未登录 Identification of small molecule estrogen-related receptor α-specific antagonists and homology modeling to predict the molecular determinants as the basis for selectivity over ERRβ and ERRγ 鉴定小分子雌激素相关受体 α 特异性拮抗剂和同源建模以预测分子决定因素作为对err β 和err γ 选择性的基础 Chisamore, Michael J.; Mosley, Ralph T.; Cai, Sheng-Jian; Birzin, Elizabeth T.; O'Donnell, Gregory; Zuck, Paul; Flores, Osvaldo; Schaeffer, James; Rohrer, Susan P.; Chen, J. Don; Wilkinson, Hilary A. 分享 收藏
Antidiabetic activity of a highly potent and selective nonpeptide somatostatin receptor subtype-2 agonist Strowski, Mathias Z.; Cashen, Doreen E.; Birzin, Elizabeth T.; Yang, Lihu; Singh, Vandana; Jacks, Thomas M.; Nowak, Krzysztof W.; Rohrer, Susan P.; Patchett, Arthur A.; Smith, Roy G.; Schaeffer, James M. 分享 收藏
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Estrogen receptor ligands.: II.: Discovery of benzoxathiins as potent, selective estrogen receptor α modulators Kim, S; Wu, JY; Birzin, ET; Frisch, K; Chan, W; Pai, LY; Yang, YT; Mosley, RT; Fitzgerald, PMD; Sharma, N; Dahllund, J; Thorsell, AG; DiNinno, F; Rohrer, SP; Schaeffer, JM; Hammond, ML 分享 收藏
Immunolocalization of estrogen receptor β in the mouse brain:: Comparison with estrogen receptor α Mitra, SW; Hoskin, E; Yudkovitz, J; Pear, L; Wilkinson, HA; Hayashi, S; Pfaff, DW; Ogawa, S; Rohrer, SP; Schaeffer, JM; McEwen, BS; Alves, SE 分享 收藏
Effects of Heterocyclic aromatic substituents on binding affinities at two distinct sites of somatostatin receptors. Correlation with the electrostatic potential of the substituents Prasad, V; Birzin, ET; McVaugh, CT; van Rijn, RD; Rohrer, SP; Chicchi, G; Underwood, DJ; Thornton, ER; Smith, AB; Hirschmann, R 分享 收藏
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A potent, nonpeptidyl 1H-quinolone antagonist for the gonadotropin-releasing hormone receptor DeVita, RJ; Walsh, TF; Young, JR; Jiang, JL; Ujjainwalla, F; Toupence, RB; Parikh, M; Huang, SX; Fair, JA; Goulet, MT; Wyvratt, MJ; Lo, JL; Ren, N; Yudkovitz, JB; Yang, YT; Cheng, K; Cui, JS; Mount, G; Rohrer, SP; Schaeffer, JM; Rhodes, L; Drisko, JE; McGowan, E; MacIntyre, DE; Vincent, S; Carlin, JR; Cameron, J; Smith, RG 分享 收藏
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Synthesis and biological activities of potent peptidomimetics selective for somatostatin receptor subtype 2 Yang, LH; Berk, SC; Rohrer, SP; Mosley, RT; Guo, LQ; Underwood, DJ; Arison, BH; Birzin, ET; Hayes, EC; Mitra, SW; Parmar, RM; Cheng, K; Wu, TJ; Butler, BS; Foor, F; Pasternak, A; Pan, YP; Silva, M; Freidinger, RM; Smith, RG; Chapman, K; Schaeffer, JM; Patchett, AA 分享 收藏
Spiro[1H-indene-1,4′-piperidine] derivatives as potent and selective non-peptide human somatostatin receptor subtype 2 (sst2) agonists Yang, LH; Guo, LQ; Pasternak, A; Mosley, R; Rohrer, S; Birzin, E; Foor, F; Cheng, K; Schaeffer, J; Patchett, AA 分享 收藏
Modulation of receptor and receptor subtype affinities using diastereomeric and enantiomeric monosaccharide scaffolds as a means to structural and biological diversity. A new route to ether synthesis Hirschmann, R; Hynes, J; Cichy-Knight, MA; van Rijn, RD; Sprengeler, PA; Spoors, PG; Shakespeare, WC; Pietranico-Cole, S; Barbosa, J; Liu, J; Yao, WQ; Rohrer, S; Smith, AB 分享 收藏
Ophiobolin M and analogues, noncompetitive inhibitors of ivermectin binding with nematocidal activity Tsipouras, A; Adefarati, AA; Tkacz, JS; Frazier, EG; Rohrer, SP; Birzin, E; Rosegay, A; Zink, DL; Goetz, MA; Singh, SB; Schaeffer, JM 分享 收藏