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Alexandros Makriyannis

northeastern university

85H指数
646论文数
2.8W被引数
收录论文 69
发表时间
Exceptionally Potent Chiral Anandamide Analogs高活性手性阿纳坎德类似物
err2025-09-01
err0
PREAI
errGeorgiadis, Markos-Orestis; Ferreras, Elena; Ji, Lipin; Ferreira, Luana Assis; Hainline, John; Tong, Fei; Dang, Vuong Q.; Faragher, Alexandra; Sadybekov, Anastasiia V.; Bohn, Laura M.; Katritch, Vsevolod; Hohmann, Andrea G.; Makriyannis, Alexandros; Nikas, Spyros P.
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Crystal structures of agonist-bound human cannabinoid receptor CB1CB1人 cannabinoid 受体的激动剂结合结构
errNature
IF48.5
err2025-08-27
err0
PREAI
errTian Hua; Kiran Vemuri; Spyros P. Nikas; Yiran Wu; Lu Qu; Mengchen Pu; Anisha Korde; Shan Jiang; Jo-Hao Ho; Gye Won Han; Kang Ding; Xuanxuan Li; Haiguang Liu; Michael A. Hanson; Suwen Zhao; Laura M. Bohn; Alexandros Makriyannis; Raymond C. Stevens; Zhi-Jie Liu
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Retraction Note: Crystal structures of agonist-bound human cannabinoid receptor CB1撤回通知:激动剂结合的人 cannabinoid 受体 CB1 的晶体结构
errNature
IF48.5
err2025-08-27
err0
PREAI
errTian Hua; Kiran Vemuri; Spyros P. Nikas; Robert B. Laprairie; Yiran Wu; Lu Qu; Mengchen Pu; Anisha Korde; Shan Jiang; Jo-Hao Ho; Gye Won Han; Kang Ding; Xuanxuan Li; Haiguang Liu; Michael A. Hanson; Suwen Zhao; Laura M. Bohn; Alexandros Makriyannis; Raymond C. Stevens; Zhi-Jie Liu
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Novel Tetraolefinic Chain Phenyl Substituted Endocannabinoid Probes新型四烯基链苯基取代的内源性大麻素探针
err2025-06-26
err0
PREAI
errMarkos-Orestis Georgiadis; Lipin Ji; Fei Tong; Vuong Q. Dang; Luana Assis Ferreira; Alexandra Faragher; Ngan Tran; Anastasiia V. Sadybekov; Suthakar Ganapathy; Nikolai Zvonok; Vsevolod Katritch; Andrea G. Hohmann; Laura M. Bohn; Alexandros Makriyannis; Spyros P. Nikas
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CB1 cannabinoid receptor agonists induce acute respiratory depression in awake miceCB1大麻素受体激动剂在清醒小鼠中引起急性呼吸抑制。
err2025-04-01
err1
errOAAI
errWatkins, Joshua; Aradi, Petra; Hahn, Rachel; Makriyannis, Alexandros; Mackie, Ken; Katona, Istvan; Hohmann, Andrea G.
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Virtual library docking for cannabinoid-1 receptor agonists with reduced side effects虚拟库对接用于寻找具有降低副作用的大麻素-1受体激动剂
err2025-03-06
err0
errOAAI
errTummino, Tia A.; Iliopoulos-Tsoutsouvas, Christos; Braz, Joao M.; O'Brien, Evan S.; Stein, Reed M.; Craik, Veronica; Tran, Ngan K.; Ganapathy, Suthakar; Liu, Fangyu; Ho, Thanh C.; Radchenko, Dmytro S.; Moroz, Yurii S.; Rosado, Sian Rodriguez; Bhardwaj, Karnika; Benitez, Jorge; Liu, Yongfeng; Kandasamy, Herthana; Normand, Claire; Semache, Meriem; Glenn, Isabella; Irwin, John J.; Kumar, Kaavya Krishna; Makriyannis, Alexandros; Shoichet, Brian K.
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Pharmacological Inhibition of N-Acylethanolamine Acid Amidase (NAAA) Mitigates Intestinal Fibrosis Through Modulation of Macrophage Activity
err2024-08-30
err0
PREAI
errNani, Maria Francesca; Pagano, Ester; De Cicco, Paola; Lucariello, Giuseppe; Cattaneo, Fabio; Tropeano, Francesca Paola; Cicia, Donatella; Amico, Rebecca; Raucci, Federica; Ercolano, Giuseppe; Maione, Francesco; Rinaldi, Maria Michela; Esposito, Fabiana; Ammendola, Rosario; Luglio, Gaetano; Capasso, Raffaele; Makriyannis, Alexandros; Petrosino, Stefania; Borrelli, Francesca; Romano, Barbara; Izzo, Angelo A.
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Cannabinoid CB2 receptors in primary sensory neurons are implicated in CB2 agonist-mediated suppression of paclitaxel-induced neuropathic nociception and sexually-dimorphic sparing of morphine tolerance
err2024-07-01
err0
errOAAI
errGuenther, Kelsey G.; Lin, Xiaoyan; Xu, Zhili; Makriyannis, Alexandros; Romero, Julian; Hillard, Cecilia J.; Mackie, Ken; Hohmann, Andrea G.
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Chiral Me-2-arachidonoyl Glycerols: The First Potent Endocannabinoid Glyceride Templates with Stability to COX-2
err2024-05-28
err2
PREAI
errNikas, Spyros P.; Ji, Lipin; Liu, Yingpeng; Georgiadis, Markos-Orestis; Dopeshwarkar, Amey; Straiker, Alex; Kudalkar, Shalley; Sadybekov, Anastasiia V.; Dvorakova, Michaela; Katritch, Vsevolod; Mackie, Ken; Marnett, Lawrence; Makriyannis, Alexandros
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Virtual Screening of a Chemically Diverse Superscaffold Library Enables Ligand Discovery for a Key GPCR Target化学上多样化的超级支架文库的虚拟筛选可以发现关键GPCR靶标的配体
err2024-04-10
err4
PREAI
errGrotsch, Katharina; Sadybekov, Anastasiia V.; Hiller, Sydney; Zaidi, Saheem; Eremin, Dmitry; Le, Austen; Liu, Yongfeng; Smith, Evan Carlton; Illiopoulis-Tsoutsouvas, Christos; Thomas, Joice; Aggarwal, Shubhangi; Pickett, Julie E.; Reyes, Cesar; Picazo, Elias; Roth, Bryan L.; Makriyannis, Alexandros; Katritch, Vsevolod; Fokin, Valery V.
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AM6527, a neutral CB1 receptor antagonist, suppresses opioid taking and seeking, as well as cocaine seeking in rodents without aversive effects
err2024-04-10
err1
errOAAI
errSoler-Cedeno, Omar; Alton, Hannah; Bi, Guo-Hua; Linz, Emily; Ji, Lipin; Makriyannis, Alexandros; Xi, Zheng-Xiong
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P2X7 receptor-dependent increase in endocannabinoid 2-arachidonoyl glycerol production by neuronal cells in culture: Dynamics and mechanism
err2024-04-06
err0
PREAI
errSingh, Simar; Sarroza, Dennis; English, Anthony; Whittington, Dale; Dong, Ao; Malamas, Michael; Makriyannis, Alexandros; van Der Stelt, Mario; Li, Yulong; Zweifel, Larry; Bruchas, Michael R.; Land, Benjamin B.; Stella, Nephi
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Eid et al. Interference with TGFβ1-Mediated Inflammation and Fibrosis Underlies Reno-Protective Effects of the CB1 Receptor Neutral Antagonists AM6545 and AM4113 in a Rat Model of Metabolic Syndrome(vol26, 866, 2021)
err2024-02-19
err0
errOAAI
errEid, Basma G.; Neamatallah, Thikryat; Hanafy, Abeer; El-Bassossy, Hany M.; Binmahfouz, Lenah; Aldawsari, Hibah M.; Hasan, Atif; Abd El-Aziz, Gamal; Vemuri, Kiran; Makriyannis, Alexandros
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A Simple Chiral 1H NMR Method for the Discrimination of (R)- and (S)-Cannabichromene in Complex Natural Mixtures and Their Effects on TRPA1 Activity
err2023-12-29
err4
PREAI
errDadiotis, Evangelos; Cui, Meng; Gerasi, Maria; Mitsis, Vangelis; Melliou, Eleni; Makriyannis, Alexandros; Logothetis, Diomedes E.; Magiatis, Prokopios
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Effects of cannabinoid agonists and antagonists in male rats discriminating the synthetic cannabinoid AM2201
err2023-12-01
err1
PREAI
errAlKhelb, Dalal; Burke, Emily L.; Zvonok, Alexander; Iliopoulos-Tsoutsouvas, Christos; Georgiadis, Markos-Orestis; Jiang, Shan; Ho, Thanh C.; Nikas, Spyros P.; Makriyannis, Alexandros; Desai, Rajeev I.
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Complex 33-beam simulated galactic cosmic radiation exposure impacts cognitive function and prefrontal cortex neurotransmitter networks in male mice
err2023-11-27
err5
errOAAI
errDesai, Rajeev I.; Kangas, Brian D.; Luc, Oanh T.; Solakidou, Eleana; Smith, Evan C.; Dawes, Monica H.; Ma, Xiaoyu; Makriyannis, Alexandros; Chatterjee, Subhamoy; Dayeh, Maher A.; Munoz-Jaramillo, Andres; Desai, Mihir I.; Limoli, Charles L.
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The neutral CB1 antagonist AM6527 reduces ethanol seeking, binge-like consumption, reinforcing, and withdrawal effects in male and female mice
err2023-11-25
err3
PREAI
errRaghav, Jimit Girish; Kumar, Hritik; Ji, Lipin; Vemuri, Kiran; Makriyannis, Alexandros; Suh, Junghyup; Leonard, Michael Z.; Dang, Vivi; Ty, Chelsea; Marandola, Stephen; Kane, Natalie; Witt, Annika S.; Shaqour, Samar; Miczek, Klaus A.
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Goods and Bads of the Endocannabinoid System as a Therapeutic Target: Lessons Learned after 30 Years
err2023-09-01
err44
errOAAI
errMaccarrone, Mauro; Di Marzo, Vincenzo; Gertsch, Jurg; Grether, Uwe; Howlett, Allyn C.; Hua, Tian; Makriyannis, Alexandros; Piomelli, Daniele; Ueda, Natsuo; van der Stelt, Mario
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Structural basis for activation of CB1 by an endocannabinoid analog内源性大麻素类似物激活CB1的结构基础
err2023-05-09
err21
errOAAI
errKumar, Kaavya Krishna; Robertson, Michael J.; Thadhani, Elina; Wang, Haoqing; Suomivuori, Carl-Mikael; Powers, Alexander S.; Ji, Lipin; Nikas, Spyros P.; Dror, Ron O.; Inoue, Asuka; Makriyannis, Alexandros; Skiniotis, Georgios; Kobilka, Brian
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