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A

Andrea Martella

Leiden University
H指数:18
被引数:1,336

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荣誉奖项

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Translational Application of the Five-Star Matrix for the Structure-Guided Optimization of a Bicyclopiperazine DEL Hit into Bcpz 1.5: A Potent Monoacylglycerol Lipase Inhibitor with Functional Inhibition in Human Brain Homogenate and Efficacy in Neuroinflammatory Models

五星级矩阵在结构导向优化双环哌嗪DEL命中化合物至Bcpz 1.5中的应用：一种在人体脑匀浆中具有功能性抑制并在神经炎症模型中具有疗效的强效单酰基甘油脂肪酶抑制剂

Journal of Medicinal Chemistry
IF6.8
2026-01-010
PRE
Benjamin Brennecke; Louise Plais; Benoit Hornsperger; Martin Binder; Christian Bartelmus; Markus Bürkler; Fionn O’Hara; Carsten Kroll; Satoshi Tsuchiya; Buelent Koçer; Hans Georg Richter; Martin Ritter; Katrin Groebke Zbinden; Maude Giroud; Manfred P Schneider; Andrea Martella; Ann Petersen; Wiebke Saal; Melanie Guérard; Axel Pähler; Luca B. Gobbi; Antonia F. Stepan; Moreno Wichert; Andreas Topp; Dominik Heer; Iris Ruf; Remo Hochstrasser; Manuel Hilbert; Sylwia Huber; Anto Pavlovic; Juliane Stephanus; Sina Simon; A. Haider; Mario van der Stelt; Matthias Wittwer; Ludovic Collin; Jörg Benz; Bernd Kuhn; Uwe Grether
Structure-Guided Discovery of cis-Hexahydro-pyrido-oxazinones as Reversible, Drug-like Monoacylglycerol Lipase Inhibitors
JOURNAL OF MEDICINAL CHEMISTRY
IF6.8
2024-10-031
PRE
Kuhn, Bernd; Ritter, Martin; Hornsperger, Benoit; Bell, Charles; Kocer, Buelent; Rombach, Didier; Lutz, Marius D. R.; Gobbi, Luca; Kuratli, Martin; Bartelmus, Christian; Burkler, Markus; Koller, Raffael; Tosatti, Paolo; Ruf, Iris; Guerard, Melanie; Pavlovic, Anto; Stephanus, Juliane; O'Hara, Fionn; Wetzl, Dennis; Saal, Wiebke; Stihle, Martine; Roth, Doris; Hug, Melanie; Huber, Sylwia; Heer, Dominik; Kroll, Carsten; Topp, Andreas; Schneider, Manfred; Gertsch, Jurg; Glasmacher, Sandra; van der Stelt, Mario; Martella, Andrea; Wittwer, Matthias Beat; Collin, Ludovic; Benz, Jorg; Richter, Hans; Grether, Uwe
Discovery of a NAPE-PLD inhibitor that modulates emotional behavior in mice
NATURE CHEMICAL BIOLOGY
IF13.7
2020-05-1154
OAAI
Mock, Elliot D.; Mustafa, Mohammed; Gunduz-Cinar, Ozge; Cinar, Resat; Petrie, Gavin N.; Kantae, Vasudev; Di, Xinyu; Ogasawara, Daisuke; Varga, Zoltan V.; Paloczi, Janos; Miliano, Cristina; Donvito, Giulia; van Esbroeck, Annelot C. M.; van der Gracht, Anouk M. F.; Kotsogianni, Ioli; Park, Joshua K.; Martella, Andrea; van der Wel, Tom; Soethoudt, Marjolein; Jiang, Ming; Wendel, Tiemen J.; Janssen, Antonius P. A.; Bakker, Alexander T.; Donovan, Colleen M.; Castillo, Laura, I; Florea, Bogdan, I; Wat, Jesse; van den Hurk, Helma; Wittwer, Matthias; Grether, Uwe; Holmes, Andrew; van Boeckel, Constant A. A.; Hankemeier, Thomas; Cravatt, Benjamin F.; Buczynski, Matthew W.; Hill, Matthew N.; Pacher, Pal; Lichtman, Aron H.; van der Stelt, Mario
Fishing for Targets of Alien Metabolites: A Novel Peroxisome Proliferator-Activated Receptor (PPAR) Agonist from a Marine Pest
MARINE DRUGS
IF5.4
2018-11-0327
OAAI
Vitale, Rosa Maria; D'Aniello, Enrico; Gorbi, Stefania; Martella, Andrea; Silvestri, Cristoforo; Giuliani, Maria Elisa; Fellous, Tariq; Gentile, Alessandra; Carbone, Marianna; Cutignano, Adele; Grauso, Laura; Magliozzi, Laura; Polese, Gianluca; D'Aniello, Biagio; Defranoux, Fanny; Felline, Serena; Terlizzi, Antonio; Calignano, Antonio; Regoli, Francesco; Di Marzo, Vincenzo; Amodeo, Pietro; Mollo, Ernesto
Selective Photoaffinity Probe That Enables Assessment of Cannabinoid CB2 Receptor Expression and Ligand Engagement in Human Cells
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
IF15.6
2018-02-0868
OAAI
Soethoudt, Marjolein; Stolze, Sara C.; Westphal, Matthias V.; van Stralen, Luuk; Martella, Andrea; van Rooden, Eva J.; Guba, Wolfgang; Varga, Zoltan V.; Deng, Hui; van Kasteren, Sander I.; Grether, Uwe; IJzerman, Adriaan P.; Pacher, Pal; Carreira, Erick M.; Overkleeft, Herman S.; Ioan-Facsinay, Andreea; Heitman, Laura H.; van der Stelt, Mario
Cannabinoid CB2 receptor ligand profiling reveals biased signalling and off-target activity
NATURE COMMUNICATIONS
IF15.7
2017-01-03282
OAAI
Soethoudt, Marjolein; Grether, Uwe; Fingerle, Juergen; Grim, Travis W.; Fezza, Filomena; de Petrocellis, Luciano; Ullmer, Christoph; Rothenhausler, Benno; Perret, Camille; van Gils, Noortje; Finlay, David; MacDonald, Christa; Chicca, Andrea; Gens, Marianela Dalghi; Stuart, Jordyn; de Vries, Henk; Mastrangelo, Nicolina; Xia, Lizi; Alachouzos, Georgios; Baggelaar, Marc P.; Martella, Andrea; Mock, Elliot D.; Deng, Hui; Heitman, Laura H.; Connor, Mark; Di Marzo, Vincenzo; Gertsch, Jurg; Lichtman, Aron H.; Maccarrone, Mauro; Pacher, Pal; Glass, Michelle; van der Stelt, Mario

研究方向

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V
Vincenzo Di Marzo
H 指数:158论文数:1,172被引数:9.6万
M
Mario van der Stelt
H 指数:49论文数:224被引数:1.0万
C
Cristoforo Silvestri
H 指数:33论文数:97被引数:3,978
U
Uwe Grether
H 指数:29论文数:160被引数:2,882
E
Elliot D. Mock
H 指数:10论文数:21被引数:1,222
M
Marjolein Soethoudt
H 指数:14论文数:18被引数:1,510
M
Matthias Wittwer
H 指数:38论文数:152被引数:4,323
P
Pál Pacher
H 指数:125论文数:508被引数:5.6万
F
Fabiana Piscitelli
H 指数:55论文数:223被引数:9,528
V
Vasudev Kantae
H 指数:14论文数:25被引数:1,019