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收藏What Does It Take to Develop Structurally Complex Molecules by Total Synthesis? Rapid Process Development and GMP Manufacturing of E7130 Drug Substance for First-in-Human Clinical Study
Sasaki, Takeo; Yahata, Kenzo; Isomura, Minetaka; Ohashi, Isao; Fukuyama, Takashi; Miyashita, Yusuke; Watanabe, Yuzo; Murai, Norio; Matsuda, Masaaki; Kamada, Atsushi; Kaburagi, Yosuke; Kira, Kazunobu; Iso, Kentaro; Sato, Yuki; Matsuura, Fumiyoshi; Matsumoto, Yasunobu; Azuma, Hiroshi; Iida, Daisuke; Ishida, Tasuku; Itano, Wataru; Nagao, Satoshi; Seki, Masashi; Yamamoto, Akihiko; Yamamoto, Yuji; Yoneda, Naoki; Matsukura, Masayuki; Asano, Osamu; Kayano, Akio; Tagami, Katsuya; Owa, Takashi; Kishi, Yoshito
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收藏Ten-Gram-Scale Total Synthesis of the Anticancer Drug Candidate E7130 to Supply Clinical Trials
Kaburagi, Yosuke; Kira, Kazunobu; Yahata, Kenzo; Iso, Kentaro; Sato, Yuki; Matsuura, Fumiyoshi; Ohashi, Isao; Matsumoto, Yasunobu; Isomura, Minetaka; Sasaki, Takeo; Fukuyama, Takashi; Miyashita, Yusuke; Azuma, Hiroshi; Iida, Daisuke; Ishida, Tasuku; Itano, Wataru; Matsuda, Masaaki; Matsukura, Masayuki; Murai, Norio; Nagao, Satoshi; Seki, Masashi; Yamamoto, Akihiko; Yamamoto, Yuji; Yoneda, Naoki; Watanabe, Yuzo; Kamada, Atsushi; Kayano, Akio; Tagami, Katsuya; Asano, Osamu; Owa, Takashi; Kishi, Yoshito
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收藏Mechanism of action analysis of anti-CAF activity of E7130, a novel tumor-microenvironment ameliorator
Abe, Takanori; Kawano, Satoshi; Ito, Ken; Yahata, Kenzo; Kira, Kazunobu; Akagi, Tsuyoshi; Asano, Makoto; Iso, Kentaro; Sato, Yuki; Matsuura, Fumiyoshi; Ohashi, Isao; Matsumoto, Yasunobu; Isomura, Minetaka; Sasaki, Takeo; Fukuyama, Takashi; Miyashita, Yusuke; Kaburagi, Yosuke; Yokoi, Akira; Asano, Osamu; Owa, Takashi; Kishi, Yoshito
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收藏E7130 derived from total synthesis of halichondrin as a novel tumor-microenvironment ameliorator
Kawano, Satoshi; Abe, Takanori; Ito, Ken; Yahata, Kenzo; Kira, Kazunobu; Akagi, Tsuyoshi; Asano, Makoto; Iso, Kentaro; Sato, Yuki; Matsuura, Fumiyoshi; Ohashi, Isao; Matsumoto, Yasunobu; Isomura, Minetaka; Sasaki, Takeo; Fukuyama, Takashi; Miyashita, Yusuke; Kaburagi, Yosuke; Yokoi, Akira; Asano, Osamu; Owa, Takashi; Kishi, Yoshito
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收藏A landmark in drug discovery based on complex natural product synthesis
Kawano, Satoshi; Ito, Ken; Yahata, Kenzo; Kira, Kazunobu; Abe, Takanori; Akagi, Tsuyoshi; Asano, Makoto; Iso, Kentaro; Sato, Yuki; Matsuura, Fumiyoshi; Ohashi, Isao; Matsumoto, Yasunobu; Isomura, Minetaka; Sasaki, Takeo; Fukuyama, Takashi; Miyashita, Yusuke; Kaburagi, Yosuke; Yokoi, Akira; Asano, Osamu; Owa, Takashi; Kishi, Yoshito
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收藏Simple, Rapid Mycobacterium ulcerans Disease Diagnosis from Clinical Samples by Fluorescence of Mycolactone on Thin Layer Chromatography
Wadagni, Anita; Frimpong, Michael; Phanzu, Delphin Mavinga; Ablordey, Anthony; Kacou, Emmanuel; Gbedevi, Mirabelle; Marion, Estelle; Xing, Yalan; Babu, Vaddela Sudheer; Phillips, Richard Odame; Wansbrough-Jones, Mark; Kishi, Yoshito; Asiedu, Kingsley
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