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George Lambrinidis

national and kapodistrian university of athens

21H指数
102论文数
1.5K被引数
收录论文 27
发表时间
Structure-Based Design of Covalent SARS-CoV-2 Main Protease Inhibitors Targeting the Nirmatrelvir-Resistant E166 Mutants
errJACS AU
IF8.7
err2026-01-01
err0
PREAI
errCai, Zhengjun; Kohaal, Navita; Georgiou, Kyriakos; Liang, Xueying; Chi, Xiang; Tan, Haozhou; Tan, Bin; Li, Kan; Fan, Guangjin; Lambrinidis, George; Kolocouris, Antonios; Deng, Xufang; Chen, Yu; Wang, Jun
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Structural and Computational Insights into the Angiotensin II Type 1 Receptor: Advances in Antagonist Design and Implications for Hypertension Therapy (2020–2024)
err2025-12-22
err0
errOAAI
errFilippos Panteleimon Chatzipieris; Errikos Petsas; George Lambrinidis; John M. Matsoukas; Thomas Mavromoustakos
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Identification of naturally occurring drug-resistant mutations of SARS-CoV-2 papain-like protease鉴定SARS-CoV-2木瓜蛋白酶样蛋白酶自然发生的耐药突变
err2025-05-16
err0
errOAAI
errTan, Haozhou; Zhang, Qianru; Georgiou, Kyriakos; Zhang, Siyu; Li, Kan; Lambrinidis, George; Kolocouris, Antonios; Deng, Xufang
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Hit-to-Lead Optimization of Heterocyclic Carbonyloxycarboximidamides as Selective Antagonists at Human Adenosine A3 Receptor
err2024-07-29
err0
errOAAI
errHuang, Xianglin; Chorianopoulou, Anna; Kalkounou, Panagoula; Georgiou, Maria; Pousias, Athanasios; Davies, Amy; Pearce, Abigail; Harris, Matthew; Lambrinidis, George; Marakos, Panagiotis; Pouli, Nicole; Kolocouris, Antonios; Lougiakis, Nikolaos; Ladds, Graham
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Hydrolytic Activity of Mitochondrial F1FO-ATP Synthase as a Target for Myocardial Ischemia-Reperfusion Injury: Discovery and In Vitro and In Vivo Evaluation of Novel Inhibitors
err2023-11-09
err2
PREAI
errNikolaou, Panagiota-Efstathia; Lambrinidis, George; Georgiou, Maria; Karagiannis, Dimitrios; Efentakis, Panagiotis; Bessis-Lazarou, Pavlos; Founta, Konstantina; Kampoukos, Stavros; Konstantin, Vasilis; Palmeira, Carlos M.; Davidson, Sean M.; Lougiakis, Nikolaos; Marakos, Panagiotis; Pouli, Nicole; Mikros, Emmanuel; Andreadou, Ioanna
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Structure-Based Lead Optimization of Enterovirus D68 2A Protease Inhibitors
err2023-10-19
err3
PREAI
errTan, Bin; Liu, Chang; Li, Kan; Jadhav, Prakash; Lambrinidis, George; Zhu, Lan; Olson, Linda; Tan, Haozhou; Wen, Yu; Kolocouris, Antonios; Liu, Wei; Wang, Jun
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Synthesis and Biological Evaluation of Resveratrol Methoxy Derivatives
err2023-07-20
err11
errOAAI
errFragopoulou, Elizabeth; Gkotsi, Katerina; Petsini, Filio; Gioti, Katerina; Kalampaliki, Amalia D. D.; Lambrinidis, George; Kostakis, Ioannis K. K.; Tenta, Roxane
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Development of Stilbenoid and Chalconoid Analogues as Potent Tyrosinase Modulators and Antioxidant Agents
err2022-08-17
err2
errOAAI
errVontzalidou, Argyro; Dimitrakoudi, Sapfo-Maria; Tsoukalas, Konstantinos; Zoidis, Grigoris; Chaita, Eliza; Dina, Evanthia; Cheimonidi, Christina; Trougakos, Ioannis P.; Lambrinidis, George; Skaltsounis, Alexios-Leandros; Mikros, Emmanuel; Aligiannis, Nektarios
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Design of Multifaceted Antioxidants: Shifting towards Anti-Inflammatory and Antihyperlipidemic Activity
err2021-08-14
err5
errOAAI
errTzara, Ariadni; Lambrinidis, George; Kourounakis, Angeliki
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Ochraceopyronide, a Rare α-Pyrone-C-lyxofuranoside from a Soil-Derived Fungus Aspergillus ochraceopetaliformis
err2021-06-29
err9
errOAAI
errAsmaey, Mostafa A.; Abatis, Dennis; Abdel-Razek, Ahmed S.; Lambrinidis, George; Chinou, Ioanna; Fokialakis, Nikolas; Tsafantakis, Nikolaos; Shaaban, Mohamed; Aligiannis, Nektarios
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Discovery of SARS-CoV-2 Papain-like Protease Inhibitors through a Combination of High-Throughput Screening and a FlipGFP-Based Reporter Assay
err2021-06-18
err132
errOAAI
errMa, Chunlong; Sacco, Michael Dominic; Xia, Zilei; Lambrinidis, George; Townsend, Julia Alma; Hu, Yanmei; Meng, Xiangzhi; Szeto, Tommy; Ba, Mandy; Zhang, Xiujun; Gongora, Maura; Zhang, Fushun; Marty, Michael Thomas; Xiang, Yan; Kolocouris, Antonios; Chen, Yu; Wang, Jun
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Biological Evaluation and In Silico Study of Benzoic Acid Derivatives from Bjerkandera adusta Targeting Proteostasis Network Modules
err2020-02-04
err14
errOAAI
errGeorgousaki, Katerina; Tsafantakis, Nikolaos; Gumeni, Sentiljana; Lambrinidis, George; Gonzalez-Menendez, Victor; Tormo, Jose R.; Genilloud, Olga; Trougakos, Ioannis P.; Fokialakis, Nikolas
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Specific Residues in a Purine Transporter Are Critical for Dimerization, ER Exit, and Function
err2019-12-01
err10
errOAAI
errKourkoulou, Anezia; Grevias, Pothos; Lambrinidis, George; Pyle, Euan; Dionysopoulou, Mariangela; Politis, Argyris; Mikros, Emmanuel; Byrne, Bernadette; Diallinas, George
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The olive constituent oleuropein, as a PPARα agonist, markedly reduces serum triglycerides
err2018-09-01
err32
errOAAI
errMalliou, Foteini; Andreadou, Joanna; Gonzalez, Frank J.; Lazou, Antigone; Xepapadaki, Eva; Vallianou, Joanna; Lambrinidis, George; Mikros, Emmanuel; Marselos, Marios; Skaltsounis, Alexios-Leandros; Konstandi, Maria
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Structure-activity relationships in fungal nucleobases transporters as dissected by the inhibitory effects of novel purine analogues
err2018-08-01
err3
PREAI
errGavriil, Efthymios-Spyridon; Dimitrakis, Spyridon; Papadaki, Georgia; Balaska, Sophia; Lambrinidis, George; Lougiakis, Nikolaos; Marakos, Panagiotis; Diallinas, George; Pouli, Nicole; Mikros, Emmanuel
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Challenges with multi-objective QSAR in drug discovery
err2018-07-12
err24
PREAI
errLambrinidis, George; Tsantili-Kakoulidou, Anna
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Discovery of Novel Adenosine Receptor Antagonists through a Combined Structure- and Ligand-Based Approach Followed by Molecular Dynamics Investigation of Ligand Binding Mode
err2018-02-27
err20
errOAAI
errLagarias, Panagiotis; Vrontaki, Eleni; Lambrinidis, George; Stamatis, Dimitrios; Convertino, Marino; Ortore, Gabriella; Mavromoustakos, Thomas; Klotz, Karl-Norbert; Kolocouris, Antonios
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Novel Carbonyl Analogs of Tamoxifen: Design, Synthesis, and Biological Evaluation
err2017-09-26
err11
errOAAI
errKasiotis, Konstantinos M.; Lambrinidis, George; Fokialakis, Nikolas; Tzanetou, Evangelia N.; Mikros, Emmanuel; Haroutounian, Serkos A.
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