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Linda H. Malkas

City of Hope Beckman Research Institute

34H指数
215论文数
4.1K被引数
收录论文 54
发表时间
Targeting Cancer-Associated PCNA with AOH1996 Induces Mitotic Catastrophe and Enhances Cisplatin Therapy in Cervical Cancer靶向癌症相关PCNA的AOH1996诱导有丝分裂灾难并增强顺铂疗法在宫颈癌中的应用
err2026-05-01
err0
PREAI
errWendel, Sebastian O.; Brooke, Grant M.; Hu, Changkun; Sandoval, Allison R.; Haratipour, Pouya; Gu, Long; Young, Malaney; Zangi, Maryam; Rasche, Brittany L.; Banerjee, N. s.; Jossart, Jennifer; Garvin, Kelly; Geisbrecht, Brian V.; Cianciolo, Rachel; Cawley, Jacob; Perry, J. Jefferson P.; Hickey, Robert J.; Malkas, Linda H.; Wallace, Nicholas A.
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AOH1996 targets mitochondrial dynamics and metabolism in leukemic stem cells via mitochondrial PCNA inhibition (vol 13, 123, 2024)AOH1996通过抑制线粒体PCNA,靶向作用于白血病干细胞中的线粒体动力学和代谢(vol 13, 123, 2024)
err2025-04-10
err0
errOAAI
errKang, HyunJun; Valerio, Melissa; Feng, Jia; Gu, Long; Hoang, Dinh Hoa; Blackmon, Amanda; Sharkas, Shawn; Pathak, Khyatiben; Jossart, Jennifer; Li, Zhuo; Zhang, Hongyu; Zhang, Bin; Pirrotte, Patrick; Perry, J. Jefferson P.; Hickey, Robert J.; Malkas, Linda; Marcucci, Guido
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Therapeutic Targeting of Oncogene-Induced Transcription-Replication Conflicts in Pancreatic Ductal Adenocarcinoma靶向癌基因诱导的转录-复制冲突在胰导管腺癌中的治疗应用
err2025-04-08
err0
errOAAI
errShanna J. Smith; Fan Meng; Robert G. Lingeman; Caroline M. Li; Min Li; Galyah Boneh; Toni T. Seppälä; Thuy Phan; Haiqing Li; Richard A. Burkhart; Vishwas Parekh; Syed Rahmanuddin; Laleh G. Melstrom; Robert J. Hickey; Vincent Chung; Yilun Liu; Linda H. Malkas; Mustafa Raoof
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AOH1996 targets mitochondrial dynamics and metabolism in leukemic stem cells via mitochondrial PCNA inhibitionAOH1996通过抑制线粒体PCNA靶向白血病干细胞的线粒体动力学和代谢
err2024-12-28
err0
errOAAI
errKang, Hyunjun; Valerio, Melissa; Feng, Jia; Gu, Long; Hoang, Dinh Hoa; Blackmon, Amanda; Sharkas, Shawn; Pathak, Khyatiben; Jossart, Jennifer; Li, Zhuo; Zhang, Hongyu; Zhang, Bin; Pirrotte, Patrick; Perry, J. Jefferson P.; Hickey, Robert J.; Malkas, Linda; Marcucci, Guido; Nguyen, Le Xuan Truong
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Disrupting Mitochondrial Dynamics and Metabolism in Leukemic Stem Cells through Mitochondrial PCNA Inhibition: The Role of AOH1996通过抑制线粒体PCNA破坏白血病干细胞中线粒体动力学和代谢:AOH1996的作用
errBLOOD
IF23.1
err2024-11-05
err0
PREAI
errKang, Hyunjun; Valerio, Melissa; Feng, Jia; Gu, Long; Hoang, Dinh Hoa; Sharkas, Shawn; V. Pathak, Khyatiben; Jossart, Jennifer; Shostak, Yuriy; Li, Zhuo; Zhang, Bin; Pirrotte, Patrick; Perry, Jefferson; Hickey, Robert; Malkas, Linda H.; Marcucci, Guido; Nguyen, Le Xuan Truong
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Identification of biomarkers associated with sensitivity to a novel PCNA inhibitor (AOH1996) by CRISPRi screening
err2024-03-22
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PREAI
errGu, Long; Li, Ming; Chen, Chun-Wei; Hickey, Robert J.; Malkas, Linda H.
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Enhanced lung cancer treatment using AOH1996, a potent PCNA inhibitor
err2024-03-22
err0
PREAI
errLingeman, Robert G.; Hickey, Robert J.; Malkas, Linda H.
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From proteomic analysis to early investigations of combining inhibitors targeting PCNA and histone deacetylase
err2024-03-22
err0
PREAI
errLi, Caroline M.; Garcia-Mansfield, Krystine; Lingeman, Robert G.; Gu, Long; Hickey, Robert J.; Pirrotte, Patrick; Malkas, Linda H.
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Developing a selective cancer chemotherapy by small molecule-based targeting of PCNA protein
err2024-03-22
err0
PREAI
errJossart, Jennifer; Gu, Long; Haratipour, Pouya; Li, Caroline; Lingeman, Robert; Hickey, Robert; Malkas, Linda; Perry, John J.
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Structure-based drug design against caPCNA for selective cancer chemotherapy development
err2024-03-22
err0
PREAI
errJossart, Jennifer; Haratipour, Pouya; Gu, Long; Li, Carone M.; Lingeman, Robert; Liu, Yilun; Hickey, Robert J.; Malkas, Linda H.; Perry, Jeff J.
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Enhancing AOH1996 through structure activity relationship exploration for caPCNA inhibition
err2024-03-22
err0
PREAI
errHaratipour, Pouya; Zangi, Maryam; Yaghoubi, Mahshid; Gu, Long; Jossart, Jennifer; Perry, John J.; Malkas, Linda H.; Hickey, Robert J.
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The potential of PCNA inhibition as a therapeutic strategy in cervical cancer
err2023-11-27
err3
errOAAI
errWendel, Sebastian O.; Snow, Jazmine A.; Gu, Long; Banerjee, Nilam Sanjib; Malkas, Linda; Wallace, Nicholas A.
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Small molecule targeting of transcription-replication conflict for selective chemotherapy选择性化疗的转录-复制冲突小分子靶向研究
err2023-10-01
err19
errOAAI
errGu, Long; Li, Min; Li, Caroline M.; Haratipour, Pouya; Lingeman, Robert; Jossart, Jennifer; Gutova, Margarita; Flores, Linda; Hyde, Caitlyn; Kenjic, Nikola; Li, Haiqing; Chung, Vincent; Li, Hongzhi; Lomenick, Brett; Von Hoff, Daniel D.; Synold, Timothy W.; Aboody, Karen S.; Liu, Yilun; Horne, David; Hickey, Robert J.; Perry, J. Jefferson P.; Malkas, Linda H.
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Arginine shortage induces replication stress and confers genotoxic resistance by inhibiting histone H4 translation and promoting PCNA ubiquitination
err2023-04-01
err0
errOAAI
errWang, Yi-Chang; Kelso, Andrew A.; Karamafrooz, Adak; Chen, Yi-Hsuan; Chen, Wei-Kai; Cheng, Chun-Ting; Qi, Yue; Gu, Long; Malkas, Linda; Taglialatela, Angelo; Kung, Hsing-Jien; Moldovan, George-Lucian; Ciccia, Alberto; Stark, Jeremy M.; Ann, David K.
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Novel Peptide Therapeutic Approaches for Cancer Treatment
errCELLS
IF5.2
err2021-10-27
err83
errOAAI
errLi, Caroline M.; Haratipour, Pouya; Lingeman, Robert G.; Perry, J. Jefferson P.; Gu, Long; Hickey, Robert J.; Malkas, Linda H.
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A Quantitative Analysis of Surgical Smoke Exposure as an Occupational Hazard
err2021-04-30
err11
PREAI
errStewart, Camille L.; Raoof, Mustafa; Lingeman, Robert; Malkas, Linda; Flores, Viviana; Caldwell, Kerry; Fong, Yuman; Melstrom, Kurt
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Molecular Targeting of Cancer-Associated PCNA Interactions in Pancreatic Ductal Adenocarcinoma Using a Cell-Penetrating Peptide
err2020-06-01
err20
errOAAI
errSmith, Shanna J.; Li, Caroline M.; Lingeman, Robert G.; Hickey, Robert J.; Liu, Yilun; Malkas, Linda H.; Raoof, Mustafa
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Mechanistic study of the superior anti-cancer properties of a first in-class small molecule targeting PCNA
err2019-12-01
err1
PREAI
errGu, Long; Li, Min; Lingeman, Robert; Hickey, Robert J.; Liu, Yilun; Malkas, Linda H.
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