Gérald Guillaumet - Publications, H-index & Citations

Gérald Guillaumet

universite d orleans

41H指数

664论文数

7.9K被引数

收录论文 97

发表时间

Targeting 5-HT7 Receptor with Biased Ligands to Alleviate Pain and Spinal Neuroinflammation 利用偏向性配体靶向5-HT7受体以缓解疼痛和脊髓神经炎症

ACS Chemical Neuroscience

IF3.9

2026-05-29

PREAI

Fahima Madouri; Cyril Guimpied; Enora Pigeon; Nadège Hervouet; David Gosset; Pascal Auzou; Mélanie Kremer; Quentin Leboulleux; Marie-Aude Hiebel; Julie Le Bescont; Gérald Guillaumet; Franck Suzenet; Patrick Baril; Raphaël Serreau; Séverine Morisset-Lopez

Regioselective Copper(I)-Catalyzed Direct C(3)-H (Hetero)arylation of 6-(Hetero)arylated 1,2,4-Triazolo[4,3-b]pyridazines: Ligand-Free Approach

JOURNAL OF ORGANIC CHEMISTRY

IF3.6

2024-11-25

PREAI

Hourma, Chaimae; Jismy, Badr; Blancou, Wafa; Driowya, Mohsine; Bougrin, Khalid; Guillaumet, Gerald; Abarbri, Mohamed

Regioselective C6-Arylation of Thieno[3,2-c]pyrazole Heterocycles with Aryl Iodides 噻吩并 [3，2-c] 吡唑杂环与芳基碘的区域选择性C6-Arylation

ADVANCED SYNTHESIS & CATALYSIS

IF4

2024-05-23

PREAI

Lfakir, Noura Ait; Jismy, Badr; Guillaumet, Gerald; Akssira, Mohamed; El Hakmaoui, Ahmed; Guillot, Regis; Tikad, Abdellatif; Abarbri, Mohamed

Design, Synthesis, Computational Studies, and Anti-Proliferative Evaluation of Novel Ethacrynic Acid Derivatives Containing Nitrogen Heterocycle, Urea, and Thiourea Moieties as Anticancer Agents

MOLECULES

IF4.6

2024-03-23

OAAI

El Abbouchi, Abdelmoula; Mkhayar, Khaoula; Elkhattabi, Souad; El Brahmi, Nabil; Hiebel, Marie-Aude; Bignon, Jerome; Guillaumet, Gerald; Suzenet, Franck; El Kazzouli, Said

New and promising type of leukotriene B4 (LTB4) antagonists based on the 1,4-benzodioxine structure

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2023-06-01

PREAI

Bouissane, Latifa; Khouili, Mostafa; Coudert, Gerard; Pujol, M. Dolors; Guillaumet, Gerald

Improvement of the Chemical Reactivity of Michael Acceptor of Ethacrynic Acid Correlates with Antiproliferative Activities

MOLECULES

IF4.6

2023-01-16

OAAI

El Abbouchi, Abdelmoula; El Brahmi, Nabil; Hiebel, Marie-Aude; Ghammaz, Hamza; El Fahime, Elmostafa; Bignon, Jerome; Guillaumet, Gerald; Suzenet, Franck; El Kazzouli, Said

Synthesis, Anticancer Activities and Molecular Docking Studies of a Novel Class of 2-Phenyl-5,6,7,8-tetrahydroimidazo [1,2-b]pyridazine Derivatives Bearing Sulfonamides

MOLECULES

IF4.6

2022-08-17

OAAI

Bourzikat, Otmane; El Abbouchi, Abdelmoula; Ghammaz, Hamza; El Brahmi, Nabil; El Fahime, Elmostfa; Paris, Arnaud; Daniellou, Richard; Suzenet, Franck; Guillaumet, Gerald; El Kazzouli, Said

Serodolin, a β-arrestin-biased ligand of 5-HT7 receptor, attenuates pain-related behaviors

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

IF9.1

2022-05-20

OAAI

El Khamlichi, Chayma; Reverchon, Flora; Hervouet-Coste, Nadege; Robin, Elodie; Chopin, Nicolas; Deau, Emmanuel; Madouri, Fahima; Guimpied, Cyril; Colas, Cyril; Menuet, Arnaud; Inoue, Asuka; Bojarski, Andrzej J.; Guillaumet, Gerald; Suzenet, Franck; Reiter, Eric; Morisset-Lopez, Severine

Regioselective C-H Functionalization of the Six-Membered Ring of the 6,5-Fused Heterocyclic Systems: An Overview

MOLECULES

IF4.6

2021-09-23

OAAI

Faarasse, Soukaina; El Brahmi, Nabil; Guillaumet, Gerald; El Kazzouli, Said

Palladium-Catalyzed Regioselective C-H Arylation of 4-Azaindazole at C3, C5 and C7 Positions

ADVANCED SYNTHESIS & CATALYSIS

IF4

2021-03-19

OAAI

Faarasse, Soukaina; El Kazzouli, Said; Bourzikat, Otmane; Bourg, Stephane; Aci-Seche, Samia; Bonnet, Pascal; Suzenet, Franck; Guillaumet, Gerald

On Water Palladium Catalyzed Direct Arylation of 1H-Indazole and 1H-7-Azaindazole

MOLECULES

IF4.6

2020-06-18

OAAI

Gambouz, Khadija; El Abbouchi, Abdelmoula; Nassiri, Sarah; Suzenet, Franck; Bousmina, Mostapha; Akssira, Mohamed; Guillaumet, Gerald; El Kazzouli, Said

Efficient Access to 3,5-Disubstituted 7-(Trifluoromethyl)pyrazolo[1,5-a]pyrimidines Involving SNAr and Suzuki Cross-Coupling Reactions

MOLECULES

IF4.6

2020-04-28

OAAI

Jismy, Badr; Tikad, Abdellatif; Akssira, Mohamed; Guillaumet, Gerald; Abarbri, Mohamed

Intramolecular Metal-Free N-N Bond Formation with Heteroaromatic Amines: Mild Access to Fused-Triazapentalene Derivatives 与杂芳胺形成分子内无金属的n-n键: 轻度获得稠合三氮杂戊烯衍生物

CHEMISTRY-A EUROPEAN JOURNAL

IF3.7

2020-01-23

PREAI

Daniel, Matthieu; Hiebel, Marie-Aude; Guillaumet, Gerald; Pasquinet, Eric; Suzenet, Franck

Development of Novel and Efficient Processes for the Synthesis of 5-Amino and 5-Iminoimidazo[1,2-a] imidazoles via Three-Component Reaction Catalyzed by Zirconium(IV) Chloride

FRONTIERS IN CHEMISTRY

IF4.2

2019-07-08

OAAI

Driowya, Mohsine; Guillot, Regis; Bonnet, Pascal; Guillaumet, Gerald

Copper-Assisted Synthesis of Novel Pyrazolo[3,4-d]thiazoles

CHEMCATCHEM

IF3.9

2019-07-04

PREAI

Ostache, Nicu-Cosmin; Hiebel, Marie-Aude; Finaru, Adriana-Luminita; Guillaumet, Gerald; Suzenet, Franck

S29434, a Quinone Reductase 2 Inhibitor: Main Biochemical and Cellular Characterization

MOLECULAR PHARMACOLOGY

IF3

2019-03-01

OAAI

Boutin, Jean A.; Bouillaud, Frederic; Janda, Elzbieta; Gacsalyi, Istvan; Guillaumet, Gerald; Hirsch, Etienne C.; Kane, Daniel A.; Nepveu, Francoise; Reybier, Karine; Dupuis, Philippe; Bertrand, Marc; Chhour, Monivan; Le Diguarher, Thierry; Antoine, Mathias; Brebner, Karen; Da Costa, Herve; Ducrot, Pierre; Giganti, Adeline; Goswami, Vishalgiri; Guedouari, Hala; Michel, Patrick P.; Patel, Aakash; Paysant, Jerome; Stojko, Johann; Viaud-Massuard, Marie-Claude; Ferry, Gilles

An original class of small sized molecules as versatile fluorescent probes for cellular imaging

CHEMICAL COMMUNICATIONS

IF4.2

2019-01-01

OAAI

Sirbu, Doina; Diharce, Julien; Martinic, Ivana; Chopin, Nicolas; Eliseeva, Svetlana V.; Guillaumet, Gerald; Petoud, Stephane; Bonnet, Pascal; Suzenet, Franck

Regioselective Synthesis of New 2,4-(Het)aryl-3H-pyrido[1′,2′:1,5]pyrazolo[4,3-d]pyrimidines Involving Palladium-Catalyzed Cross-Coupling Reactions

MOLECULES

IF4.6

2018-10-23

OAAI

Ejjoummany, Abdelaziz; Belaroussi, Rabia; El Hakmaoui, Ahmed; Akssira, Mohamed; Guillaumet, Gerald; Buron, Frederic; Routier, Sylvain

Palladium-Catalyzed C3-Arylations of 1H- and 2H-Pyrazolo[4,3-b]pyridines on Water

JOURNAL OF ORGANIC CHEMISTRY

IF3.6

2018-09-21

PREAI

Faarasse, Soukaina; El Kazzouli, Said; Suzenet, Franck; Guillaumet, Gerald

Efficient synthesis and first regioselective C-6 direct arylation of imidazo[2,1-c][1,2,4]triazine scaffold and their evaluation in H2O2-induced oxidative stress

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2018-02-01

PREAI

Loubidi, Mohammed; Jouha, Jabrane; Tber, Zahira; Khouili, Mostafa; Suzenet, Franck; Akssira, Mohamed; Erdogan, Mumin Alper; Kose, Fadime Aydin; Dagci, Taner; Armagan, Guliz; Saso, Luciano; Guillaumet, Gerald

研究方向