未登录 分享 收藏
分享 收藏
Coupling the Antimalarial Cell Penetrating Peptide TP10 to Classical Antimalarial Drugs Primaquine and Chloroquine Produces Strongly Hemolytic Conjugates Aguiar, Luisa; Biosca, Arnau; Lantero, Elena; Gut, Jiri; Vale, Nuno; Rosenthal, Philip J.; Nogueira, Fatima; Andreu, David; Fernandez-Busquets, Xavier; Gomes, Paula 分享 收藏
Identification of a potent benzoxaborole drug candidate for treating cryptosporidiosis Lunde, Christopher S.; Stebbins, Erin E.; Jumani, Rajiv S.; Hasan, Md Mahmudul; Miller, Peter; Barlow, John; Freund, Yvonne R.; Berry, Pamela; Stefanakis, Rianna; Gut, Jiri; Rosenthal, Philip J.; Love, Melissa S.; McNamara, Case W.; Easom, Eric; Plattner, Jacob J.; Jacobs, Robert T.; Huston, Christopher D. 分享 收藏
Falcipain Inhibitors Based on the Natural Product Gallinamide A Are Potent in Vitro and in Vivo Antimalarials Stoye, Alexander; Juillard, Annette; Tang, Arthur H.; Legac, Jennifer; Gut, Jiri; White, Karen L.; Charman, Susan A.; Rosenthal, Philip J.; Grau, Georges E. R.; Hunt, Nicholas H.; Payne, Richard J. 分享 收藏
Efficacy of subcutaneous doses and a new oral amorphous solid dispersion formulation of flubendazole on male jirds (Meriones unguiculatus) infected with the filarial nematode Brugia pahangi Fischer, Chelsea; Urriza, Iosune Ibiricu; Bulman, Christina A.; Lim, K. C.; Gut, Jiri; Lachau-Durand, Sophie; Engelen, Marc; Quirynen, Ludo; Tekle, Fetene; Baeten, Benny; Beerntsen, Brenda; Lustigman, Sara; Sakanari, Judy 分享 收藏
[(7-CHLOROQUINOLIN-4-YL)AMINO]ACETOPHENONES AND THEIR COPPER(II) DERIVATIVES: SYNTHESIS, CHARACTERIZATION, COMPUTATIONAL STUDIES AND ANTIMALARIAL ACTIVITY Parra, Yonathan de J.; Andueza L, Felix D.; Ferrer M, Rosa E.; Bruno Colmenarez, Julia; Acosta, Maria E.; Charris, Jaime; Rosenthal, Philip J.; Gut, Jiri 分享 收藏
Endoperoxide-8-aminoquinoline hybrids as dual-stage antimalarial agents with enhanced metabolic stability Capela, Rita; Magalhaes, Joana; Miranda, Daniela; Machado, Marta; Sanches-Vaz, Margarida; Albuquerque, Ines S.; Sharma, Moni; Gut, Jiri; Rosenthal, Philip J.; Frade, Raquel; Perry, Maria J.; Moreira, Rui; Prudencio, Miguel; Lopes, Francisca 分享 收藏
分享 收藏
分享 收藏
Development of Novel Peptide-Based Michael Acceptors Targeting Rhodesain and Falcipain-2 for the Treatment of Neglected Tropical Diseases (NTDs) Previti, Santo; Ettari, Roberta; Cosconati, Sandro; Arnendola, Giorgio; Chouchene, Khawla; Wagner, Annika; Hellmich, Ute A.; Ulrich, Kathrin; Krauth-Siegel, R. Luise; Wich, Peter R.; Schmid, Ira; Schirmeister, Tanja; Gut, Jiri; Rosenthal, Philip J.; Grasso, Silvana; Zappala, Maria 分享 收藏
分享 收藏
分享 收藏
A potent antimalarial benzoxaborole targets a Plasmodium falciparum cleavage and polyadenylation specificity factor homologue Sonoiki, Ebere; Ng, Caroline L.; Lee, Marcus C. S.; Guo, Denghui; Zhang, Yong-Kang; Zhou, Yasheen; Alley, M. R. K.; Ahyong, Vida; Sanz, Laura M.; Jose Lafuente-Monasterio, Maria; Dong, Chen; Schupp, Patrick G.; Gut, Jiri; Legac, Jenny; Cooper, Roland A.; Gamo, Francisco-Javier; DeRisi, Joseph; Freund, Yvonne R.; Fidock, David A.; Rosenthal, Philip J. 分享 收藏
分享 收藏
Cryptosporidium and Toxoplasma Parasites Are Inhibited by a Benzoxaborole Targeting Leucyl-tRNA Synthetase Palencia, Andres; Liu, Ru-Juan; Lukarska, Maria; Gut, Jiri; Bougdour, Alexandre; Touquet, Bastien; Wang, En-Duo; Li, Xianfeng; Alley, M. R. K.; Freund, Yvonne R.; Rosenthal, Philip J.; Hakimi, Mohamed-Ali; Cusack, Stephen 分享 收藏
Probing the Azaaurone Scaffold against the Hepatic and Erythrocytic Stages of Malaria Parasites Carrasco, Marta P.; Machado, Marta; Goncalves, Lidia; Sharma, Moni; Gut, Jiri; Lukens, Amanda K.; Wirth, Dyann F.; Andre, Vania; Duarte, Maria Teresa; Guedes, Rita C.; dos Santos, Daniel J. V. A.; Rosenthal, Philip J.; Mazitschek, Ralph; Prudencio, Miguel; Moreira, Rui 分享 收藏
Antimalarial Benzoxaboroles Target Plasmodium falciparum Leucyl-tRNA Synthetase Sonoiki, Ebere; Palencia, Andres; Guo, Denghui; Ahyong, Vida; Dong, Chen; Li, Xianfeng; Hernandez, Vincent S.; Zhang, Yong-Kang; Choi, Wai; Gut, Jiri; Legac, Jennifer; Cooper, Roland; Alley, M. R. K.; Freund, Yvonne R.; DeRisi, Joseph; Cusack, Stephen; Rosenthal, Philip J. 分享 收藏
分享 收藏
Enantiopure Indolizinoindolones with in vitro Activity against Blood- and Liver-Stage Malaria Parasites Pereira, Nuno A. L.; Monteiro, Angelo; Machado, Marta; Gut, Jiri; Molins, Elies; Perry, M. Jesus; Dourado, Jorge; Moreira, Rui; Rosenthal, Philip J.; Prudencio, Miguel; Santos, Maria M. M. 分享 收藏