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Yongtai Yang

fudan university
H指数:18
被引数:1,009

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Discovery of N-(2-chloro-5-(3-(pyridin-4-yl)-1H-pyrazolo[3,4-b] pyridin-5-yl)pyridin-3-yl)-4-fluorobenzenesulfonamide (FD274) as a highly potent PI3K/mTOR dual inhibitor for the treatment of acute myeloid leukemia

发现N-(2-氯-5-(3-(pyridin-4-yl)-1h-吡唑并 [3,4-b] pyridin-5-yl)pyridin-3-yl)-4-氟苯磺酰胺 (FD274) 作为高效PI3K/mTOR双重抑制剂用于治疗急性髓细胞性白血病

2023-10-014
PRE
Bioisosteric replacements of the indole moiety for the development of a potent and selective PI3Kδ inhibitor: Design, synthesis and biological evaluation

用于开发有效和选择性PI3Kδ 抑制剂的吲哚部分的生物等排取代: 设计,合成和生物学评估

2021-11-0112
PREAI