未登录 Structural and functional properties of the Kunitz-type and C-terminal domains of Amblyomin-X supporting its antitumor activity Morais, K. L. P.; Ciccone, L.; Stura, E.; Alvarez-Flores, M. P.; Mourier, G.; Driessche, M. Vanden; Sciani, J. M.; Iqbal, A.; Kalil, S. P.; Pereira, G. J.; Marques-Porto, R.; Cunegundes, P.; Juliano, L.; Servent, D.; Chudzinski-Tavassi, A. M. 分享 收藏
Evaluation of the Spider (Phlogiellus genus) Phlotoxin 1 and Synthetic Variants as Antinociceptive Drug Candidates Goncalves, Tania C.; Lesport, Pierre; Kuylle, Sarah; Stura, Enrico; Ciolek, Justyna; Mourier, Gilles; Servent, Denis; Bourinet, Emmanuel; Benoit, Evelyne; Gilles, Nicolas 分享 收藏
分享 收藏
分享 收藏
Development of Thioaryl-Based Matrix Metalloproteinase-12 Inhibitors with Alternative Zinc-Binding Groups: Synthesis, Potentiometric, NMR, and Crystallographic Studies Nuti, Elisa; Cuffaro, Doretta; Bernardini, Elisa; Camodeca, Caterina; Panelli, Laura; Chaves, Silvia; Ciccone, Lidia; Tepshi, Livia; Vera, Laura; Orlandini, Elisabetta; Nencetti, Susanna; Stura, Enrico A.; Santos, M. Amelia; Dive, Vincent; Rossello, Armando 分享 收藏
Green mamba peptide targets type-2 vasopressin receptor against polycystic kidney disease 绿色曼巴肽靶向2型加压素受体对抗多囊肾病 Ciolek, Justyna; Reinfrank, Helen; Quinton, Loic; Viengchareun, Say; Stura, Enrico A.; Vera, Laura; Sigismeau, Sabrina; Mouillac, Bernard; Orcel, Helene; Peigneur, Steve; Tytgat, Jan; Droctove, Laura; Beau, Fabrice; Nevoux, Jerome; Lombes, Marc; Mourier, Gilles; De Pauw, Edwin; Servent, Denis; Mendre, Christiane; Witzgall, Ralph; Gilles, Nicolas 分享 收藏
分享 收藏
Bifunctional Inhibitors as a New Tool To Reduce Cancer Cell Invasion by Impairing MMP-9 Homodimerization Nuti, Elisa; Rosalia, Lea; Cuffaro, Doretta; Camodeca, Caterina; Giacomelli, Chiara; Da Pozzo, Eleonora; Tuccinardi, Tiziano; Costa, Barbara; Antoni, Claudia; Vera, Laura; Ciccone, Lidia; Orlandin, Elisabetta; Nencetti, Susanna; Dive, Vincent; Martini, Claudia; Stura, Enrico A.; Rossello, Armando 分享 收藏
分享 收藏
Highly selective inhibition of myosin motors provides the basis of potential therapeutic application Sirigu, Serena; Hartman, James J.; Planelles-Herrero, Vicente Jose; Ropars, Virginie; Clancy, Sheila; Wang, Xi; Chuang, Grace; Qian, Xiangping; Lu, Pu-Ping; Barrett, Edward; Rudolph, Karin; Royer, Christopher; Morgan, Bradley P.; Stura, Enrico A.; Malik, Fady I.; Houdusse, Anne M. 分享 收藏
Synthesis and in Vitro and in Vivo Evaluation of MMP-12 Selective Optical Probes Bordenave, Thomas; Helle, Marion; Beau, Fabrice; Georgiadis, Dimitris; Tepshi, Livia; Bernes, Mylene; Ye, Yunpeng; Levenez, Laure; Poquet, Enora; Nozach, Herve; Razavian, Mahmoud; Toczek, Jakub; Stura, Enrico A.; Dive, Vincent; SadeghiP, Mehran M.; Devel, Laurent 分享 收藏
分享 收藏
Sugar-Based Arylsulfonamide Carboxylates as Selective and Water-Soluble Matrix Metalloproteinase-12 Inhibitors Nuti, Elisa; Cuffaro, Doretta; D'Andrea, Felicia; Rosalia, Lea; Tepshi, Livia; Fabbi, Marina; Carbotti, Grazia; Ferrini, Silvano; Santamaria, Salvatore; Camodeca, Caterina; Ciccone, Lidia; Orlandini, Elisabetta; Nencetti, Susanna; Stura, Enrico A.; Dive, Vincent; Rossello, Armando 分享 收藏
分享 收藏
分享 收藏
分享 收藏
Mambalgin-1 Pain-relieving Peptide, Stepwise Solid-phase Synthesis, Crystal Structure, and Functional Domain for Acid-sensing Ion Channel 1a Inhibition Mourier, Gilles; Salinas, Miguel; Kessler, Pascal; Stura, Enrico A.; Leblanc, Mathieu; Tepshi, Livia; Besson, Thomas; Diochot, Sylvie; Baron, Anne; Douguet, Dominique; Lingueglia, Eric; Servent, Denis 分享 收藏
N-O-Isopropyl Sulfonamido-Based Hydroxamates as Matrix Metalloproteinase Inhibitors: Hit Selection and in Vivo Antiangiogenic Activity Nuti, Elisa; Cantelmo, Anna Rita; Gallo, Cristina; Bruno, Antonino; Bassani, Barbara; Camodeca, Caterina; Tuccinardi, Tiziano; Vera, Laura; Orlandini, Elisabetta; Nencetti, Susanna; Stura, Enrico A.; Martinelli, Adriano; Dive, Vincent; Albini, Adriana; Rossello, Armando 分享 收藏
分享 收藏
分享 收藏