Fabrice Piu - Publications, H-index & Citations

Fabrice Piu

acadia pharmaceuticals inc.

24H指数

61论文数

2.3K被引数

收录论文 20

发表时间

CHARACTERIZATION OF THE JAK INHIBITORS TOFACITINIB AND UPADACITINIB IN HUMAN PRIMARY CELL 3D MODELS OF CROHN'S DISEASE AND ULCERATIVE COLITIS JAK抑制剂的表征：托法替尼和乌帕替尼在克罗恩病和溃疡性结肠炎的人源原代细胞三维模型中

INFLAMMATORY BOWEL DISEASES

IF4.3

2025-02-28

PREAI

Dudum, Rachel; Olson, Payton; Toohey, Cole; Gervacio, Sherwin; Rosette, Caridad; Piu, Fabrice

AP-1 repressor protein JDP-2: Inhibition of UV-mediated apoptosis through p53 down-regulation

MOLECULAR AND CELLULAR BIOLOGY

IF2.7

2023-03-28

OAAI

Piu, F; Aronheim, A; Katz, S; Karin, M

Comparison of the Pharmacokinetic Properties of Triamcinolone and Dexamethasone for Local Therapy of the Inner Ear

FRONTIERS IN CELLULAR NEUROSCIENCE

IF4

2019-07-30

OAAI

Salt, Alec Nicholas; Hartsock, Jared James; Hou, Jennifer; Piu, Fabrice

Local Drug Delivery for the Treatment of Neurotology Disorders 局部给药治疗神经系统疾病

FRONTIERS IN CELLULAR NEUROSCIENCE

IF4

2019-06-03

OAAI

Piu, Fabrice; Bishop, Kathie M.

Identification of the Antiarrhythmic Drugs Amiodarone and Lorcainide as Potent H3 Histamine Receptor Inverse Agonists

JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

IF3.8

2014-01-01

PREAI

Del Tredici, Andria L.; Ma, Jian-Nong; Piu, Fabrice; Burstein, Ethan S.

Discovery of potential antipsychotic agents possessing pro-cognitive properties

NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY

IF3.1

2011-11-15

PREAI

Lameh, Jelveh; McFarland, Krista; Ohlsson, Jorgen; Ek, Fredrik; Piu, Fabrice; Burstein, Ethan S.; Tabatabaei, Ali; Olsson, Roger; Bradley, Stefania Risso; Bonhaus, Douglas W.

Synthesis, Structure-Activity Relationships, and Characterization of Novel Nonsteroidal and Selective Androgen Receptor Modulators

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2009-10-26

PREAI

Schlienger, Nathalie; Lund, Birgitte W.; Pawlas, Jan; Badalassi, Fabrizio; Bertozzi, Fabio; Lewinsky, Rasmus; Fejzic, Alma; Thygesen, Mikkel B.; Tabatabaei, Ali; Bradley, Stefania Risso; Gardell, Luis R.; Piu, Fabrice; Olsson, Roger

Synthesis and Evaluation of Dibenzothiazepines: A Novel Class of Selective Cannabinoid-1 Receptor Inverse Agonists

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2009-03-11

PREAI

Pettersson, Hanna; Bulow, Anne; Ek, Fredrik; Jensen, Jacob; Ottesen, Lars K.; Fejzic, Alma; Ma, Jian-Nong; Del Tredici, Andria L.; Currier, Erika A.; Gardell, Luis R.; Tabatabaei, Ali; Craig, Darren; McFarland, Krista; Ott, Thomas R.; Piu, Fabrice; Burstein, Ethan S.; Olsson, Roger

Design, Synthesis, and Structure-Activity Analysis of Isoform-Selective Retinoic Acid Receptor β Ligands

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2009-02-24

PREAI

Lund, Birgitte W.; Knapp, Anne Eeg; Piu, Fabrice; Gauthier, Natalie K.; Begtrup, Mikael; Hacksell, Uli; Olsson, Roger

Identification of novel selective V2 receptor non-peptide agonists

BIOCHEMICAL PHARMACOLOGY

IF5.6

2008-10-01

PREAI

Del Tredici, Andria L.; Vanover, Kim E.; Knapp, Anne E.; Bertozzi, Sine M.; Nash, Norman R.; Burstein, Ethan S.; Lameh, Jelveh; Currier, Erika A.; Davis, Robert E.; Brann, Mark R.; Mohell, Nina; Olsson, Roger; Piu, Fabrice

Differential modulation of inflammatory pain by a selective estrogen receptor beta agonist

EUROPEAN JOURNAL OF PHARMACOLOGY

IF4.7

2008-09-01

PREAI

Gardell, Luis R.; Hyldtoft, Lene; Del Tredici, Andria L.; Andersen, Carsten B.; Fairbairn, Luke C.; Lund, Birgitte W.; Gustafsson, Magnus; Brann, Mark R.; Olsson, Roger; Piu, Fabrice

Broad modulation of neuropathic pain states by a selective estrogen receptor beta agonist

EUROPEAN JOURNAL OF PHARMACOLOGY

IF4.7

2008-08-01

PREAI

Piu, Fabrice; Cheevers, Cindy; Hyldtoft, Lene; Gardell, Luis R.; Del Tredici, Andria L.; Andersen, Carsten B.; Fairbairn, Luke C.; Lund, Birgitte W.; Gustafsson, Magnus; Schiffer, Hans H.; Donello, John E.; Olsson, Roger; Gil, Daniel W.; Brann, Mark R.

Identification of the first synthetic steroidogenic factor 1 inverse agonists: Pharmacological modulation of steroidogenic enzymes

MOLECULAR PHARMACOLOGY

IF3

2008-03-01

PREAI

Del Tredici, Andria L.; Andersen, Carsten B.; Currier, Erika A.; Ohrmund, Steven R.; Fairbain, Luke C.; Lund, Birgitte W.; Nash, Norman; Olsson, Roger; Piu, Fabrice

Monitoring interactions between receptor tyrosine kinases and their downstream effector proteins in living cells using bioluminescence resonance energy transfer

MOLECULAR PHARMACOLOGY

IF3

2007-12-01

PREAI

Tan, Philip K.; Wang, Jean; Littler, Pey-Lih H.; Wong, Kenneth K.; Sweetnam, Timothy A.; Keefe, William; Nash, Norman R.; Reding, Esther C.; Piu, Fabrice; Brann, Mark R.; Schiffer, Hans H.

Pharmacology and signaling properties of epidermal growth factor receptor isoforms studied by bioluminescence resonance energy transfer

MOLECULAR PHARMACOLOGY

IF3

2007-02-01

PREAI

Schiffer, Hans H.; Reding, Esther C.; Fuhs, Stephen R.; Lu, Qing; Piu, Fabrice; Wong, Steven; Littler, Pey-Lih H.; Weiner, Dave M.; Keefe, William; Tan, Phil K.; Nash, Norman R.; Knapp, Anne E.; Olsson, Roger; Brann, Mark R.

Pharmacological and behavioral profile of N-(4-fluorophenylmethyl)-N-(1-methylpiperidin-4-yl)-N′-(4-(2-methylpropyloxy)phenylmethyl) carbamide (2R, 3R)-dihydroxybutanedioate (2:1) (ACP-103), a novel 5-hydroxytryptamine2A receptor inverse agonist

JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

IF3.8

2006-05-01

207

PREAI

Vanover, KE; Weiner, DM; Makhay, M; Veinbergs, I; Gardell, LR; Lameh, J; del Tredici, AL; Piu, F; Schiffer, HH; Ott, TR; Burstein, ES; Uldam, AK; Thygesen, MB; Schlienger, N; Andersson, CM; Son, TY; Harvey, SC; Powell, SB; Geyer, MA; Tolf, BR; Brann, MR; Davis, RE

Identification of novel subtype selective RAR agonists

BIOCHEMICAL PHARMACOLOGY

IF5.6

2005-12-01

PREAI

Piu, F; Gauthier, NK; Olsson, R; Currier, EA; Lund, BW; Croston, GE; Hacksell, U; Brann, MR

Discovery of a potent, orally available, and isoform-selective retinoic acid β2 receptor agonist

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2005-11-04

PREAI

Lund, BW; Piu, F; Gauthier, NK; Eeg, A; Currier, E; Sherbukhin, V; Brann, MR; Hacksell, T; Olsson, R