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收藏A Phase 1 Assessment of the Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of (2R,6R)-Hydroxynorketamine in Healthy Volunteers
Raja, Shruti M.; Guptill, Jeffrey T.; Mack, Michelle; Peterson, Marni; Byard, Stephen; Twieg, Robert; Jordan, Lynn; Rich, Natalie; Castledine, Richard; Bourne, Samuel; Wilmshurst, Martin; Oxendine, Sarah; Avula, Satya G. C.; Zuleta, Helen; Quigley, Paul; Lawson, Sheila; McQuaker, Stephen J.; Ahmadkhaniha, Reza; Appelbaum, Lawrence G.; Kowalski, Kevin; Barksdale, Chineta T.; Gufford, Brandon T.; Awan, Asaad; Sancho, Alfredo R.; Moore, Max C.; Berrada, Karim; Cogan, Gregory B.; DeLarosa, Jesse; Radcliffe, Jeanne; Pao, Maryland; Kennedy, Michelle; Lawrence, Quentin; Goldfeder, Lisa; Amanfo, Leslie; Zanos, Panos; Gilbert, Jessica R.; Morris, Patrick J.; Moaddel, Ruin; Gould, Todd D.; Zarate, Carlos A.; Thomas, Craig J.
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收藏Identification and Characterization of ACP-5862, the Major Circulating Active Metabolite of Acalabrutinib: Both Are Potent and Selective Covalent Bruton Tyrosine Kinase Inhibitors
Podoll, Terry; Pearson, Paul G.; Kaptein, Allard; Evarts, Jerry; de Bruin, Gerjan; Emmelot-van Hoek, Maaike; de Jong, Anouk; van Lith, Bart; Sun, Hao; Byard, Stephen; Fretland, Adrian; Hoogenboom, Niels; Barf, Tjeerd; Slatter, J. Greg
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收藏Structure elucidation, metabolism, and drug interaction potential of ACP-5862, an active, major, circulating metabolite of acalabrutinib
Podoll, Terry; Pearson, Paul G.; Everts, Jerry; Ingallinera, Tim; Sun, Hao; Byard, Stephen; Fretland, Adrian J.; Slatter, J. Greg
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收藏Process Development toward a Pro-Drug of Buprenorphine
Berrell, Sophie L.; Byard, Stephen J.; Carey, John S.; Codina, Antonio; Davis, J. Alf; Filer, Katherine; Garnett, Alasdair; Marshall, Robin; Martin, Stephen J.; Mykytiuk, John; Northen, Julian; Pandya, Urvish; Reid, Gary; Smyth, Catherine; Watson, Lesa
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