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A dual mechanism of action of AT-527 against SARS-CoV-2 polymerase Shannon, Ashleigh; Fattorini, Veronique; Sama, Bhawna; Selisko, Barbara; Feracci, Mikael; Falcou, Camille; Gauffre, Pierre; El Kazzi, Priscila; Delpal, Adrien; Decroly, Etienne; Alvarez, Karine; Eydoux, Cecilia; Guillemot, Jean-Claude; Moussa, Adel; Good, Steven S.; La Colla, Paolo; Lin, Kai; Sommadossi, Jean-Pierre; Zhu, Yingxiao; Yan, Xiaodong; Shi, Hui; Ferron, Francois; Canard, Bruno 分享 收藏
Evaluation of AT-752, a Double Prodrug of a Guanosine Nucleotide Analog with In Vitro and In Vivo Activity against Dengue and Other Flaviviruses Good, Steven S.; Shannon, Ashleigh; Lin, Kai; Moussa, Adel; Julander, Justin G.; La Colla, Paolo; Collu, Gabriella; Canard, Bruno; Sommadossi, Jean-Pierre 分享 收藏
AT-527, a Double Prodrug of a Guanosine Nucleotide Analog, Is a Potent Inhibitor of SARS-CoV-2 In Vitro and a Promising Oral Antiviral for Treatment of COVID-19 Good, Steven S.; Westover, Jonna; Jung, Kie Hoon; Zhou, Xiao-Jian; Moussa, Adel; La Colla, Paolo; Collu, Gabriella; Canard, Bruno; Sommadossi, Jean-Pierre 分享 收藏
Synthesis, cytotoxicity and antiviral evaluation of new series of imidazo[4,5-g]quinoline and pyrido[2,3-g]quinoxalinone derivatives Briguglio, Irene; Loddo, Roberta; Laurini, Erik; Fermeglia, Maurizio; Piras, Sandra; Corona, Paola; Giunchedi, Paolo; Gavini, Elisabetta; Sanna, Giuseppina; Giliberti, Gabriele; Ibba, Cristina; Farci, Pamela; La Colla, Paolo; Pricl, Sabrina; Carta, Antonio 分享 收藏
Antiviral activity of benzotriazole derivatives. 5-[4-(Benzotriazol-2-yl)phenoxy]-2,2-dimethylpentanoic acids potently and selectively inhibit Coxsackie Virus B5 Loddo, Roberta; Novelli, Federica; Sparatore, Anna; Tasso, Bruno; Tonelli, Michele; Boido, Vito; Sparatore, Fabio; Collu, Gabriella; Delogu, Ilenia; Giliberti, Gabriele; La Colla, Paolo 分享 收藏
Isolation and anticancer, anthelminthic, and antiviral (HIV) activity of acylphloroglucinols, and regioselective synthesis of empetrifranzinans from Hypericum roeperianum 酰基间苯二酚的隔离和抗癌,驱虫和抗病毒 (HIV) 活性,以及金丝桃属植物中empetrifranzinans的区域选择性合成 Fobofou, Serge Alain Tanemossu; Franke, Katrin; Sanna, Giuseppina; Porzel, Andrea; Bullita, Enrica; La Colla, Paolo; Wessjohann, Ludger A. 分享 收藏
Antiviral activity of benzimidazole derivatives. III. Novel anti-CVB-5, anti-RSV and anti-Sb-1 agents Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Vazzana, Iana; Sparatore, Anna; Boido, Vito; Sparatore, Fabio; La Colla, Paolo; Sanna, Giuseppina; Giliberti, Gabriele; Busonera, Bernardetta; Farci, Pamela; Ibba, Cristina; Loddo, Roberta 分享 收藏
Synthesis and antiviral activity of new phenylimidazopyridines and N-benzylidenequinolinamines derived by molecular simplification of phenylimidazo[4,5-g]quinolines Loddo, Roberta; Briguglio, Irene; Corona, Paola; Piras, Sandra; Loriga, Mario; Paglietti, Giuseppe; Carta, Antonio; Sanna, Giuseppina; Giliberti, Gabriele; Ibba, Cristina; Farci, Pamela; La Colla, Paolo 分享 收藏
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Disubstituted thiourea derivatives and their activity on CNS: Synthesis and biological evaluation Stefanska, Joanna; Szulczyk, Daniel; Koziol, Anna E.; Miroslaw, Barbara; Kedzierska, Ewa; Fidecka, Sylwia; Busonera, Bernardetta; Sanna, Giuseppina; Giliberti, Gabriele; La Colla, Paolo; Struga, Marta 分享 收藏
5-Acetyl-2-arylbenzimidazoles as antiviral agents. Part 4 Vitale, Gabriella; Corona, Paola; Loriga, Mario; Carta, Antonio; Paglietti, Giuseppe; Giliberti, Gabriele; Sanna, Giuseppina; Farci, Pamela; Marongiu, Maria Elena; La Colla, Paolo 分享 收藏
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Quinoline tricyclic derivatives. Design, synthesis and evaluation of the antiviral activity of three new classes of RNA-dependent RNA polymerase inhibitors Carta, Antonio; Briguglio, Irene; Piras, Sandra; Corona, Paola; Boatto, Giampiero; Nieddu, Maria; Giunchedi, Paolo; Marongiu, Maria Elena; Giliberti, Gabriele; Iuliano, Filippo; Blois, Sylvain; Ibba, Cristina; Busonera, Bernardetta; La Colla, Paolo 分享 收藏
3-Aryl-2-[1H-benzotriazol-1-yl]acrylonitriles: A novel class of potent tubulin inhibitors Carta, Antonio; Briguglio, Irene; Piras, Sandra; Boatto, Giampiero; La Colla, Paolo; Loddo, Roberta; Tolomeo, Manlio; Grimaudo, Stefania; Di Cristina, Antonietta; Pipitone, Rosaria Maria; Laurini, Erik; Paneni, Maria Silvia; Posocco, Paola; Fermeglia, Maurizio; Pricl, Sabrina 分享 收藏
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2,3-Dihydro-1,2-Diphenyl-substituted 4H-Pyridinone Derivatives as New Anti Flaviviridae Inhibitors Peduto, Antonella; Massa, Antonio; Di Mola, Antonia; de Caprariis, Paolo; La Colla, Paolo; Loddo, Roberta; Altamura, Sergio; Maga, Giovanni; Filosa, Rosanna 分享 收藏
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