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Y

Yves Chapleur

universite de lorraine
H指数:30
被引数:3,231
浏览量:0

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Carbohydrate-based peptidomimetics targeting neuropilin-1: Synthesis, molecular docking study and in vitro biological activities
BIOORGANIC & MEDICINAL CHEMISTRY
IF3
2016-11-0123
OAAI
Richard, Mylene; Chateau, Alicia; Jelsch, Christian; Didierjean, Claude; Manival, Xavier; Charron, Christophe; Maigret, Bernard; Barberi-Heyob, Muriel; Chapleur, Yves; Boura, Cedric; Pellegrini-Moise, Nadia
'Click' glycosylation of peptides through cysteine propargylation and CuAAC

通过半胱氨酸前列腺素化和CuAAC对肽进行 “点击” 糖基化

BIOORGANIC & MEDICINAL CHEMISTRY
IF3
2014-12-0129
PREAI
Lamande-Langle, Sandrine; Collet, Charlotte; Hensienne, Raphael; Vala, Christine; Chretien, Francoise; Chapleur, Yves; Mohamadi, Amel; Lacolley, Patrick; Regnault, Veronique
Optimization of troglitazone derivatives as potent anti-proliferative agents: Towards more active and less toxic compounds
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
IF5.9
2014-08-0129
PREAI
Bordessa, Andrea; Colin-Cassin, Christelle; Grillier-Vuissoz, Isabelle; Kuntz, Sandra; Mazerbourg, Sabine; Husson, Gauthier; Vo, Myriam; Flament, Stephane; Martin, Helene; Chapleur, Yves; Boisbrun, Michel
Cytotoxic effects of four Caryophyllaceae species extracts on macrophage cell lines
PHARMACEUTICAL BIOLOGY
IF4.8
2014-05-2716
PREAI
Gevrenova, R.; Joubert, O.; Mandova, Tsv.; Zaiou, M.; Chapleur, Y.; Henry, M.
PPARγ-Inactive Δ2-Troglitazone Independently Triggers ER Stress and Apoptosis in Breast Cancer Cells
MOLECULAR CARCINOGENESIS
IF3.2
2013-11-3018
PREAI
Colin-Cassin, Christelle; Yao, Xiao; Cerella, Claudia; Chbicheb, Sarra; Kuntz, Sandra; Mazerbourg, Sabine; Boisbrun, Michel; Chapleur, Yves; Diederich, Marc; Flament, Stephane; Grillier-Vuissoz, Isabelle
New Thiazolidinedione Derivatives With PPARgamma-independent Activity - High Inhibition of Breast Cancer Cell Proliferation With Low Toxicity Towards Human Hepatocytes
EUROPEAN JOURNAL OF CANCER
IF7.1
2012-07-010
OAAI
Colin, C.; Chbicheb, S.; Yao, X.; Bordessa, A.; Boisbrun, M.; Grillier-Vuissoz, I.; Kuntz, S.; Mazerbourg, S.; Chapleur, Y.; Flament, S.
Synthesis of new troglitazone derivatives: Anti-proliferative activity in breast cancer cell lines and preliminary toxicological study
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
IF5.9
2012-05-0165
PREAI
Salamone, Stephane; Colin, Christelle; Grillier-Vuissoz, Isabelle; Kuntz, Sandra; Mazerbourg, Sabine; Flament, Stephane; Martin, Helene; Richert, Lysiane; Chapleur, Yves; Boisbrun, Michel
Kinetic Study of the Rearrangement of Deuterium-Labeled 4′-O-Methylnorbelladine in Leucojum aestivum Shoot Cultures by Mass Spectrometry. Influence of Precursor Feeding on Amaryllidaceae Alkaloid Accumulation
JOURNAL OF NATURAL PRODUCTS
IF3.6
2011-10-2021
PRE
El Tahchy, Anna; Ptak, Agata; Boisbrun, Michel; Barre, Elvina; Guillou, Catherine; Dupire, Francois; Chretien, Francoise; Henry, Max; Chapleur, Yves; Laurain-Mattar, Dominique
Design, synthesis and antiproliferative activities of biarylolefins based on polyhydroxylated and carbohydrate scaffolds
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
IF5.9
2011-09-0121
PREAI
Novoa, Alexandre; Pellegrini-Moise, Nadia; Bourg, Stephane; Thoret, Sylviane; Dubois, Joelle; Aubert, Genevieve; Cresteil, Thierry; Chapleur, Yves
EGR1 expression: A calcium and ERK1/2 mediated PPARγ-independent event involved in the antiproliferative effect of 15-deoxy-Δ12,14-prostaglandin J2 and thiazolidinediones in breast cancer cells
BIOCHEMICAL PHARMACOLOGY
IF5.6
2011-05-0119
OAAI
Chbicheb, Sarra; Yao, Xiao; Rodeau, Jean-Luc; Salamone, Stephane; Boisbrun, Michel; Thiel, Gerald; Spohn, Daniel; Grillier-Vuissoz, Isabelle; Chapleur, Yves; Flament, Stephane; Mazerbourg, Sabine
Sugar-based peptidomimetics as potential inhibitors of the vascular endothelium growth factor binding to neuropilin-1
BIOORGANIC & MEDICINAL CHEMISTRY
IF3
2010-05-0145
PRE
Novoa, Alexandre; Pellegrini-Moise, Nadia; Bechet, Denise; Barberi-Heyob, Muriel; Chapleur, Yves
New troglitazone derivatives devoid of PPARγ agonist activity display an increased antiproliferative effect in both hormone-dependent and hormone-independent breast cancer cell lines
BREAST CANCER RESEARCH AND TREATMENT
IF3
2010-01-0723
OA
Colin, Christelle; Salamone, Stephane; Grillier-Vuissoz, Isabelle; Boisbrun, Michel; Kuntz, Sandra; Lecomte, Julie; Chapleur, Yves; Flament, Stephane
An Efficient Route to Acyclic C-Nucleosides and Fused-Ring Analogues of Uridine from exo-Glycals
JOURNAL OF ORGANIC CHEMISTRY
IF3.6
2009-09-3020
PRE
Enderlin, Gerald; Taillefumier, Claude; Didierjean, Claude; Chapleur, Yves
Synthesis and Solution Conformation of Homo-β-peptides Consisting of N-Mannofuranosyl-3-ulosonic acids
JOURNAL OF ORGANIC CHEMISTRY
IF3.6
2009-09-2328
PRE
Andreini, Manuel; Taillefumier, Claude; Chretien, Francoise; Thery, Vincent; Chapleur, Yves
LCMS and GCMS for the Screening of Alkaloids in Natural and in Vitro Extracts of Leucojum aestivum
JOURNAL OF NATURAL PRODUCTS
IF3.6
2008-12-3148
PRE
Ptak, Agata; El Tahchy, Anna; Dupire, Francois; Boisbrun, Michel; Henry, Max; Chapleur, Yves; Mos, Maria; Laurain-Mattar, Dominique
Disruption of ERα signalling pathway by PPARγ agonists: evidences of PPARγ-independent events in two hormone-dependent breast cancer cell lines
BREAST CANCER RESEARCH AND TREATMENT
IF3
2008-01-2033
PREAI
Lecomte, Julie; Flament, Stephane; Salamone, Stephane; Boisbrun, Michel; Mazerbourg, Sabine; Chapleur, Yves; Grillier-Vuissoz, Isabelle
Irreversible inhibition of glucose-6-phosphate dehydrogenase by the coenzyme A conjugate of ketoprofen:: A key to oxidative stress induced by non-steroidal anti-inflammatory drugs?
BIOCHEMICAL PHARMACOLOGY
IF5.6
2007-02-0135
PREAI
Asensio, Carine; Levoin, Nicolas; Guillaume, Cecile; Guerquin, Marie-Justine; Rouguieg, Koukeb; Chretien, Francoise; Chapleur, Yves; Netter, Patrick; Minn, Alain; Lapicque, Francoise
Elucidation of the mechanism of inhibition of cyclooxygenases by acyl-coenzyme A and acylglucuronic conjugates of ketoprofen
BIOCHEMICAL PHARMACOLOGY
IF5.6
2004-11-0114
PREAI
Levoin, N; Blondeau, C; Guillaume, C; Grandcolas, L; Chretien, F; Jouzeau, JY; Benoit, E; Chapleur, Y; Netter, P; Lapicque, F
Combining pharmacophore search, automated docking, and molecular dynamics simulations as a novel strategy for flexible docking.: Proof of concept:: Docking of arginine-glycine-aspartic acid-like compounds into the αvβ3 binding site
JOURNAL OF MEDICINAL CHEMISTRY
IF6.8
2004-07-2065
PREAI
Moitessier, N; Henry, C; Maigret, B; Chapleur, Y
Vitronectin Receptor -αVβ3 Integrin- Antagonists: Chemical and Structural Requirements for Activity and Selectivity
MINI-REVIEWS IN MEDICINAL CHEMISTRY
IF3.3
2002-12-0136
PREAI
Henry, Christophe; Moitessier, Nicolas; Chapleur, Yves

研究方向

暂未获取到该数据
M
Michel Boisbrun
H 指数:19论文数:98被引数:922
H 指数:0论文数:97被引数:0
S
Stéphane Flament
H 指数:28论文数:219被引数:2,549
I
Isabelle Grillier‐Vuissoz
H 指数:18论文数:70被引数:1,075
N
Nicolas Moitessier
H 指数:39论文数:205被引数:5,201
S
Sabine Mazerbourg
H 指数:23论文数:71被引数:2,943
C
Christelle Colin
H 指数:19论文数:95被引数:1,132
S
Sandra Kuntz
H 指数:16论文数:57被引数:567
S
Stéphane Salamone
H 指数:10论文数:32被引数:301
B
Bernard Maigret
H 指数:42论文数:210被引数:6,190