未登录 D3R Grand Challenge 3: blind prediction of protein-ligand poses and affinity rankings Gaieb, Zied; Parks, Conor D.; Chiu, Michael; Yang, Huanwang; Shao, Chenghua; Walters, W. Patrick; Lambert, Millard H.; Nevins, Neysa; Bembenek, Scott D.; Ameriks, Michael K.; Mirzadegan, Tara; Burley, Stephen K.; Amaro, Rommie E.; Gilson, Michael K. 分享 收藏
CSAR 2014: A Benchmark Exercise Using Unpublished Data from Pharma Carlson, Heather A.; Smith, Richard D.; Damm-Ganamet, Kelly L.; Stuckey, Jeanne A.; Ahmed, Aqeel; Convery, Maire A.; Somers, Donald O.; Kranz, Michael; Elkins, Patricia A.; Cui, Guanglei; Peishoff, Catherine E.; Lambert, Millard H.; Dunbar, James B., Jr. 分享 收藏
Structure of Rev-erbα bound to N-CoR reveals a unique mechanism of nuclear receptor-co-repressor interaction Phelan, Caroline A.; Gampe, Robert T., Jr.; Lambert, Millard H.; Parks, Derek J.; Montana, Valerie; Bynum, Jane; Broderick, Timothy M.; Hu, Xiao; Williams, Shawn P.; Nolte, Robert T.; Lazar, Mitchell A. 分享 收藏
Substituted 2-[(4-aminomethyl)phenoxy]-2-methylpropionic acid PPARα agonists.: 1.: Discovery of a novel series of potent HDLc raising agents Sierra, Michael L.; Beneton, Veronique; Boullay, Anne-Benedict; Boyer, Thierry; Brewster, Andrew G.; Donche, Frederic; Forest, Marie-Claire; Fouchet, Marie-Helene; Gellibert, Francoise J.; Grillot, Didier A.; Lambert, Millard H.; Laroze, Alain; Le Grumelec, Christelle; Linget, Jean Michel; Montana, Valerie G.; Nguyen, Van-Loc; Nicodeme, Edwige; Patel, Vipul; Penfornis, Annie; Pineau, Olivier; Pohin, Danig; Potvain, Florent; Poulain, Geraldine; Ruault, Cecile Bertho; Saunders, Michael; Toum, Jerome; Xu, H. Eric; Xu, Robert X.; Pianetti, Pascal M. 分享 收藏
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A ligand-mediated hydrogen bond network required for the activation of the mineralocorticoid receptor Bledsoe, RK; Madauss, KP; Holt, JA; Apolito, CJ; Lambert, MH; Pearce, KH; Stanley, TB; Stewart, EL; Trump, RP; Willson, TM; Williams, SP 分享 收藏
A critical assessment of docking programs and scoring functions Warren, Gregory L.; Andrews, C. Webster; Capelli, Anna-Maria; Clarke, Brian; LaLonde, Judith; Lambert, Millard H.; Lindvall, Mika; Nevins, Neysa; Semus, Simon F.; Senger, Stefan; Tedesco, Giovanna; Wall, Ian D.; Woolven, James M.; Peishoff, Catherine E.; Head, Martha S. 分享 收藏
A structural basis for constitutive activity in the human CAR/RXRα heterodimer Xu, RX; Lambert, MH; Wisely, BB; Warren, EN; Weinert, EE; Waitt, GM; Williams, JD; Collins, JL; Moore, LB; Willson, TM; Moore, JT 分享 收藏
Progesterone receptor ligand binding pocket flexibility: Crystal structures of the norethindrone and mometasone furoate complexes Madauss, KP; Deng, SJ; Austin, RJH; Lambert, MH; McLay, I; Pritchard, J; Short, SA; Stewart, EL; Uings, IJ; Williams, SP 分享 收藏
X-ray crystal structure of the liver X receptor β ligand binding domain -: Regulation by a histidine-tryptophan switch Williams, S; Bledsoe, RK; Collins, JL; Boggs, S; Lambert, MH; Miller, AB; Moore, J; McKee, DD; Moore, L; Nichols, J; Parks, D; Watson, M; Wisely, B; Willson, TM 分享 收藏
Identification of a novel human constitutive androstane receptor (CAR) agonist and its use in the identification of CAR target genes Maglich, JM; Parks, DJ; Moore, LB; Collins, JL; Goodwin, B; Billin, AN; Stoltz, CA; Kliewer, SA; Lambert, MH; Willson, TM; Moore, JT 分享 收藏
A new series of estrogen receptor modulators that display selectivity for estrogen receptor β Henke, BR; Consler, TG; Go, N; Hale, RL; Hohman, DR; Jones, SA; Lu, AT; Moore, LB; Moore, JT; Orband-Miller, LA; Robinett, RG; Shearin, J; Spearing, PK; Stewart, EL; Turnbull, PS; Weaver, SL; Williams, SP; Wisely, GB; Lambert, MH 分享 收藏
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Structural determinants of ligand binding selectivity between the peroxisome proliferator-activated receptors Xu, HE; Lambert, MH; Montana, VG; Plunket, KD; Moore, LB; Collins, JB; Oplinger, JA; Kliewer, SA; Gampe, RT; McKee, DD; Moore, JT; Willson, TM 分享 收藏
Design of selective and soluble inhibitors of tumor necrosis factor-α converting enzyme (TACE) Rabinowitz, MH; Andrews, RC; Becherer, JD; Bickett, DM; Bubacz, DG; Conway, JG; Cowan, DJ; Gaul, M; Glennon, K; Lambert, MH; Leesnitzer, MA; McDougald, DL; Moss, ML; Musso, DL; Rizzolio, MC 分享 收藏
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A selective peroxisome proliferator-activated receptor δ agonist promotes reverse cholesterol transport Oliver, WR; Shenk, JL; Snaith, MR; Russell, CS; Plunket, KD; Bodkin, NL; Lewis, MC; Winegar, DA; Sznaidman, ML; Lambert, MH; Xu, HE; Sternbach, DD; Kliewer, SA; Hansen, BC; Willson, TM 分享 收藏
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Pharmacophore analysis of the nuclear oxysterol receptor LXRα Spencer, TA; Li, DS; Russel, JS; Collins, JL; Bledsoe, RK; Consler, TG; Moore, LB; Galardi, CM; McKee, DD; Moore, JT; Watson, MA; Parks, DJ; Lambert, MH; Willson, TM 分享 收藏
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