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Paul Gehrtz

university of regensburg

15H指数
309论文数
2.1K被引数
收录论文 14
发表时间
OICR-41103 as a chemical probe for the DCAF1 WD40 domainOICR-41103 作为 DCAF1 WD40 结构域的化学探针
err2025-07-19
err0
errOAAI
errSerah W. Kimani; Mahmoud Noureldin; Brian Wilson; Laurent Hoffer; Stuart R. Green; Magdalena M. Szewczyk; Héctor González-Álvarez; Mohammed Mohammed; Manuel Chan; Chiara Krausser; Alice Shi Ming Li; Taraneh Hajian; Sarah Tucker; Dhananjay Joshi; Punit Saraon; Brigitte Thériault; Ji Sup Kim; Vijayaratnam Santhakumar; Peter Loppnau; Yanjun Li; Almagul Seitova; Aiping Dong; Taira Kiyota; Tobias Hammann; Paul Gehrtz; Bhashant Patel; Vaibhavi Rathod; Anand Vala; Bhimsen Rout; Paras Jagodra; Peter J. Brown; Ahmed Aman; Jailall Ramnauth; Gennady Poda; David Uehling; Cheryl H. Arrowsmith; Dalia Barsyte-Lovejoy; Richard Marcellus; Suzanne Ackloo; Ahmed Mamai; Rima Al-awar; Levon Halabelian
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Workflow for E3 Ligase Ligand Validation for PROTAC Development
err2025-02-11
err0
errOAAI
errMiletic, Nebojsa; Weckesser, Janik; Mosler, Thorsten; Rathore, Rajeshwari; Hoffmann, Marina E.; Gehrtz, Paul; Schlesiger, Sarah; Hartung, Ingo V.; Berner, Nicola; Wilhelm, Stephanie; Mueller, Juliane; Adhikari, Bikash; Nemec, Vaclav; Sivashanmugam, Saran Aswathaman; Elson, Lewis; Holzmann, Hanna; Schwalm, Martin P.; Hoffmann, Lasse; Azeez, Kamal Rayees Abdul; Mueller, Susanne; Kuster, Bernhard; Wolf, Elmar; Dikic, Ivan; Knapp, Stefan
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Optimization of Covalent MKK7 Inhibitors via Crude Nanomole- Scale Libraries
err2022-07-30
err8
errOAAI
errGehrtz, Paul; Marom, Shir; Buehrmann, Mike; Hardick, Julia; Kleinboelting, Silke; Shraga, Amit; Dubiella, Christian; Gabizon, Ronen; Wiese, Jan N.; Mueller, Matthias P.; Cohen, Galit; Babaev, Ilana; Shurrush, Khriesto; Avram, Liat; Resnick, Efrat; Barr, Haim; Rauh, Daniel; London, Nir
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An automatic pipeline for the design of irreversible derivatives identifies a potent SARS-CoV-2 Mpro inhibitor
err2021-12-01
err54
errOAAI
errZaidman, Daniel; Gehrtz, Paul; Filep, Mihajlo; Fearon, Daren; Gabizon, Ronen; Douangamath, Alice; Prilusky, Jaime; Duberstein, Shirly; Cohen, Galit; Owen, C. David; Resnick, Efrat; Strain-Damerell, Claire; Lukacik, Petra; Barr, Haim; Walsh, Martin A.; von Delft, Frank; London, Nir
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Crystallographic and electrophilic fragment screening of the SARS-CoV-2 main protease
err2020-10-07
err223
errOAAI
errDouangamath, Alice; Fearon, Daren; Gehrtz, Paul; Krojer, Tobias; Lukacik, Petra; Owen, C. David; Resnick, Efrat; Strain-Damerell, Claire; Aimon, Anthony; Abranyi-Balogh, Peter; Brandao-Neto, Jose; Carbery, Anna; Davison, Gemma; Dias, Alexandre; Downes, Thomas D.; Dunnett, Louise; Fairhead, Michael; Firth, James D.; Jones, S. Paul; Keeley, Aaron; Keserue, Gyoergy M.; Klein, Hanna F.; Martin, Mathew P.; Noble, Martin E. M.; O'Brien, Peter; Powell, Ailsa; Reddi, Rambabu N.; Skyner, Rachael; Snee, Matthew; Waring, Michael J.; Wild, Conor; London, Nir; von Delft, Frank; Walsh, Martin A.
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Efficient Targeted Degradation via Reversible and Irreversible Covalent PROTACs (May, 10.1021/jacs.9b13907, 2020)通过可逆和不可逆的共价protac进行有效的靶向降解 (may, 10.1021/jacs.9b13907,2020)
err2020-06-10
err10
errOAAI
errGabizon, Ronen; Shraga, Amit; Gehrtz, Paul; Livnah, Ella; Shorer, Yamit; Gurwicz, Neta; Avram, Liat; Unger, Tamar; Aharoni, Hila; Albeck, Shira; Brandis, Alexander; Shulman, Ziv; Katz, Ben-Zion; Herishanu, Yair; London, Nir
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Efficient Targeted Degradation via Reversible and Irreversible Covalent PROTACs
err2020-05-05
err138
errOAAI
errGabizon, Ronen; Shraga, Amit; Gehrtz, Paul; Livnah, Ella; Shorer, Yamit; Gurwicz, Neta; Avram, Liat; Unger, Tamar; Aharoni, Hila; Albeck, Shira; Brandis, Alexander; Shulman, Ziv; Katz, Ben-Zion; Herishanu, Yair; London, Nir
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Tandem Acyl Substitution/Michael Addition of Thioesters with Vinylmagnesium Bromide
err2019-04-01
err12
PREAI
errHirschbeck, Vera; Boeldl, Marlene; Gehrtz, Paul H.; Fleischer, Ivana
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Cross-Coupling of Chloro(hetero)arenes with Thiolates Employing a Ni(0)-Precatalyst
err2018-12-17
err37
PREAI
errGehrtz, Paul H.; Geiger, Valentin; Schmidt, Tanno; Srsan, Laura; Fleischer, Ivana
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Nickel-Catalyzed Coupling of Arylzinc Halides with Thioesters
err2018-05-25
err26
PREAI
errGehrtz, Paul H.; Kathe, Prasad; Fleischer, Ivana
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Metal-Catalyzed Synthesis and Use of Thioesters: Recent Developments
err2018-02-05
err146
PREAI
errHirschbeck, Vera; Gehrtz, Paul H.; Fleischer, Ivana
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Regioselective Thiocarbonylation of Vinyl Arenes
err2016-12-14
err93
PREAI
errHirschbeck, Vera; Gehrtz, Paul H.; Fleischer, Ivana
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