未登录Targeting KDM1A in Neuroblastoma with NCL-1 Induces a Less Aggressive Phenotype and Suppresses Angiogenesis
Spruessel, Annika; Suzuki, Takayoshi; Miyata, Naoki; Astrahantseff, Kathy; Szymansky, Annabell; Toedling, Joern; Thole-Kliesch, Theresa M.; Ballagee, Annika; Lodrini, Marco; Kuenkele, Annette; Truss, Matthias; Heukamp, Lukas C.; Mathia, Susanne; Hertwig, Falk; Rosenberger, Christian; Eggert, Angelika; Deubzer, Hedwig E.; Schulte, Johannes H.
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收藏Design, synthesis, and evaluation of Trolox-conjugated amyloid-β C-terminal peptides for therapeutic intervention in an in vitro model of Alzheimer's disease
Arai, Takuya; Ohno, Akiko; Kazunori, Mori; Kakizawa, Taeko; Kuwata, Hiroshi; Ozawa, Toshihiko; Shibanuma, Motoko; Hara, Shuntaro; Ishida, Seiichi; Kurihara, Masaaki; Miyata, Naoki; Nakagawa, Hidehiko; Fukuhara, Kiyoshi
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收藏Identification of SNAIL1 Peptide-Based Irreversible Lysine-Specific Demethylase 1-Selective Inactivators
Itoh, Yukihiro; Aihara, Keisuke; Mellini, Paolo; Tojo, Toshifumi; Ota, Yosuke; Tsumoto, Hiroki; Solomon, Viswas Raja; Zhan, Peng; Suzuki, Miki; Ogasawara, Daisuke; Shigenaga, Akira; Inokuma, Tsubasa; Nakagawa, Hidehiko; Miyata, Naoki; Mizukami, Tamio; Otaka, Akira; Suzuki, Takayoshi
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收藏Profiling and relative quantification of multiply nitrated and oxidized fatty acids多重硝化和氧化脂肪酸的分析和相对定量
Milic, Ivana; Griesser, Eva; Vemula, Venukumar; Ieda, Naoya; Nakagawa, Hidehiko; Miyata, Naoki; Galano, Jean-Marie; Oger, Camille; Durand, Thierry; Fedorova, Maria
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收藏Design, Synthesis, and Biological Activity of NCC149 Derivatives as Histone Deacetylase 8-Selective Inhibitors
Suzuki, Takayoshi; Muto, Nobusuke; Bando, Masashige; Itoh, Yukihiro; Masaki, Ayako; Ri, Masaki; Ota, Yosuke; Nakagawa, Hidehiko; Iida, Shinsuke; Shirahige, Katsuhiko; Miyata, Naoki
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收藏Identification of the KDM2/7 Histone Lysine Demethylase Subfamily Inhibitor and its Antiproliferative Activity
Suzuki, Takayoshi; Ozasa, Hiroki; Itoh, Yukihiro; Zhan, Peng; Sawada, Hideyuki; Mino, Koshiki; Walport, Louise; Ohkubo, Rei; Kawamura, Akane; Yonezawa, Masato; Tsukada, Yuichi; Tumber, Anthony; Nakagawa, Hidehiko; Hasegawa, Makoto; Sasaki, Ryuzo; Mizukami, Tamio; Schofield, Christopher J.; Miyata, Naoki
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收藏The KDM1A histone demethylase is a promising new target for the epigenetic therapy of medulloblastoma
Pajtler, Kristian W.; Weingarten, Christina; Thor, Theresa; Kunkele, Annette; Heukamp, Lukas C.; Buttner, Reinhard; Suzuki, Takayoshi; Miyata, Naoki; Grotzer, Michael; Rieb, Anja; Sprussel, Annika; Eggert, Angelika; Schramm, Alexander; Schulte, Johannes H.
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收藏FFA1-selective agonistic activity based on docking simulation using FFA1 and GPR120 homology models
Takeuchi, Masato; Hirasawa, Akira; Hara, Takafumi; Kimura, Ikuo; Hirano, Tatsuya; Suzuki, Takayoshi; Miyata, Naoki; Awaji, Takeo; Ishiguro, Masaji; Tsujimoto, Gozoh
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收藏Targeting the PELP1-KDM1 axis as a potential therapeutic strategy for breast cancer (vol 14, pg R108, 2012)
Cortez, Valerie; Mann, Monica; Tekmal, Seshidhar; Suzuki, Takayoshi; Miyata, Naoki; Rodriguez-Aguayo, Cristian; Lopez-Berestein, Gabriel; Sood, Anil K.; Vadlamudi, Ratna K.
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收藏Rapid Discovery of Highly Potent and Selective Inhibitors of Histone Deacetylase 8 Using Click Chemistry to Generate Candidate Libraries
Suzuki, Takayoshi; Ota, Yosuke; Ri, Masaki; Bando, Masashige; Gotoh, Aogu; Itoh, Yukihiro; Tsumoto, Hiroki; Tatum, Prima R.; Mizukami, Tamio; Nakagawa, Hidehiko; Iida, Shinsuke; Ueda, Ryuzo; Shirahige, Katsuhiko; Miyata, Naoki
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