未登录 AI-Driven De Novo Design and Development of Nontoxic DYRK1A Inhibitors (vol 68, pg 10346, 2025) AI驱动的无毒DYRK1A抑制剂的从头设计和开发 (第68卷,10346页,2025) Garcia, Eduardo Gonzalez; Varas Pardo, Pablo; Gonzalez-Naranjo, Pedro; Ulzurrun, Eugenia; Marcos-Ayuso, Guillermo; Perez, Concepcion; Paez, Juan A.; Insua, David Rios; Santana, Simon Rodriguez; Campillo, Nuria E. 分享 收藏
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AI-Driven De Novo Design and Development of Nontoxic DYRK1A Inhibitors AI驱动的新型无毒DYRK1A抑制剂的设计与开发 Garcia, EduardoGonzalez; Varas, Pablo; Gonzalez-Naranjo, Pedro; Ulzurrun, Eugenia; Marcos-Ayuso, Guillermo; Perez, Concepcion; Paez, Juan A.; Insua, David Rios; Santana, Simon Rodriguez; Campillo, Nuria E. 分享 收藏
Allosteric modulation of the CXCR4:CXCL12 axis by targeting receptor nanoclustering via the TMV-TMVI domain 通过tmv-tmvi结构域靶向受体纳米簇对CXCR4:CXCL12轴的变构调节 Garcia-Cuesta, Eva M.; Martinez, Pablo; Selvaraju, Karthik; Ulltjarn, Gabriel; Pozo, Adrian Miguel Gomez; D'Agostino, Gianluca; Gardeta, Sofia; Quijada-Freire, Adriana; Gabella, Patricia Blanco; Roca, Carlos; Hoyo, Daniel del; Jimenez-Saiz, Rodrigo; Garcia-Rubia, Alfonso; Palacios, Blanca Soler; Lucas, Pilar; Ayala-Bueno, Rosa; Acerete, Noelia Santander; Carrasco, Yolanda; Sorzano, Carlos Oscar; Martinez, Ana; Campillo, Nuria E.; Jensen, Lasse D.; Frade, Jose Miguel Rodriguez; Santiago, Cesar; Mellado, Mario 分享 收藏
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N?-Phenylacetohydrazide Derivatives as Potent Ebola Virus Entry Inhibitors with an Improved Pharmacokinetic Profile N?-苯基乙酰肼衍生物作为有效的埃博拉病毒进入抑制剂,具有改善的药代动力学特征 Garcia-Rubia, Alfonso; Lasala, Fatima; Ginex, Tiziana; Morales-Tenorio, Marcos; Olal, Catherine; Heung, Michelle; Oquist, Paola; Galindo, Inmaculada; Cuesta-Geijo, Miguel Aprimengel; Casasnovas, Jose M.; Campillo, Nuria E.; Canales, Angeles; Alonso, Covadonga; Martinez, Ana; Munoz-Fontela, Cesar; Delgado, Rafael; Gil, Carmen 分享 收藏
Suboptimal Concentrations of Ceftazidime/Avibactam (CAZ-AVI) May Select for CAZ-AVI Resistance in Extensively Drug-Resistant Pseudomonas aeruginosa: In Vivo and In Vitro Evidence Lopez-Montesinos, Inmaculada; Milagro Montero, Maria; Domene-Ochoa, Sandra; Lopez-Causape, Carla; Echeverria, Daniel; Sorli, Luisa; Campillo, Nuria; Luque, Sonia; Padilla, Eduardo; Prim, Nuria; Grau, Santiago; Oliver, Antonio; Horcajada, Juan P. 分享 收藏
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Multitarget drugs as potential therapeutic agents for alzheimer's disease. A new family of 5-substituted indazole derivatives as cholinergic and BACE1 inhibitors 多靶点药物作为阿尔茨海默病的潜在治疗药物。作为胆碱能和BACE1抑制剂的5-取代吲唑衍生物的新家族 Gonzalez-Naranjo, Pedro; Perez, Concepcion; Gonzalez-Sanchez, Marina; Gironda-Martinez, Adrian; Ulzurrun, Eugenia; Bartolome, Fernando; Rubio-Fernandez, Marcos; Martin-Requero, Angeles; Campillo, Nuria E.; Paez, Juan A. 分享 收藏
Comparison of Ceftolozane/Tazobactam Infusion Regimens in a Hollow-Fiber Infection Model against Extensively Drug-Resistant Pseudomonas aeruginosa Isolates Milagro Montero, Maria; Domene-Ochoa, Sandra; Lopez-Causape, Carla; Lopez-Montesinos, Inmaculada; Luque, Sonia; Sorli, Luisa; Campillo, Nuria; Padilla, Eduardo; Prim, Nuria; Ferrer Alapont, Lorena; Grau, Santiago; Oliver, Antonio; Horcajada, Juan P. 分享 收藏
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Time-Kill Evaluation of Antibiotic Combinations Containing Ceftazidime-Avibactam against Extensively Drug-Resistant Pseudomonas aeruginosa and Their Potential Role against Ceftazidime-Avibactam-Resistant Isolates 含头孢他啶-阿维巴坦的抗生素组合对广泛耐药铜绿假单胞菌的杀灭时间评估及其对头孢他啶-阿维巴坦耐药菌株的潜在作用 Montero, Maria M.; Ochoa, Sandra Domene; Lopez-Causape, Carla; Luque, Sonia; Sorli, Luisa; Campillo, Nuria; Lopez Montesinos, Inmaculada; Padilla, Eduardo; Prim, Nuria; Angulo-Brunet, Ariadna; Grau, Santiago; Oliver, Antonio; Horcajada, Juan P. 分享 收藏
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