未登录Structure-Based Design of Covalent SARS-CoV-2 Main Protease Inhibitors Targeting the Nirmatrelvir-Resistant E166 Mutants
Cai, Zhengjun; Kohaal, Navita; Georgiou, Kyriakos; Liang, Xueying; Chi, Xiang; Tan, Haozhou; Tan, Bin; Li, Kan; Fan, Guangjin; Lambrinidis, George; Kolocouris, Antonios; Deng, Xufang; Chen, Yu; Wang, Jun
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收藏Hit-to-Lead Optimization of Heterocyclic Carbonyloxycarboximidamides as Selective Antagonists at Human Adenosine A3 Receptor
Huang, Xianglin; Chorianopoulou, Anna; Kalkounou, Panagoula; Georgiou, Maria; Pousias, Athanasios; Davies, Amy; Pearce, Abigail; Harris, Matthew; Lambrinidis, George; Marakos, Panagiotis; Pouli, Nicole; Kolocouris, Antonios; Lougiakis, Nikolaos; Ladds, Graham
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收藏Hydrolytic Activity of Mitochondrial F1FO-ATP Synthase as a Target for Myocardial Ischemia-Reperfusion Injury: Discovery and In Vitro and In Vivo Evaluation of Novel Inhibitors
Nikolaou, Panagiota-Efstathia; Lambrinidis, George; Georgiou, Maria; Karagiannis, Dimitrios; Efentakis, Panagiotis; Bessis-Lazarou, Pavlos; Founta, Konstantina; Kampoukos, Stavros; Konstantin, Vasilis; Palmeira, Carlos M.; Davidson, Sean M.; Lougiakis, Nikolaos; Marakos, Panagiotis; Pouli, Nicole; Mikros, Emmanuel; Andreadou, Ioanna
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收藏Structure-Based Lead Optimization of Enterovirus D68 2A Protease Inhibitors
Tan, Bin; Liu, Chang; Li, Kan; Jadhav, Prakash; Lambrinidis, George; Zhu, Lan; Olson, Linda; Tan, Haozhou; Wen, Yu; Kolocouris, Antonios; Liu, Wei; Wang, Jun
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收藏Development of Stilbenoid and Chalconoid Analogues as Potent Tyrosinase Modulators and Antioxidant Agents
Vontzalidou, Argyro; Dimitrakoudi, Sapfo-Maria; Tsoukalas, Konstantinos; Zoidis, Grigoris; Chaita, Eliza; Dina, Evanthia; Cheimonidi, Christina; Trougakos, Ioannis P.; Lambrinidis, George; Skaltsounis, Alexios-Leandros; Mikros, Emmanuel; Aligiannis, Nektarios
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收藏Ochraceopyronide, a Rare α-Pyrone-C-lyxofuranoside from a Soil-Derived Fungus Aspergillus ochraceopetaliformis
Asmaey, Mostafa A.; Abatis, Dennis; Abdel-Razek, Ahmed S.; Lambrinidis, George; Chinou, Ioanna; Fokialakis, Nikolas; Tsafantakis, Nikolaos; Shaaban, Mohamed; Aligiannis, Nektarios
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收藏Discovery of SARS-CoV-2 Papain-like Protease Inhibitors through a Combination of High-Throughput Screening and a FlipGFP-Based Reporter Assay
Ma, Chunlong; Sacco, Michael Dominic; Xia, Zilei; Lambrinidis, George; Townsend, Julia Alma; Hu, Yanmei; Meng, Xiangzhi; Szeto, Tommy; Ba, Mandy; Zhang, Xiujun; Gongora, Maura; Zhang, Fushun; Marty, Michael Thomas; Xiang, Yan; Kolocouris, Antonios; Chen, Yu; Wang, Jun
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收藏Specific Residues in a Purine Transporter Are Critical for Dimerization, ER Exit, and Function
Kourkoulou, Anezia; Grevias, Pothos; Lambrinidis, George; Pyle, Euan; Dionysopoulou, Mariangela; Politis, Argyris; Mikros, Emmanuel; Byrne, Bernadette; Diallinas, George
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收藏The olive constituent oleuropein, as a PPARα agonist, markedly reduces serum triglycerides
Malliou, Foteini; Andreadou, Joanna; Gonzalez, Frank J.; Lazou, Antigone; Xepapadaki, Eva; Vallianou, Joanna; Lambrinidis, George; Mikros, Emmanuel; Marselos, Marios; Skaltsounis, Alexios-Leandros; Konstandi, Maria
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收藏Structure-activity relationships in fungal nucleobases transporters as dissected by the inhibitory effects of novel purine analogues
Gavriil, Efthymios-Spyridon; Dimitrakis, Spyridon; Papadaki, Georgia; Balaska, Sophia; Lambrinidis, George; Lougiakis, Nikolaos; Marakos, Panagiotis; Diallinas, George; Pouli, Nicole; Mikros, Emmanuel
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