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Anil Vasudevan

technology and therapeutic platforms, discovery research, abbvie inc., north chicago, illinois 60064, united states

33H指数
144论文数
2.7K被引数
收录论文 40
发表时间
Proteome-Wide Discovery of Degradable Proteins Using Bifunctional Molecules利用双功能分子进行全蛋白质组降解蛋白的发现
err2025-10-21
err0
errOAAI
errInes Forrest; Louis P. Conway; Clara Gathmann; Appaso M. Jadhav; Tzu-Yuan Chiu; Christian M. Chaheine; Michelle Estrada; Anurupa Shrestha; Kathy Sarris; Justin M. Reitsma; Scott E. Warder; Anil Vasudevan; Shaun M. McLoughlin; Christopher G. Parker
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Discovery of a tau-aggregate clearing compound that covalently targets P4HB靶向P4HB并清除tau聚集物的共价化合物发现
err2025-10-06
err0
PREAI
errLouis P. Conway; Michelle A. Estrada; Weichao Li; Stephen Walker; Benjamin Mielich-Süss; Anurupa Shrestha; Matthew Townsend; Jürgen Korffmann; Greg Potts; Janice Lee; Kenneth P. Robinson; Shiyao Wang; Brian Bierie; John R. Koenig; Phil Cox; Paul Richardson; Manisha Jhala; Becca McCloud; Sujatha Gopalakrishnan; Kevin Woller; Anil Vasudevan; Scott E. Warder; Shaun M. McLoughlin; Christopher G. Parker
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Discovery of Orally Efficacious Bridged Piperazines as smTNF Modulators作为口服有效的桥连哌嗪的smTNF调节剂的发现
err2025-07-09
err0
PREAI
errZhiguo Bian; Robert G. Schmidt; Noel S. Wilson; David B. Duignan; Eric Breinlinger; Amanda W. Dombrowski; Paul Erdman; C. Michael Foley; Michael Friedman; Gregory A. Gfesser; Christian A. Goess; Arthur Gomtsyan; Russell A. Judge; Ryota Kikuchi; Yevgeniya Koshman; Xiaoqin Liu; Kenton L. Longenecker; Andrea McClure; Kevin Sippy; Jill M. Wetter; Robert Stoffel; Anil Vasudevan
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Harnessing the FBXW7 Somatic Mutant R465C for Targeted Protein Degradation利用FBXW7体细胞突变体R465C进行靶向蛋白降解
err2025-02-06
err0
errOAAI
errBasu, Ananya A.; Zhang, Chenlu; Rouhimoghadam, Milad; Vasudevan, Anil; Reitsma, Justin M.; Zhang, Xiaoyu
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Quantitative Measurement of Rate of Targeted Protein Degradation
err2024-07-09
err6
PREAI
errLynch, Thomas L.; Marin, Violeta L.; McClure, Ryan A.; Phipps, Colin; Ronau, Judith A.; Rouhimoghadam, Milad; Adams, Ashley M.; Kandi, Soumya; Wolke, Malerie L.; Shergalis, Andrea G.; Potts, Gregory K.; Nacham, Omprakash; Richardson, Paul; Kakavas, Stephan J.; Chhor, Gekleng; Jenkins, Gary J.; Woller, Kevin R.; Warder, Scott E.; Vasudevan, Anil; Reitsma, Justin M.
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Antibacterial bone adhesive cement for preventing sternal infections after cardiac surgery
err2023-05-01
err6
PREAI
errPradeep, Aathira; Varma, Praveen Kerala; Arumugam, Thennavan; Vijayan, Anjaly Maravattikal; Vasudevan, Anil Kumar; Rangasamy, Jayakumar
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CRISPR Screen Reveals BRD2/4 Molecular Glue-like Degrader via Recruitment of DCAF16CRISPR筛选通过招募DCAF16揭示了BRD2/4分子胶样降解剂
err2023-01-19
err42
PREAI
errShergalis, Andrea G.; Marin, Violeta L.; Rhee, David Y.; Senaweera, Sameera; McCloud, Rebecca L.; Ronau, Judith A.; Hutchins, Charles W.; McLoughlin, Shaun; Woller, Kevin R.; Warder, Scott E.; Vasudevan, Anil; Reitsma, Justin M.
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Identification and structure-based drug design of cell-active inhibitors of interleukin 17A at a novel C-terminal site
err2022-08-26
err8
errOAAI
errGoedken, Eric R.; Argiriadi, Maria A.; Dietrich, Justin D.; Petros, Andrew M.; Krishnan, Navasona; Panchal, Sanjay C.; Qiu, Wei; Wu, Haihong; Zhu, Haizhong; Adams, Ashley M.; Bodelle, Pierre M.; Goguen, Lucas; Richardson, Paul L.; Slivka, Peter F.; Srikumaran, Myron; Upadhyay, Anup K.; Wu, Bainan; Judge, Russell A.; Vasudevan, Anil; Gopalakrishnan, Sujatha M.; Cox, Philip B.; Stoll, Vincent S.; Sun, Chaohong
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Development of Orally Efficacious Allosteric Inhibitors of TNFα via Fragment-Based Drug Design
err2020-12-30
err21
PREAI
errDietrich, Justin D.; Longenecker, Kenton L.; Wilson, Noel S.; Goess, Christian; Panchal, Sanjay C.; Swann, Steven L.; Petros, Andrew M.; Hobson, Adrian D.; Ihle, David; Song, Danying; Richardson, Paul; Comess, Kenneth M.; Cox, Philip B.; Dombrowski, Amanda; Sarris, Kathy; Donnelly-Roberts, Diana L.; Duignan, David B.; Gomtsyan, Arthur; Jung, Paul; Krueger, A. Chris; Mathieu, Suzanne; McClure, Andrea; Stoll, Vincent S.; Wetter, Jill; Mankovich, John A.; Hajduk, Philip J.; Vasudevan, Anil; Stoffel, Robert H.; Sun, Chaohong
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A Dual-Purpose Bromocoumarin Tag Enables Deep Profiling of the Cellular Cysteinome
err2019-05-08
err0
PREAI
errRabalski, Adam J.; Williams, Jon D.; McClure, Ryan A.; Vasudevan, Anil; Baranczak, Aleksandra
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Combination of Repurposed Drug Diosmin with Amoxicillin-Clavulanic acid Causes Synergistic Inhibition of Mycobacterial Growth
err2019-05-01
err32
errOAAI
errPushkaran, Anju Choorakottayil; Vinod, Vivek; Vanuopadath, Muralidharan; Nair, Sudarslal Sadasivan; Nair, Shantikumar V.; Vasudevan, Anil Kumar; Biswas, Raja; Mohan, Chethampadi Gopi
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Identification of Selective Dual ROCK1 and ROCK2 Inhibitors Using Structure-Based Drug Design
err2018-11-01
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errOAAI
errHobson, Adrian D.; Judge, Russell A.; Aguirre, Ana L.; Brown, Brian S.; Cui, Yifang; Ding, Ping; Dominguez, Eric; DiGiammarino, Enrico; Egan, David A.; Freiberg, Gail M.; Gopalakrishnan, Sujatha M.; Harris, Christopher M.; Honore, Marie P.; Kage, Karen L.; Kapecki, Nicolas J.; Ling, Christopher; Ma, Junli; Mack, Helmut; Mamo, Mulugeta; Maurus, Stefan; McRae, Bradford; Moore, Nigel S.; Muellery, Bernhard K.; Mueller, Reinhold; Namovic, Marian T.; Patel, Kaushal; Pratt, Steve D.; Putman, C. Brent; Queeney, Kara L.; Sarris, Kathy K.; Schaffter, Lisa M.; Stoll, Vincent; Vasudevan, Anil; Wang, Lei; Wang, Lu; Wirthl, William; Yacht, Kimberly
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Discovery of Novel Aminotetralines and Aminochromanes as Selective and Competitive Glycine Transporter 1 (GlyT1) Inhibitors
err2018-08-06
err10
PREAI
errAmberg, Willi; Lange, Udo E. W.; Ochse, Michael; Pohlki, Frauke; Behl, Berthold; Relo, Ana Lucia; Hornberger, Wilfried; Hoft, Carolin; Mezler, Mario; Sydor, Jens; Wang, Ying; Zhao, Hongyu; Brewer, Jason T.; Dietrich, Justin; Li, Huanqiu; Akritopoulou-Zanze, Irini; Lao, Yanbin; Hannick, Steven M.; Ku, Yi-Yin; Vasudevan, Anil
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Novel Modes of Inhibition of Wild-Type Isocitrate Dehydrogenase 1 (IDH1): Direct Covalent Modification of His315
err2018-07-13
err38
PREAI
errJakob, Clarissa G.; Upadhyay, Anup K.; Donner, Pamela L.; Nicholl, Emily; Addo, Sadiya N.; Qiu, Wei; Ling, Christopher; Gopalakrishnan, Sujatha M.; Torrent, Maricel; Cepa, Steven P.; Shanley, Jason; Shoemaker, Alexander R.; Sun, Chaohong C.; Vasudevan, Anil; Woller, Kevin R.; Shotwell, J. Brad; Shaw, Bailin; Bian, Zhiguo; Hutti, Jessica E.
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De Novo Design, Synthesis, and Biological Evaluation of 3,4-Disubstituted Pyrrolidine Sulfonamides as Potent and Selective Glycine Transporter 1 Competitive Inhibitors
err2018-07-03
err15
PREAI
errWang, Ying; Zhao, Hongyu; Brewer, Jason T.; Li, Huanqiu; Lao, Yanbin; Amberg, Willi; Behl, Berthold; Akritopoulou-Zanze, Irini; Dietrich, Justin; Lange, Udo E. W.; Pohlki, Frauke; Hoft, Carolin; Hornberger, Wilfried; Djuric, Stevan W.; Sydor, Jens; Mezler, Mario; Relo, Ana Lucia; Vasudevan, Anil
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Emerging Approaches for the Identification of Protein Targets of Small Molecules - A Practitioners' Perspective
err2018-05-02
err56
PREAI
errComess, Kenneth M.; McLoughlin, Shaun M.; Oyer, Jon A.; Richardson, Paul L.; Stockmann, Henning; Vasudevan, Anil; Warder, Scott E.
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Understanding the adhesion mechanism of a mucin binding domain from Lactobacillus fermentum and its role in enteropathogen exclusion
err2018-04-01
err40
PREAI
errChatterjee, Maitrayee; Pushkaran, Anju Choorakottayil; Vasudevan, Anil Kumar; Menon, Krishna Kumar N.; Biswas, Raja; Mohan, Chethampadi Gopi
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Cell-Surface Receptor Ligand Interaction Analysis with Homogeneous Time-Resolved FRET and Metabolic Glycan Engineering: Application to Transmembrane and GPI-Anchored Receptors
err2017-11-09
err20
PREAI
errStockmann, Henning; Todorovic, Viktor; Richardson, Paul L.; Marin, Violeta; Scott, Victoria; Gerstein, Clare; Lake, Marc; Wang, Leyu; Sadhukhan, Ramkrishna; Vasudevan, Anil
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