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收藏A structure-based framework for selective inhibitor design and optimization基于结构的框架用于选择性抑制剂的研发与优化
Zou, Yurong; Guo, Tao; Fu, Zhiyuan; Guo, Zhongning; Bo, Weichen; Yan, Dengjie; Wang, Qiantao; Zeng, Jun; Xu, Dingguo; Wang, Taijin; Chen, Lijuan
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收藏Local Scaffold Diversity-Contributed Generator for Discovering Potential NLRP3 Inhibitors
Bo, Weichen; Duan, Yangqin; Zou, Yurong; Ma, Ziyan; Yang, Tao; Wang, Peng; Guo, Tao; Fu, Zhiyuan; Wang, Jianmin; Fan, Linchuan; Liu, Jie; Wang, Taijin; Chen, Lijuan
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收藏Discovery of a highly selective JAK3 inhibitor for the treatment of rheumatoid arthritis
Pei, Heying; He, Linhong; Shao, Mingfeng; Yang, Zhuang; Ran, Yan; Li, Dan; Zhou, Yuanyuan; Tang, Minghai; Wang, Taijin; Gong, Yanqiu; Chen, Xiaoxin; Yang, Shengyong; Xiang, Mingli; Chen, Lijuan
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收藏Design, synthesis, and SAR study of highly potent, selective, irreversible covalent JAK3 inhibitors高效,选择性,不可逆共价JAK3抑制剂的设计,合成和SAR研究
He, Linhong; Shao, Mingfeng; Wang, Taijin; Lan, Tingxuan; Zhang, Chufeng; Chen, Lijuan
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收藏Design, synthesis and biological evaluation of 4-anilinoquinoline derivatives as novel potent tubulin depolymerization agents
Zhou, Yuanyuan; Yan, Wei; Cao, Dong; Shao, Mingfeng; Li, Dan; Wang, Fang; Yang, Zhuang; Chen, Yong; He, Linhong; Wang, Taijin; Shen, Mingsheng; Chen, Lijuan
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收藏Design, Synthesis, and Evaluation of in Vitro and in Vivo Anticancer Activity of 4-Substituted Coumarins: A Novel Class of Potent Tubulin Polymerization Inhibitors
Cao, Dong; Liu, Yibin; Yan, Wei; Wang, Chunyu; Bai, Peng; Wang, Taijin; Tang, Minghai; Wang, Xiaoyan; Yang, Zhuang; Ma, Buyun; Ma, Liang; Lei, Lei; Wang, Fang; Xu, Bixue; Zhou, Yuanyuan; Yang, Tao; Chen, Lijuan
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收藏Development of Purine-Based Hydroxamic Acid Derivatives: Potent Histone Deacetylase Inhibitors with Marked in Vitro and in Vivo Antitumor Activities嘌呤基异羟肟酸衍生物的开发: 有效的组蛋白去乙酰化酶抑制剂,具有明显的体外和体内抗肿瘤活性
Chen, Yong; Wang, Xiaoyan; Xiang, Wei; He, Lin; Tang, Minghai; Wang, Fang; Wang, Taijin; Yang, Zhuang; Yi, Yuyao; Wang, Hairong; Niu, Ting; Zheng, Li; Lei, Lei; Li, Xiaobin; Song, Hang; Chen, Lijuan
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收藏Discovery of Selective Histone Deacetylase 6 Inhibitors Using the Quinazoline as the Cap for the Treatment of Cancer
Yang, Zhuang; Wang, Taijin; Wang, Fang; Niu, Ting; Liu, Zhuowei; Chen, Xiaoxin; Long, Chaofeng; Tang, Minghai; Cao, Dong; Wang, Xiaoyan; Xiang, Wei; Yi, Yuyao; Ma, Liang; You, Jingsong; Chen, Lijuan
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