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B

Biao Hong

tianjin medical university
H指数:13
被引数:507

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PEAKS activation by PROTAC EPIC-0726 potentiates temozolomide in glioblastoma via K63/K48 ubiquitination-dependent ERK/AKT suppression and p21 stabilization

PEAKS激活通过PROTAC EPIC-0726在胶质母细胞瘤中增强替莫唑胺的效果,其机制涉及K63/K48泛素化依赖的ERK/AKT抑制及p21稳定化。

2025-10-270
PRE
Linagliptin synergizes with cPLA2 inhibition to enhance temozolomide efficacy by interrupting DPP4-mediated EGFR stabilization in glioma

Linagliptin通过中断DPP4介导的EGFR稳定化,与cPLA2抑制协同作用以增强替莫唑胺在胶质瘤中的疗效。

2025-05-210
OAAI