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Philippe Delagrange

cnrs - institute of chemistry (inc)

53H指数
235论文数
1.0W被引数
收录论文 120
发表时间
Efficient axonal transport of endolysosomes relies on the balanced ratio of microtubule tyrosination and detyrosination
err2024-04-30
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errOAAI
errKonietzny, Anja; Han, Yuhao; Popp, Yannes; van Bommel, Bas; Sharma, Aditi; Delagrange, Philippe; Arbez, Nicolas; Moutin, Marie-Jo; Peris, Leticia; Mikhaylova, Marina
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Mapping the Melatonin Receptor. 8. Selective MT2 Agonists Derived from 5,6-Dihydroindolo[2,1-a]isoquinolines and Related Systems绘制褪黑激素受体。8.源自5,6-二氢吲哚并 [2,1-a] 异喹啉和相关系统的选择性MT2激动剂
err2022-05-09
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errOAAI
errTsotinis, Andrew; Afroudakis, Pandelis A.; Papanastasiou, Ioannis P.; Sakellaropoulou, Aikaterini; Boniakou, Marina; Komiotis, Dimitri; Garratt, Peter J.; Delagrange, Philippe; Bocianowska-Zbrog, Alina; Sugden, David
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Tubulin tyrosination regulates synaptic function and is disrupted in Alzheimer's disease
errBRAIN
IF11.7
err2022-02-11
err32
errOAAI
errPeris, Leticia; Parato, Julie; Qu, Xiaoyi; Soleilhac, Jean-Marc; Lante, Fabien; Kumar, Atul; Pero, Maria Elena; Martinez-Hernandez, Jose; Corrao, Charlotte; Falivelli, Giulia; Payet, Floriane; Gory-Faure, Sylvie; Bosc, Christophe; Ramirez, Marian Blanca; Sproul, Andrew; Brocard, Jacques; Di Cara, Benjamin; Delagrange, Philippe; Buisson, Alain; Goldberg, Yves; Moutin, Marie-Jo; Bartolini, Francesca; Andrieux, Annie
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Synthesis and SAR Studies of Isoquinoline and Tetrahydroisoquinoline Derivatives as Melatonin Receptor Ligands
err2021-12-01
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errOAAI
errEttaoussi, Mohamed; Laversin, Amelie; Vreulz, Brandon; Rami, Marouane; Lebegue, Nicolas; Delagrange, Philippe; Caignard, Daniel Henri; Melnyk, Patricia; Liberelle, Maxime; Yous, Said
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Primary role for melatonin MT2 receptors in the regulation of anhedonia and circadian temperature rhythm
err2021-03-01
err7
PREAI
errBorja Belloch, Francisco; Beltran, Elena; Venzala, Elisabeth; Montalt-Tordera, Javier; Diaz-Perdigon, Teresa; Cecon, Erika; Puerta, Elena; Delagrange, Philippe; Maria Tordera, Rosa
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Pharmacological evidence for transactivation within melatonin MT2 and serotonin 5-HT2C receptor heteromers in mouse brain
err2020-11-06
err17
PREAI
errGerbier, Romain; Ndiaye-Lobry, Delphine; Martinez de Morentin, Pablo B.; Cecon, Erika; Heisler, Lora K.; Delagrange, Philippe; Gbahou, Florence; Jockers, Ralf
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Melatonin MT2 receptors modulate anhedonic behaviour and circadian temperature rhythm
err2020-11-01
err0
PREAI
errTordera, R.; Belloch, B.; Beltran, E.; Venzala, E.; Montalt, J.; Diaz-Perdigon, T.; Cecon, E.; Puerta, E.; Delagrange, P.
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Quinazoline and phthalazine derivatives as novel melatonin receptor ligands analogues of agomelatine
err2020-03-01
err15
errOAAI
errBolteau, Raphael; Descamps, Florian; Ettaoussi, Mohamed; Caignard, Daniel H.; Delagrange, Philippe; Melnyk, Patricia; Yous, Said
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GPR50-Ctail cleavage and nuclear translocation: a new signal transduction mode for G protein-coupled receptorsGPR50-Ctail裂解和核易位: g蛋白偶联受体的新信号转导模式
err2020-01-03
err14
errOAAI
errAhmad, Raise; Lahuna, Olivier; Sidibe, Anissa; Daulat, Avais; Zhang, Qiang; Luka, Marine; Guillaume, Jean-Luc; Gallet, Sarah; Guillonneau, Francois; Hamroune, Juliette; Polo, Sophie; Prevot, Vincent; Delagrange, Philippe; Dam, Julie; Jockers, Ralf
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Quantitative assessment of oligomeric amyloid β peptide binding to α7 nicotinic receptor
err2019-05-20
err24
errOAAI
errCecon, Erika; Dam, Julie; Luka, Marine; Gautier, Clement; Chollet, Anne-Marie; Delagrange, Philippe; Danober, Laurence; Jockers, Ralf
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Detection of recombinant and endogenous mouse melatonin receptors by monoclonal antibodies targeting the C-terminal domain
err2019-01-17
err17
PREAI
errCecon, Erika; Ivanova, Anna; Luka, Marine; Gbahou, Florence; Friederich, Anne; Guillaume, Jean-Luc; Keller, Patrick; Knoch, Klaus; Ahmad, Raise; Delagrange, Philippe; Solimena, Michele; Jockers, Ralf
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Melatonin receptors limit dopamine reuptake by regulating dopamine transporter cell-surface exposure
err2018-07-24
err14
errOAAI
errBenleulmi-Chaachoua, Abla; Hegron, Alan; Le Boulch, Marine; Karamitri, Angeliki; Wierzbicka, Marta; Wong, Victoria; Stagljar, Igor; Delagrange, Philippe; Ahmad, Raise; Jockers, Ralf
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Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands
err2018-03-29
err15
errOAAI
errRivara, Silvia; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Caignard, Daniel-Henri; Delagrange, Philippe; Collina, Simona; Lucini, Valeria; Scaglione, Francesco; Furiassi, Lucia; Mari, Michele; Lucarini, Simone; Bedini, Annalida; Spadoni, Gilberto
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The orphan GPR50 receptor promotes constitutive TGFβ receptor signaling and protects against cancer development
err2018-03-23
err30
errOAAI
errWojciech, Stefanie; Ahmad, Raise; Belaid-Choucair, Zakia; Journe, Anne-Sophie; Gallet, Sarah; Dam, Julie; Daulat, Avais; Ndiaye-Lobry, Delphine; Lahuna, Olivier; Karamitri, Angeliki; Guillaume, Jean-Luc; Do Cruzeiro, Marcio; Guillonneau, Francois; Saade, Anastasia; Clement, Nathalie; Courivaud, Thomas; Kaabi, Nawel; Tadagaki, Kenjiro; Delagrange, Philippe; Prevot, Vincent; Hermine, Olivier; Prunier, Celine; Jockers, Ralf
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Synthesis and biological evaluation of new naphtho- and quinolinocyclopentane derivatives as potent melatoninergic (MT1/MT2) and serotoninergic (5-HT2c) dual ligands
err2017-12-01
err13
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errDuroux, Romain; Rami, Marouan; Landagaray, Elodie; Ettaoussi, Mohamed; Caignard, Daniel-Henri; Delagrange, Philippe; Melnyk, Patricia; Yous, Said
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Importance of the second extracellular loop for melatonin MT1 receptor function and absence of melatonin binding in GPR50
err2017-10-27
err18
errOAAI
errClement, Nathalie; Renault, Nicolas; Guillaume, Jean-Luc; Cecon, Erika; Journe, Anne-Sophie; Laurent, Xavier; Tadagaki, Kenjiro; Coge, Francis; Gohier, Arnaud; Delagrange, Philippe; Chavatte, Philippe; Jockers, Ralf
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Design and validation of the first cell-impermeant melatonin receptor agonist
err2017-06-11
err46
errOAAI
errGbahou, Florence; Cecon, Erika; Viault, Guillaume; Gerbier, Romain; Jean-Alphonse, Frederic; Karamitri, Angeliki; Guillaumet, Gerald; Delagrange, Philippe; Friedlander, Robert M.; Vilardaga, Jean-Pierre; Suzenet, Franck; Jockers, Ralf
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New quinolinic derivatives as melatonergic ligands: Synthesis and pharmacological evaluation
err2017-02-01
err10
PREAI
errLandagaray, Elodie; Ettaoussi, Mohamed; Rami, Marouan; Boutin, Jean A.; Caignard, Daniel-Henri; Delagrange, Philippe; Melnyk, Patricia; Berthelot, Pascal; Yous, Said
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Update on melatonin receptors: IUPHAR Review 20
err2016-08-08
err323
errOAAI
errJockers, Ralf; Delagrange, Philippe; Dubocovich, Margarita L.; Markus, Regina P.; Renault, Nicolas; Tosini, Gianluca; Cecon, Erika; Zlotos, Darius P.
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Synthesis of 2-arylfuro[3,2-b]pyridines: Effect of the C2-aryl group on melatoninergic activity
err2016-02-01
err9
PREAI
errCouhert, Audrey; Delagrange, Philippe; Caignard, Daniel-Henri; Chartier, Agnes; Suzenet, Franck; Guillaumet, Gerald
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