未登录 Novel 2,3-dihydro-1,4-benzoxazines as potent and orally bioavailable inhibitors of tumor-driven angiogenesis La, Daniel S.; Belzile, Julie; Bready, James V.; Coxon, Angela; DeMelfi, Thomas; Doerr, Nicholas; Estrada, Juan; Flynn, Julie C.; Flynn, Shaun R.; Graceffa, Russell F.; Harriman, Shawn P.; Larrow, Jay F.; Long, Alexander. M.; Martin, Matthew W.; Morrison, Michael J.; Patel, Vinod F.; Roveto, Philip M.; Wang, Ling; Weiss, Matthew M.; Whittington, Douglas A.; Teffera, Yohannes; Zhao, Zhiyang; Polverino, Anthony J.; Harmanget, Jean-Christophe 分享 收藏
Design, synthesis, and evaluation of orally active benzimidazoles and benzoxazoles as vascular endothelial growth factor-2 receptor tyrosine kinase inhibitors (vol 50, pg 4351, 2007) Potashman, Michele H.; Bready, James; Coxon, Angela; DeMelfi, Thomas M., Jr.; DiPietro, Lucian; Doerr, Nicholas; Elbaum, Paniel; Estrada, Juan; Gallant, Paul; Germain, Julie; Gu, Yan; Harmange, Jean-Christophe; Kaufman, Stephen A.; Kendall, Rick; Kim, Joseph L.; Kumar, Gondi N.; Long, Alexander M.; Neervannan, Seshadri; Patel, Vinod F.; Polverino, Anthony; Rose, Paul; van der Plas, Simon; Whittington, Douglas; Zanon, Roger; Zhao, Huilin 分享 收藏
Design, synthesis, and evaluation of orally active Benzimidazoles and Benzoxazoles as vascular endothelial growth factor-2 receptor tyrosine kinase inhibitors Potashman, Michele H.; Bready, James; Coxon, Angela; DeMelfi, Thomas M., Jr.; DiPietro, Lucian; Doerr, Nicholas; Elbaum, Daniel; Estrada, Juan; Gallan, Paul; Germain, Julie; Gu, Yan; Harmange, Jean-Christophe; Kaufman, Stephen A.; Kendall, Rick; Kim, Joseph L.; Kumar, Gondi N.; Long, Alexander M.; Neervannan, Seshadri; Patel, Vinod F.; Polverino, Anthony; Rose, Paul; van der Plas, Simon; Whittington, Douglas; Zanon, Roger; Zhao, Huilin 分享 收藏
AMG 706, an oral, multikinase inhibitor that selectively targets vascular endothelial growth factor, platelet-derived growth factor, and Kit receptors, potently inhibits angiogenesis and induces regression in tumor xenografts Polverino, Anthony; Coxon, Angela; Starnes, Charlie; Diaz, Zobedia; DeMelfi, Thomas; Wang, Ling; Bready, James; Estrada, Juan; Cattley, Russell; Kaufman, Stephen; Chen, Danlin; Gan, Yongmei; Kumar, Gondi; Meyer, James; Neervannan, Sesha; Alva, Gonzalo; Talvenheimo, Jane; Montestruque, Silvia; Tasker, Andrew; Patel, Vinod; Radinsky, Robert; Kendall, Richard 分享 收藏
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