; Comess, Kenneth M.; Shaw, Bailin; The, Juliana; Lima-Fernandes, Evelyne; Szewczyk, Magdalena M.; Cheng, Dong; Klinge, Kelly L.; Li, Huan-Qiu; Pliushchev, Marina; Algire, Mikkel A.; Maag, David; Guo, Jun; Dietrich, Justin; Panchal, Sanjay C.; Petros, Andrew M.; Sweis, Ramzi F.; Torrent, Maricel; Bigelow, Lance J.; Senisterra, Guillermo; Li, Fengling; Kennedy, Steven; Wu, Qin; Osterling, Donald J.; Lindley, David J.; Gao, Wenqing; Galasinski, Scott; Barsyte-Lovejoy, Dalia; Vedadi, Masoud; Buchanan, Fritz G.; Arrowsmith, Cheryl H.; Chiang, Gary G.; Sun, Chaohong; Pappano, William N.
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Fragment-Based, Structure-Enabled Discovery of Novel Pyridones and Pyridone Macrocycles as Potent Bromodomain and Extra-Terminal Domain (BET) Family Bromodomain Inhibitors
err2017-04-21
err59
errOAAI
errWang, Le; Pratt, John K.; Soltwedel, Todd; Sheppard, George S.; Fidanze, Steven D.; Liu, Dachun; Hasvold, Lisa A.; Mantei, Robert A.; Holms, James H.; McClellan, William J.; Wendt, Michael D.; Wada, Carol; Frey, Robin; Hansen, T. Matthew; Hubbard, Robert; Park, Chang H.; Li, Leiming; Magoc, Terrance J.; Albert, Daniel H.; Lin, Xiaoyu; Warder, Scott E.; Kovar, Peter; Huang, Xiaoli; Wilcox, Denise; Wang, Rongqi; Rajaraman, Ganesh; Petros, Andrew M.; Hutchins, Charles W.; Panchal, Sanjay C.; Sun, Chaohong; Elmore, Steven W.; Shen, Yu; Kati, Warren M.; McDaniel, Keith F.
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The EED protein-protein interaction inhibitor A-395 inactivates the PRC2 complex
err2017-01-30
err187
PREAI
errHe, Yupeng; Selvaraju, Sujatha; Curtin, Michael L.; Jakob, Clarissa G.; Zhu, Haizhong; Comess, Kenneth M.; Shaw, Bailin; The, Juliana; Lima-Fernandes, Evelyne; Szewczyk, Magdalena M.; Cheng, Dong; Klinge, Kelly L.; Li, Huan-Qiu; Pliushchev, Marina; Algire, Mikkel A.; Maag, David; Guo, Jun; Dietrich, Justin; Panchal, Sanjay C.; Petros, Andrew M.; Sweis, Ramzi F.; Torrent, Maricel; Bigelow, Lance J.; Senisterra, Guillermo; Li, Fengling; Kennedy, Steven; Wu, Qin; Osterling, Donald J.; Lindley, David J.; Gao, Wenqing; Galasinski, Scott; Barsyte-Lovejoy, Dalia; Vedadi, Masoud; Buchanan, Fritz G.; Arrowsmith, Cheryl H.; Chiang, Gary G.; Sun, Chaohong; Pappano, William N.
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Turning a Substrate Peptide into a Potent Inhibitor for the Histone Methyltransferase SETD8
err2016-10-17
err13
errOAAI
errJudge, Russell A.; Zhu, Haizhong; Upadhyay, Anup K.; Bodelle, Pierre M.; Hutchins, Charles W.; Torrent, Maricel; Marin, Violeta L.; Yu, Wenyu; Vedadi, Masoud; Li, Fengling; Brown, Peter J.; Pappano, William N.; Sun, Chaohong; Petros, Andrew M.
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Discovery of BET family proteins as cancer targets using phenotypic-based profiling and affinity capture mass spectrometry
err2016-07-15
err0
PREAI
errWarder, Scott E.; McLoughlin, Shaun M.; Hansen, T. Matthew; Richardson, Paul L.; Wilcox, Denise M.; Addo, Sadiya N.; Tang, Hua; Sun, Chaohong; Petros, Andrew M.; Panchal, Sanjay C.; Park, Chang H.; Duggan, M. Shannon; Patterson, Melanie J.; Buchanan, F. Greg; Cheng, Dong; Davis, Heather M.; Calderwood, David J.; Elmore, Steven W.; Shen, Yu
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Functional group elaboration of a low molecular weight fragment to yield the novel BET family bromodomain inhibitor ABBV-075
err2016-07-15
err0
PREAI
errMcDaniel, Keith; Le Wang; Sheppard, George; Fidanze, Steve; Pratt, John; Liu, Dachun; Hasvold, Lisa; Mantei, Robert; Park, Chang; Sarthy, Aparna; Li, Leiming; Albert, Daniel H.; Lin, Xiaoyu; Warder, Scott; Faivre, Emily; Bui, Mai H.; Huang, Xiaoli; Wilcox, Denise; Wang, Rongqi; Magoc, Terry; Rajaraman, Ganesh; Petros, Andrew; Panchal, Sanjay; Sun, Chaohong; Fang, Guowei; Elmore, Steven W.; Rosenberg, Saul; Shen, Yu; Kati, Warren
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Structure-Guided Design of a Series of MCL-1 Inhibitors with High Affinity and Selectivity (vol 58, pg 2180, 2015)
err2015-05-01
err5
PREAI
errBruncko, Milan; Wang, Le; Sheppard, George S.; Phillips, Darren C.; Tahir, Stephen K.; Xue, John; Erickson, Scott; Fidanze, Steve; Fry, Elizabeth; Hasvold, Lisa; Jenkins, Gary J.; Jin, Sha; Judge, Russell A.; Kovar, Peter J.; Madar, David; Nimmer, Paul; Park, Chang; Petros, Andrew M.; Rosenberg, Saul H.; Smith, Morey L.; Song, Xiaohong; Sun, Chaohong; Tao, Zhi-Fu; Wang, Xilu; Xiao, Yu; Zhang, Haichao; Tse, Chris; Leverson, Joel D.; Elmore, Steven W.; Souers, Andrew J.
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Structure-Guided Design of a Series of MCL-1 Inhibitors with High Affinity and Selectivity
err2015-02-26
err158
PREAI
errBruncko, Milan; Wang, Le; Sheppard, George S.; Phillips, Darren C.; Tahir, Stephen K.; Xue, John; Erickson, Scott; Fidanze, Steve; Fry, Elizabeth; Hasvold, Lisa; Jenkins, Gary J.; Jin, Sha; Judge, Russell A.; Kovar, Peter J.; Madar, David; Nimmer, Paul; Park, Chang; Petros, Andrew M.; Rosenberg, Saul H.; Smith, Morey L.; Song, Xiaohong; Sun, Chaohong; Tao, Zhi-Fu; Wang, Xilu; Xiao, Yu; Zhang, Haichao; Tse, Chris; Leverson, Joel D.; Elmore, Steven W.; Souers, Andrew J.
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Discovery of A-366, a novel small molecule inhibitor that uncovers an unappreciated role for G9a/GLP in the epigenetics of leukemia
err2014-10-01
err0
PREAI
errGuo, Jun; Pliushchev, Marina; He, Yupeng; Ferguson, Debra; Jagadeeswaran, Sujatha; Petros, Andrew; Sun, Chaohong; Soni, Niru B.; Shaw, Bailin; Korepanova, Alla; Maag, David; Sweis, Ramzi; Buchanan, Fritz G.; Michaelides, Michael; Shoemaker, Alex; Tse, Chris; Chiang, Gary G.; Pappano, William N.
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Discovery of a Potent and Selective BCL-XL Inhibitor with in Vivo Activity
err2014-09-08
err286
errOAAI
errTao, Zhi-Fu; Hasvold, Lisa; Wang, Le; Wang, Xilu; Petros, Andrew M.; Park, Chang H.; Boghaert, Erwin R.; Catron, Nathaniel D.; Chen, Jun; Colman, Peter M.; Czabotar, Peter E.; Deshayes, Kurt; Fairbrother, Wayne J.; Flygare, John A.; Hymowitz, Sarah G.; Jin, Sha; Judge, Russell A.; Koehler, Michael F. T.; Kovar, Peter J.; Lessene, Guillaume; Mitten, Michael J.; Ndubaku, Chudi O.; Nimmer, Paul; Purkey, Hans E.; Oleksijew, Anatol; Phillips, Darren C.; Sleebs, Brad E.; Smith, Brian J.; Smith, Morey L.; Tahir, Stephen K.; Watson, Keith G.; Xiao, Yu; Xue, John; Zhang, Haichao; Zobel, Kerry; Rosenberg, Saul H.; Tse, Chris; Leverson, Joel D.; Elmore, Steven W.; Souers, Andrew J.
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Discovery and Development of Potent and Selective Inhibitors of Histone Methyltransferase G9a组蛋白甲基转移酶G9a的有效和选择性抑制剂的发现和开发
err2014-01-02
err181
errOAAI
errSweis, Ramzi F.; Pliushchev, Marina; Brown, Peter J.; Guo, Jun; Li, Fengling; Maag, David; Petros, Andrew M.; Soni, Nirupama B.; Tse, Chris; Vedadi, Masoud; Michaelides, Michael R.; Chiang, Gary G.; Pappano, William N.
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Fragment-based lead discovery: challenges and opportunities
err2011-07-06
err25
PREAI
errSun, Chaohong; Petros, Andrew M.; Hajduk, Philip J.
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Labeled Ligand Displacement: Extending NMR-Based Screening of Protein Targets
err2010-06-24
err10
errOAAI
errSwann, Steven L.; Song, Danying; Sun, Chaohong; Hajduk, Philip J.; Petros, Andrew M.
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Discovery and design of novel HSP90 inhibitors using multiple fragment-based design strategies
err2007-07-11
err114
PREAI
errHuth, Jeffrey R.; Park, Chang; Petros, Andrew M.; Kunzer, Aaron R.; Wendt, Michael D.; Wang, Xilu; Lynch, Christopher L.; Mack, Jamey C.; Swift, Kerry M.; Judge, Russell A.; Chen, Jun; Richardson, Paul L.; Jin, Sha; Tahir, Stephen K.; Matayoshi, Edward D.; Dorwin, Sarah A.; Ladror, Uri S.; Severin, Jean M.; Walter, Karl A.; Bartley, Diane M.; Fesik, Stephen W.; Elmore, Steven W.; Hajduk, Philip J.
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Studies leading to potent, dual inhibitors of bcl-2 and Bcl-xL
err2007-01-26
err372
PREAI
errBruncko, Milan; Oost, Thorsten K.; Belli, Barbara A.; Ding, Hong; Joseph, Mary K.; Kunzer, Aaron; Martineau, Darlene; McClellan, William J.; Mitten, Michael; ng, Shi-Chu Ng; Nimmer, Paul M.; Oltersdorf, Tilman; Park, Cheol-Min; Petros, Andrew M.; Shoemaker, Alexander R.; Song, Xiaohong; Wang, Xilu; Wendt, Michael D.; Zhang, Haichao; Fesik, Stephen W.; Rosenberg, Saul H.; Elmore, Steven W.
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