未登录Efficient axonal transport of endolysosomes relies on the balanced ratio of microtubule tyrosination and detyrosination
Konietzny, Anja; Han, Yuhao; Popp, Yannes; van Bommel, Bas; Sharma, Aditi; Delagrange, Philippe; Arbez, Nicolas; Moutin, Marie-Jo; Peris, Leticia; Mikhaylova, Marina
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收藏Mapping the Melatonin Receptor. 8. Selective MT2 Agonists Derived from 5,6-Dihydroindolo[2,1-a]isoquinolines and Related Systems绘制褪黑激素受体。8.源自5,6-二氢吲哚并 [2,1-a] 异喹啉和相关系统的选择性MT2激动剂
Tsotinis, Andrew; Afroudakis, Pandelis A.; Papanastasiou, Ioannis P.; Sakellaropoulou, Aikaterini; Boniakou, Marina; Komiotis, Dimitri; Garratt, Peter J.; Delagrange, Philippe; Bocianowska-Zbrog, Alina; Sugden, David
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收藏Tubulin tyrosination regulates synaptic function and is disrupted in Alzheimer's disease
Peris, Leticia; Parato, Julie; Qu, Xiaoyi; Soleilhac, Jean-Marc; Lante, Fabien; Kumar, Atul; Pero, Maria Elena; Martinez-Hernandez, Jose; Corrao, Charlotte; Falivelli, Giulia; Payet, Floriane; Gory-Faure, Sylvie; Bosc, Christophe; Ramirez, Marian Blanca; Sproul, Andrew; Brocard, Jacques; Di Cara, Benjamin; Delagrange, Philippe; Buisson, Alain; Goldberg, Yves; Moutin, Marie-Jo; Bartolini, Francesca; Andrieux, Annie
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收藏Synthesis and SAR Studies of Isoquinoline and Tetrahydroisoquinoline Derivatives as Melatonin Receptor Ligands
Ettaoussi, Mohamed; Laversin, Amelie; Vreulz, Brandon; Rami, Marouane; Lebegue, Nicolas; Delagrange, Philippe; Caignard, Daniel Henri; Melnyk, Patricia; Liberelle, Maxime; Yous, Said
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收藏GPR50-Ctail cleavage and nuclear translocation: a new signal transduction mode for G protein-coupled receptorsGPR50-Ctail裂解和核易位: g蛋白偶联受体的新信号转导模式
Ahmad, Raise; Lahuna, Olivier; Sidibe, Anissa; Daulat, Avais; Zhang, Qiang; Luka, Marine; Guillaume, Jean-Luc; Gallet, Sarah; Guillonneau, Francois; Hamroune, Juliette; Polo, Sophie; Prevot, Vincent; Delagrange, Philippe; Dam, Julie; Jockers, Ralf
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收藏Detection of recombinant and endogenous mouse melatonin receptors by monoclonal antibodies targeting the C-terminal domain
Cecon, Erika; Ivanova, Anna; Luka, Marine; Gbahou, Florence; Friederich, Anne; Guillaume, Jean-Luc; Keller, Patrick; Knoch, Klaus; Ahmad, Raise; Delagrange, Philippe; Solimena, Michele; Jockers, Ralf
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收藏Melatonin receptors limit dopamine reuptake by regulating dopamine transporter cell-surface exposure
Benleulmi-Chaachoua, Abla; Hegron, Alan; Le Boulch, Marine; Karamitri, Angeliki; Wierzbicka, Marta; Wong, Victoria; Stagljar, Igor; Delagrange, Philippe; Ahmad, Raise; Jockers, Ralf
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收藏Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands
Rivara, Silvia; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Caignard, Daniel-Henri; Delagrange, Philippe; Collina, Simona; Lucini, Valeria; Scaglione, Francesco; Furiassi, Lucia; Mari, Michele; Lucarini, Simone; Bedini, Annalida; Spadoni, Gilberto
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收藏The orphan GPR50 receptor promotes constitutive TGFβ receptor signaling and protects against cancer development
Wojciech, Stefanie; Ahmad, Raise; Belaid-Choucair, Zakia; Journe, Anne-Sophie; Gallet, Sarah; Dam, Julie; Daulat, Avais; Ndiaye-Lobry, Delphine; Lahuna, Olivier; Karamitri, Angeliki; Guillaume, Jean-Luc; Do Cruzeiro, Marcio; Guillonneau, Francois; Saade, Anastasia; Clement, Nathalie; Courivaud, Thomas; Kaabi, Nawel; Tadagaki, Kenjiro; Delagrange, Philippe; Prevot, Vincent; Hermine, Olivier; Prunier, Celine; Jockers, Ralf
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收藏Importance of the second extracellular loop for melatonin MT1 receptor function and absence of melatonin binding in GPR50
Clement, Nathalie; Renault, Nicolas; Guillaume, Jean-Luc; Cecon, Erika; Journe, Anne-Sophie; Laurent, Xavier; Tadagaki, Kenjiro; Coge, Francis; Gohier, Arnaud; Delagrange, Philippe; Chavatte, Philippe; Jockers, Ralf
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收藏Design and validation of the first cell-impermeant melatonin receptor agonist
Gbahou, Florence; Cecon, Erika; Viault, Guillaume; Gerbier, Romain; Jean-Alphonse, Frederic; Karamitri, Angeliki; Guillaumet, Gerald; Delagrange, Philippe; Friedlander, Robert M.; Vilardaga, Jean-Pierre; Suzenet, Franck; Jockers, Ralf
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