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M.A. Convery

university of michigan system

26H指数
155论文数
2.2K被引数
收录论文 22
发表时间
Optimization of Potent and Selective Cyclohexyl Acid ERAP1 Inhibitors Using Structure- and Property-Based Drug Design
err2024-11-06
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errOAAI
errHryczanek, Ross P.; Hackett, Andrew S.; Rowland, Paul; Chung, Chun-wa; Convery, Maire A.; Holmes, Duncan S.; Hutchinson, Jonathan P.; Kitchen, Semra; Korczynska, Justyna; Law, Robert P.; Lea, Jonathan D.; Liddle, John; Lonsdale, Richard; Neu, Margarete; Nickels, Leng; Phillipou, Alex; Rowedder, James E.; Schneck, Jessica L.; Scott-Stevens, Paul; Sheehan, Hester; Tayler, Chloe L.; Temponeras, Ioannis; Tinworth, Christopher P.; Walker, Ann L.; Wojno-Picon, Justyna; Young, Robert J.; Lindsay, David M.; Stratikos, Efstratios
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Discovery of GSK251: A Highly Potent, Highly Selective, Orally Bioavailable Inhibitor of PI3Kδ with a Novel Binding Mode
err2021-09-11
err3
PREAI
errDown, Kenneth; Amour, Augustin; Anderson, Niall A.; Barton, Nick; Campos, Sebastien; Cannons, Edward P.; Clissold, Cole; Convery, Maire A.; Coward, John J.; Doyle, Kevin; Duempelfeld, Birgit; Edwards, Christopher D.; Goldsmith, Michael D.; Krause, Jana; Mallett, David N.; McGonagle, Grant A.; Patel, Vipulkumar K.; Rowedder, James; Rowland, Paul; Sharpe, Andrew; Sriskantharajah, Srividya; Thomas, Daniel A.; Thomson, Douglas W.; Uddin, Sorif; Hamblin, J. Nicole; Hessel, Edith M.
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GSK137, a potent small-molecule BCL6 inhibitor with in vivo activity, suppresses antibody responses in mice
err2021-08-01
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errOAAI
errPearce, Andrew C.; Bamford, Mark J.; Barber, Ruth; Bridges, Angela; Convery, Maire A.; Demetriou, Constantinos; Evans, Sian; Gobbetti, Thomas; Hirst, David J.; Holmes, Duncan S.; Hutchinson, Jonathan P.; Jayne, Sandrine; Lezina, Larissa; McCabe, Michael T.; Messenger, Cassie; Morley, Joanne; Musso, Melissa C.; Scott-Stevens, Paul; Manso, Ana Sousa; Schofield, Jennifer; Slocombe, Tom; Somers, Don; Walker, Ann L.; Wyce, Anastasia; Zhang, Xi-Ping; Wagner, Simon D.
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Design and Development of a Macrocyclic Series Targeting Phosphoinositide 3-Kinase δ
err2020-06-03
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errOAAI
errSpencer, Jonathan A.; Baldwin, Ian R.; Barton, Nick; Chung, Chun-Wa; Convery, Maire A.; Edwards, Christopher D.; Jamieson, Craig; Mallett, David N.; Rowedder, James E.; Rowland, Paul; Thomas, Daniel A.; Hardy, Charlotte J.
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Identification of Quinoline-Based RIP2 Kinase Inhibitors with an Improved Therapeutic Index to the hERG Ion Channel (vol 9, pg 1039, 2018)
err2020-06-02
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errOAAI
errHaile, Pamela A.; Casillas, Linda N.; Bury, Michael J.; Mehlmann, John F.; Singhaus, Robert, Jr.; Charnley, Adam K.; Hughes, Terry V.; DeMartino, Michael P.; Wang, Gren Z.; Romano, Joseph J.; Dong, Xiaoyang; Plotnikov, Nikolay V.; Lakdawala, Ami S.; Duraiswami, Chaya; Convery, Maire A.; Votta, Bartholomew J.; Lipshutz, David B.; Desai, Biva M.; Swift, Barbara; Capriotti, Carol A.; Berger, Scott B.; Mahajan, Mukesh K.; Reilly, Michael A.; Rivera, Elizabeth J.; Sun, Helen H.; Nagilla, Rakesh; LePage, Carol; Ouellette, Michael T.; Totoritis, Rachel D.; Donovan, Brian T.; Brown, Barry S.; Chaudhary, Khuram W.; Gough, Peter J.; Bertin, John; Marquis, Robert W.
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Optimization of Orally Bioavailable PI3Kδ Inhibitors and Identification of Vps34 as a Key Selectivity Target口服可生物利用的PI3Kδ 抑制剂的优化和Vps34作为关键选择性靶标的鉴定
err2019-12-19
err19
PREAI
errHenley, Zoe A.; Amour, Augustin; Barton, Nick; Bantscheff, Marcus; Bergamini, Giovanna; Bertrand, Sophie M.; Convery, Maire; Down, Kenneth; Duempelfeld, Birgit; Edwards, Chris D.; Grandi, Paola; Gore, Paul M.; Keeling, Steve; Livia, Stefano; Mallett, David; Maxwell, Aoife; Price, Mark; Rau, Christina; Reinhard, Friedrich B. M.; Rowedder, James; Rowland, Paul; Taylor, Jonathan A.; Thomas, Daniel A.; Hessel, Edith M.; Hamblin, J. Nicole
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Discovery of Pyrazolocarboxamides as Potent and Selective Receptor Interacting Protein 2 (RIP2) Kinase Inhibitors
err2019-10-11
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errOAAI
errHaffner, Curt D.; Charnley, Adam K.; Aquino, Christopher J.; Casillas, Linda; Convery, Maire A.; Cox, Julie A.; Elban, Mark A.; Goodwin, Nicole C.; Gough, Peter J.; Haile, Pamela A.; Hughes, Terry V.; Knapp-Reed, Beth; Kreatsoulas, Constantine; Lakdawala, Ami S.; Li, Huijie; Lian, Yiqian; Lipshutz, David; Mehlmann, John F.; Ouellette, Michael; Romano, Joseph; Shewchuk, Lisa; Shu, Arthur; Votta, Bartholomew J.; Zhou, Huiqiang; Bertin, John; Marquis, Robert W.
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Discovery of 3-Oxabicyclo[4.1.0]heptane, a Non-nitrogen Containing Morpholine Isostere, and Its Application in Novel Inhibitors of the PI3K-AKT-mTOR Pathway (vol 62, pg 6972, 2019)
err2019-09-25
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errOAAI
errHobbs, Heather; Bravi, Gianpaolo; Campbell, Ian; Convery, Maire; Davies, Hannah; Inglis, Graham; Pal, Sandeep; Peace, Simon; Redmond, Joanna; Summers, Declan
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Discovery of 3-Oxabicyclo[4.1.0]heptane, a Non-nitrogen Containing Morpholine Isostere, and Its Application in Novel Inhibitors of the PI3K-AKT-mTOR Pathway
err2019-07-08
err19
PREAI
errHobbs, Heather; Bravi, Gianpaolo; Campbell, Ian; Convery, Maire; Davies, Hannah; Inglis, Graham; Pal, Sandeep; Peace, Simon; Redmond, Joanna; Summers, Declan
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Discovery of a First-in-Class Receptor Interacting Protein 2 (RIP2) Kinase Specific Clinical Candidate, 2-((4-(Benzo[d]thiazol-5-ylamino)-6-(tert-butylsulfonyl)quinazolin-7-yl)oxy)ethyl Dihydrogen Phosphate, for the Treatment of Inflammatory Diseases
err2019-07-02
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errHaile, Pamela A.; Casillas, Linda N.; Votta, Bartholomew J.; Wang, Gren Z.; Charnley, Adam K.; Dong, Xiaoyang; Bury, Michael J.; Romano, Joseph J.; Mehlmann, John F.; King, Bryan W.; Erhard, Karl F.; Hanning, Charles R.; Lipshutz, David B.; Desai, Biva M.; Capriotti, Carol A.; Schaeffer, Michelle C.; Berger, Scott B.; Mahajan, Mukesh K.; Reilly, Michael A.; Nagilla, Rakesh; Rivera, Elizabeth J.; Sun, Helen H.; Kenna, John K.; Beal, Allison M.; Ouellette, Michael T.; Kelly, Mike; Stemp, Gillian; Convery, Maire A.; Vossenkamper, Anna; MacDonald, Thomas T.; Gough, Peter J.; Bertin, John; Marquis, Robert W.
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Discovery of Potent, Efficient, and Selective Inhibitors of Phosphoinositide 3-Kinase δ through a Deconstruction and Regrowth Approach
err2018-12-11
err10
PREAI
errBarton, Nick; Convery, Maire; Cooper, Anthony W. J.; Down, Kenneth; Hamblin, J. Nicole; Inglis, Graham; Peace, Simon; Rowedder, James; Rowland, Paul; Taylor, Jonathan A.; Wellaway, Natalie
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Identification of Quinoline-Based RIP2 Kinase Inhibitors with an Improved Therapeutic Index to the hERG Ion Channel
err2018-09-26
err29
errOAAI
errHaile, Pamela A.; Casillas, Linda N.; Bury, Michael J.; Mehlmann, John F.; Singhaus, Robert, Jr.; Charnley, Adam K.; Hughes, Terry V.; DeMartino, Michael P.; Wang, Gren Z.; Romano, Joseph J.; Dong, Xiaoyang; Plotnikov, Nikolay V.; Lakdawala, Ami S.; Convery, Maire A.; Votta, Bartholomew J.; Lipshutz, David B.; Desai, Biva M.; Swift, Barbara; Capriotti, Carol A.; Berger, Scott B.; Mahajan, Mukesh K.; Reilly, Michael A.; Rivera, Elizabeth J.; Sun, Helen H.; Nagilla, Rakesh; LePage, Carol; Ouellette, Michael T.; Totoritis, Rachel D.; Donovan, Brian T.; Brown, Barry S.; Chaudhary, Khuram W.; Gough, Peter J.; Bertin, John; Marquis, Robert W.
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Screening of a Novel Fragment Library with Functional Complexity against Mycobacterium tuberculosis InhA
err2018-02-19
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errPrati, Federica; Zuccotto, Fabio; Fletcher, Daniel; Convery, Maire A.; Fernandez-Menendez, Raquel; Bates, Robert; Encinas, Lourdes; Zeng, Jingkun; Chung, Chun-wa; De Dios Anton, Paco; Mendoza-Losana, Alfonso; Mackenzie, Claire; Green, Simon R.; Huggett, Margaret; Barros, David; Wyatt, Paul G.; Ray, Peter C.
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Selectively Targeting the Kinome-Conserved Lysine of PI3Kδ as a General Approach to Covalent Kinase Inhibition选择性靶向PI3Kδ 的激酶保守赖氨酸作为共价激酶抑制的一般方法
err2018-01-09
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errDalton, Samuel E.; Dittus, Lars; Thomas, Daniel A.; Convery, Maire A.; Nunes, Joao; Bush, Jacob T.; Evans, John P.; Werner, Thilo; Bantscheff, Marcus; Murphy, John A.; Campos, Sebastien
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CSAR 2014: A Benchmark Exercise Using Unpublished Data from Pharma
err2016-05-17
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errCarlson, Heather A.; Smith, Richard D.; Damm-Ganamet, Kelly L.; Stuckey, Jeanne A.; Ahmed, Aqeel; Convery, Maire A.; Somers, Donald O.; Kranz, Michael; Elkins, Patricia A.; Cui, Guanglei; Peishoff, Catherine E.; Lambert, Millard H.; Dunbar, James B., Jr.
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The Identification and Pharmacological Characterization of 6-(tert-Butylsulfonyl)-N-(5-fluoro-1H-indazol-3-yl)quinolin-4-amine (GSK583), a Highly Potent and Selective Inhibitor of RIP2 Kinase
err2016-05-04
err100
PREAI
errHaile, Pamela A.; Votta, Bartholomew J.; Marquis, Robert W.; Bury, Michael J.; Mehlmann, John F.; Singhaus, Robert, Jr.; Charnley, Adam K.; Lakdawala, Ami S.; Convery, Maire A.; Lipshutz, David B.; Desai, Biva M.; Swift, Barbara; Capriotti, Carol A.; Berger, Scott B.; Mahajan, Mukesh K.; Reilly, Michael A.; Rivera, Elizabeth J.; Sun, Helen H.; Nagilla, Rakesh; Beal, Allison M.; Finger, Joshua N.; Cook, Michael N.; King, Bryan W.; Ouellette, Michael T.; Totoritis, Rachel D.; Pierdomenico, Maria; Negroni, Anna; Stronati, Laura; Cucchiara, Salvatore; Ziolkowski, Bartlomiej; Vossenkamper, Anna; MacDonald, Thomas T.; Gough, Peter J.; Bertin, John; Casillas, Linda N.
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New direct inhibitors of InhA with antimycobacterial activity based on a tetrahydropyran scaffold
err2016-04-01
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PREAI
errPajk, Stane; Zivec, Matej; Sink, Roman; Sosic, Izidor; Neu, Margarete; Chung, Chun-wa; Martinez-Hoyos, Maria; Perez-Herran, Esther; Alvarez-Gomez, Daniel; Alvarez-Ruiz, Emilio; Mendoza-Losana, Alfonso; Castro-Pichel, Julia; Barros, David; Ballell-Pages, Lluis; Young, Robert J.; Convery, Maire A.; Encinas, Lourdes; Gobec, Stanislav
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N-Benzyl-4-((heteroaryl)methyl)benzamides: A New Class of Direct NADH-Dependent 2-trans Enoyl-Acyl Carrier Protein Reductase (InhA) Inhibitors with Antitubercular Activity
err2016-03-02
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PREAI
errGuardia, Ana; Gulten, Gulcin; Fernandez, Raquel; Gomez, Jesus; Wang, Feng; Convery, Maire; Blanco, Delia; Martinez, Maria; Perez-Herran, Esther; Alonso, Marta; Ortega, Fatima; Rullas, Joaquin; Calvo, David; Mata, Lydia; Young, Robert; Sacchettini, James C.; Mendoza-Losana, Alfonso; Remuinan, Modesto; Ballell Pages, Lluis; Castro-Pichel, Julia
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Crystal structures of human RIP2 kinase catalytic domain complexed with ATP-competitive inhibitors: Foundations for understanding inhibitor selectivity
err2015-11-01
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PREAI
errCharnley, Adam K.; Convery, Maire A.; Shah, Ami Lakdawala; Jones, Emma; Hardwicke, Philip; Bridges, Angela; Ouellette, Michael; Totoritis, Rachel; Schwartz, Benjamin; King, Bryan W.; Wisnoski, David D.; Kang, James; Eidam, Patrick M.; Votta, Bartholomew J.; Gough, Peter J.; Marquis, Robert W.; Bertin, John; Casillas, Linda
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Encoded Library Technology as a Source of Hits for the Discovery and Lead Optimization of a Potent and Selective Class of Bactericidal Direct Inhibitors of Mycobacterium tuberculosis InhA
err2014-02-05
err115
PREAI
errEncinas, Lourdes; O'Keefe, Heather; Neu, Margarete; Remuinan, Modesto J.; Patel, Amish M.; Guardia, Ana; Davie, Christopher P.; Perez-Macias, Natalia; Yang, Hongfang; Convery, Maire A.; Messer, Jeff A.; Perez-Herran, Esther; Centrella, Paolo A.; Alvarez-Gomez, Daniel; Clark, Matthew A.; Huss, Sophie; O'Donovan, Gary K.; Ortega-Muro, Fatima; McDowell, William; Castaneda, Pablo; Arico-Muendel, Christopher C.; Pajk, Stane; Rullas, Joaquin; Angulo-Barturen, Inigo; Alvarez-Ruiz, Emilio; Mendoza-Losana, Alfonso; Pages, Lluis Ballell; Castro-Pichel, Julia; Evindar, Ghotas
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