未登录 Exceptionally Potent Chiral Anandamide Analogs 高活性手性阿纳坎德类似物 Georgiadis, Markos-Orestis; Ferreras, Elena; Ji, Lipin; Ferreira, Luana Assis; Hainline, John; Tong, Fei; Dang, Vuong Q.; Faragher, Alexandra; Sadybekov, Anastasiia V.; Bohn, Laura M.; Katritch, Vsevolod; Hohmann, Andrea G.; Makriyannis, Alexandros; Nikas, Spyros P. 分享 收藏
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Virtual library docking for cannabinoid-1 receptor agonists with reduced side effects 虚拟库对接用于寻找具有降低副作用的大麻素-1受体激动剂 Tummino, Tia A.; Iliopoulos-Tsoutsouvas, Christos; Braz, Joao M.; O'Brien, Evan S.; Stein, Reed M.; Craik, Veronica; Tran, Ngan K.; Ganapathy, Suthakar; Liu, Fangyu; Ho, Thanh C.; Radchenko, Dmytro S.; Moroz, Yurii S.; Rosado, Sian Rodriguez; Bhardwaj, Karnika; Benitez, Jorge; Liu, Yongfeng; Kandasamy, Herthana; Normand, Claire; Semache, Meriem; Glenn, Isabella; Irwin, John J.; Kumar, Kaavya Krishna; Makriyannis, Alexandros; Shoichet, Brian K. 分享 收藏
Pharmacological Inhibition of N-Acylethanolamine Acid Amidase (NAAA) Mitigates Intestinal Fibrosis Through Modulation of Macrophage Activity Nani, Maria Francesca; Pagano, Ester; De Cicco, Paola; Lucariello, Giuseppe; Cattaneo, Fabio; Tropeano, Francesca Paola; Cicia, Donatella; Amico, Rebecca; Raucci, Federica; Ercolano, Giuseppe; Maione, Francesco; Rinaldi, Maria Michela; Esposito, Fabiana; Ammendola, Rosario; Luglio, Gaetano; Capasso, Raffaele; Makriyannis, Alexandros; Petrosino, Stefania; Borrelli, Francesca; Romano, Barbara; Izzo, Angelo A. 分享 收藏
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Chiral Me-2-arachidonoyl Glycerols: The First Potent Endocannabinoid Glyceride Templates with Stability to COX-2 Nikas, Spyros P.; Ji, Lipin; Liu, Yingpeng; Georgiadis, Markos-Orestis; Dopeshwarkar, Amey; Straiker, Alex; Kudalkar, Shalley; Sadybekov, Anastasiia V.; Dvorakova, Michaela; Katritch, Vsevolod; Mackie, Ken; Marnett, Lawrence; Makriyannis, Alexandros 分享 收藏
Virtual Screening of a Chemically Diverse Superscaffold Library Enables Ligand Discovery for a Key GPCR Target 化学上多样化的超级支架文库的虚拟筛选可以发现关键GPCR靶标的配体 Grotsch, Katharina; Sadybekov, Anastasiia V.; Hiller, Sydney; Zaidi, Saheem; Eremin, Dmitry; Le, Austen; Liu, Yongfeng; Smith, Evan Carlton; Illiopoulis-Tsoutsouvas, Christos; Thomas, Joice; Aggarwal, Shubhangi; Pickett, Julie E.; Reyes, Cesar; Picazo, Elias; Roth, Bryan L.; Makriyannis, Alexandros; Katritch, Vsevolod; Fokin, Valery V. 分享 收藏
AM6527, a neutral CB1 receptor antagonist, suppresses opioid taking and seeking, as well as cocaine seeking in rodents without aversive effects Soler-Cedeno, Omar; Alton, Hannah; Bi, Guo-Hua; Linz, Emily; Ji, Lipin; Makriyannis, Alexandros; Xi, Zheng-Xiong 分享 收藏
P2X7 receptor-dependent increase in endocannabinoid 2-arachidonoyl glycerol production by neuronal cells in culture: Dynamics and mechanism Singh, Simar; Sarroza, Dennis; English, Anthony; Whittington, Dale; Dong, Ao; Malamas, Michael; Makriyannis, Alexandros; van Der Stelt, Mario; Li, Yulong; Zweifel, Larry; Bruchas, Michael R.; Land, Benjamin B.; Stella, Nephi 分享 收藏
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Eid et al. Interference with TGFβ1-Mediated Inflammation and Fibrosis Underlies Reno-Protective Effects of the CB1 Receptor Neutral Antagonists AM6545 and AM4113 in a Rat Model of Metabolic Syndrome(vol26, 866, 2021) Eid, Basma G.; Neamatallah, Thikryat; Hanafy, Abeer; El-Bassossy, Hany M.; Binmahfouz, Lenah; Aldawsari, Hibah M.; Hasan, Atif; Abd El-Aziz, Gamal; Vemuri, Kiran; Makriyannis, Alexandros 分享 收藏
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Effects of cannabinoid agonists and antagonists in male rats discriminating the synthetic cannabinoid AM2201 AlKhelb, Dalal; Burke, Emily L.; Zvonok, Alexander; Iliopoulos-Tsoutsouvas, Christos; Georgiadis, Markos-Orestis; Jiang, Shan; Ho, Thanh C.; Nikas, Spyros P.; Makriyannis, Alexandros; Desai, Rajeev I. 分享 收藏
Complex 33-beam simulated galactic cosmic radiation exposure impacts cognitive function and prefrontal cortex neurotransmitter networks in male mice Desai, Rajeev I.; Kangas, Brian D.; Luc, Oanh T.; Solakidou, Eleana; Smith, Evan C.; Dawes, Monica H.; Ma, Xiaoyu; Makriyannis, Alexandros; Chatterjee, Subhamoy; Dayeh, Maher A.; Munoz-Jaramillo, Andres; Desai, Mihir I.; Limoli, Charles L. 分享 收藏
The neutral CB1 antagonist AM6527 reduces ethanol seeking, binge-like consumption, reinforcing, and withdrawal effects in male and female mice Raghav, Jimit Girish; Kumar, Hritik; Ji, Lipin; Vemuri, Kiran; Makriyannis, Alexandros; Suh, Junghyup; Leonard, Michael Z.; Dang, Vivi; Ty, Chelsea; Marandola, Stephen; Kane, Natalie; Witt, Annika S.; Shaqour, Samar; Miczek, Klaus A. 分享 收藏
Goods and Bads of the Endocannabinoid System as a Therapeutic Target: Lessons Learned after 30 Years Maccarrone, Mauro; Di Marzo, Vincenzo; Gertsch, Jurg; Grether, Uwe; Howlett, Allyn C.; Hua, Tian; Makriyannis, Alexandros; Piomelli, Daniele; Ueda, Natsuo; van der Stelt, Mario 分享 收藏
Structural basis for activation of CB1 by an endocannabinoid analog 内源性大麻素类似物激活CB1的结构基础 Kumar, Kaavya Krishna; Robertson, Michael J.; Thadhani, Elina; Wang, Haoqing; Suomivuori, Carl-Mikael; Powers, Alexander S.; Ji, Lipin; Nikas, Spyros P.; Dror, Ron O.; Inoue, Asuka; Makriyannis, Alexandros; Skiniotis, Georgios; Kobilka, Brian 分享 收藏