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Philip J. Merta

University of Washington

19H指数
51论文数
1.2K被引数
收录论文 15
发表时间
Tricyclic Covalent Inhibitors Selectively Target Jak3 through an Active Site Thiol
err2015-02-01
err99
errOAAI
errGoedken, Eric R.; Argiriadi, Maria A.; Banach, David L.; Fiamengo, Bryan A.; Foley, Sage E.; Frank, Kristine E.; George, Jonathan S.; Harris, Christopher M.; Hobson, Adrian D.; Ihle, David C.; Marcotte, Douglas; Merta, Philip J.; Michalak, Mark E.; Murdock, Sara E.; Tomlinson, Medha J.; Voss, Jeffrey W.
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Pyrimidine-Based Tricyclic Molecules as Potent and Orally Efficacious Inhibitors of Wee1 Kinase基于嘧啶的三环分子作为Wee1激酶的有效和口服有效抑制剂
err2014-08-06
err29
errOAAI
errTong, Yunsong; Torrent, Maricel; Florjancic, Alan S.; Bromberg, Kenneth D.; Buchanan, Fritz G.; Ferguson, Debra C.; Johnson, Eric F.; Lasko, Loren M.; Maag, David; Merta, Philip J.; Olson, Amanda M.; Osterling, Donald J.; Soni, Nirupama; Shoemaker, Alexander R.; Penning, Thomas D.
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Potent and Selective Inhibitors of CDPK1 from T. gondii and C. parvum Based on a 5-Aminopyrazole-4-carboxamide Scaffold
err2013-11-20
err55
errOAAI
errZhang, Zhongsheng; Ojo, Kayode K.; Vidadala, RamaSubbaRao; Huang, Wenlin; Geiger, Jennifer A.; Scheele, Suzanne; Choi, Ryan; Reid, Molly C.; Keyloun, Katelyn R.; Rivas, Kasey; Siddaramaiah, Latha Kallur; Comess, Kenneth M.; Robinson, Kenneth P.; Merta, Philip J.; Kifle, Lemma; Hol, Wim G. J.; Parsons, Marilyn; Merritt, Ethan A.; Maly, Dustin J.; Verlinde, Christophe L. M. J.; Van Voorhis, Wesley C.; Fan, Erkang
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Azaindole-Based Inhibitors of Cdc7 Kinase: Impact of the Pre-DFG Residue, Val 195基于氮杂吲哚的Cdc7激酶抑制剂: 前DFG残基Val 195的影响
err2013-01-18
err29
errOAAI
errTong, Yunsong; Stewart, Kent D.; Florjancic, Alan S.; Harlan, John E.; Merta, Philip J.; Przytulinska, Magdalena; Soni, Nirupama; Swinger, Kerren K.; Zhu, Haizhong; Johnson, Eric F.; Shoemaker, Alexander R.; Penning, Thomas D.
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Therapeutic Implications for the Induced Levels of Chk1 in Myc-Expressing Cancer Cells
err2011-11-14
err120
errOAAI
errHoeglund, Andreas; Nilsson, Lisa M.; Muralidharan, Somsundar Veppil; Hasvold, Lisa A.; Merta, Philip; Rudelius, Martina; Nikolova, Viktoriya; Keller, Ulrich; Nilsson, Jonas A.
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JAK2V617F drives Mcl-1 expression and sensitizes acute myeloid leukemia cells to dual inhibition of JAK2 and Bcl-XL
err2011-04-01
err0
PREAI
errGuo, Jun; Roberts, Lisa; Kraft, Jeffrey B.; Merta, Philip J.; Glaser, Keith B.; Shah, Omar J.
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Navigating the kinome
err2011-02-20
err240
PREAI
errMetz, James T.; Johnson, Eric F.; Soni, Niru B.; Merta, Philip J.; Kifle, Lemma; Hajduk, Philip J.
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A Unified, Probabilistic Framework for Structure- and Ligand-Based Virtual Screening
err2011-02-10
err71
PREAI
errSwann, Steven L.; Brown, Scott P.; Muchmore, Steven W.; Patel, Hetal; Merta, Philip; Locklear, John; Hajduk, Philip J.
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Design, synthesis, and biological activity of 5,10-dihydro-dibenzo[b,e][1,4]diazepin-11-one-based potent and selective Chk-1 inhibitors
err2007-07-21
err49
PREAI
errWang, Le; Sullivan, Gerard M.; Hexamer, Laura A.; Hasvold, Lisa A.; Thalji, Reema; Przytulinska, Magdalena; Tao, Zhi-Fu; Li, Gaoquan; Chen, Zehan; Xiao, Zhan; Gu, Wen-Zhen; Xue, John; Bui, Mai-Ha; Merta, Philip; Kovar, Peter; Bouska, Jennifer J.; Zhang, Haiying; Park, Chang; Stewart, Kent D.; Sham, Hing L.; Sowin, Thomas J.; Rosenberg, Saul H.; Lin, Nan-Horng
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From bacterial genomes to novel antibacterial agents:: discovery, characterization, and antibacterial activitv of compounds that bind to HI0065 (YjeE) from Haemophilus influenzae
err2007-06-06
err20
PREAI
errLerner, Claude G.; Hajduk, Philip J.; Wagner, Rolf; Wagenaar, Frank L.; Woodall, Charlotte; Gu, Yu-Gui; Searle, Xenia B.; Florjancic, Alan S.; Zhang, Tianyuan; Clark, Richard F.; Cooper, Curt S.; Mack, Jamey C.; Yu, Liping; Cai, Mengli; Betz, Steven F.; Chovan, Linda E.; McCall, J. Owen; Black-Schaefer, Candace L.; Kakavas, Stephan J.; Schurdak, Mark E.; Comess, Kenneth M.; Walter, Karl A.; Edalji, Rohinton; Dorwin, Sarah A.; Smith, Richard A.; Hebert, Eric J.; Harlan, John E.; Metzger, Randy E.; Marta, Philip J.; Baranowski, John L.; Coen, Michael L.; Thornewell, Susan J.; Shivakumar, Annapur G.; Saiki, Anne Y.; Soni, Niru; Bui, Mai; Balli, Darlene J.; Sanders, William J.; Nilius, Angela M.; Holzman, Thomas F.; Fesik, Stephen W.; Beutel, Bruce A.
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Structure-based design, synthesis, and biological evaluation of potent and selective macrocyclic checkpoint kinase 1 inhibitors
err2007-03-13
err88
PREAI
errTao, Zhi-Fu; Wang, Le; Stewart, Kent D.; Chen, Zehan; Gu, Wendy; Bui, Mai-Ha; Merta, Philip; Zhang, Haiying; Kovar, Peter; Johnson, Eric; Park, Chang; Judge, Russell; Rosenberg, Saul; Sowin, Thomas; Lin, Nan-Horng
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Novel antibacterial class: A series of tetracyclic derivatives
err2006-07-11
err18
PREAI
errHinman, Mira M.; Rosenberg, Teresa A.; Balli, Darlene; Black-Schaefer, Candace; Chovan, Linda E.; Kalvin, Douglas; Merta, Philip J.; Nilius, Angela M.; Pratt, Steve D.; Soni, Niru B.; Wagenaar, Frank L.; Weitzberg, Moshe; Wagner, Rolf; Beutel, Bruce A.
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Novel antibacterial class
err2003-12-01
err30
errOAAI
errDandliker, PJ; Pratt, SD; Nilius, AM; Black-Schaefer, C; Ruan, X; Towne, DL; Clark, RF; Englund, EE; Wagner, R; Weitzberg, M; Chovan, LE; Hickman, RK; Daly, MM; Kakavas, S; Zhong, P; Cao, ZS; David, CA; Xuei, XL; Lerner, CG; Soni, NB; Bui, M; Shen, LL; Cai, YN; Merta, PJ; Saiki, AYC; Beutel, BA
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