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收藏Identification of Potent Leucine-Rich Repeat Kinase 2 Inhibitors by Virtual Screening and Biological Evaluation
Shen, Hualiang; Yu, Guoqi; Cai, Tao; Hu, Kai; Shang, Tianbo; Luo, Yanjuan; Zhu, Jiawei; Bai, Xiaoxue; Xiong, Yicheng; Xi, Meiyang; Shen, Runpu
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收藏Antibody-drug conjugates for targeted cancer therapy: Recent advances in potential payloads用于靶向癌症治疗的抗体-药物结合物: 潜在有效载荷的最新进展
Xi, Meiyang; Zhu, Jingjing; Zhang, Fengxia; Shen, Hualiang; Chen, Jianhui; Xiao, Ziyan; Huangfu, Yanping; Wu, Chunlei; Sun, Haopeng; Xia, Gang
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收藏Hyaluronic Acid Poly(glyceryl)10-Stearate Derivatives: Novel Emulsifiers for Improving the Gastrointestinal Stability and Bioaccessibility of Coenzyme Q10 Nanoemulsions
Luo, Xiang; Ao, Sha; Wu, Hongze; McClements, David Julian; Fang, Likun; Huang, Mengyu; Zhou, Yanyan; Yin, Xuguang; Xi, Meiyang; Cai, Tao; Zhu, Kewu
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收藏Therapeutic potential of targeting kynurenine pathway in neurodegenerative diseases靶向犬尿氨酸途径在神经退行性疾病中的治疗潜力
Shen, Hualiang; Xu, Xinde; Bai, Yalong; Wang, Xiaoping; Wu, Yibin; Zhong, Jia; Wu, Qiyi; Luo, Yanjuan; Shang, Tianbo; Shen, Runpu; Xi, Meiyang; Sun, Haopeng
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收藏Small molecule PROTACs in targeted therapy: An emerging strategy to induce protein degradation
Xi, Meiyang; Chen, Yi; Yang, Hongyu; Xu, Huiting; Du, Kui; Wu, Chunlei; Xu, Yanfei; Deng, Liping; Luo, Xiang; Yu, Lemao; Wu, Yonghua; Gao, Xiaozhong; Cai, Tao; Chen, Bin; Shen, Runpu; Sun, Haopeng
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收藏Discovery and Modification of in Vivo Active Nrf2 Activators with 1,2,4-Oxadiazole Core: Hits Identification and Structure-Activity Relationship Study
Xu, Li-Li; Zhu, Jun-Feng; Xu, Xiao-Li; Zhu, Jie; Li, Li; Xi, Mei-Yang; Jiang, Zhen-Yu; Zhang, Ming-Ye; Liu, Fang; Lu, Meng-chen; Bao, Qi-Chao; Li, Qi; Zhao, Chao; Wei, Jin-Lian; Zhang, Xiao-Jin; Zhang, Lian-Shan; You, Qi-Dong; Sun, Hao-Peng
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收藏Discovery of Potent Keap1-Nrf2 Protein-Protein Interaction Inhibitor Based on Molecular Binding Determinants Analysis
Jiang, Zheng-Yu; Lu, Meng-Chen; Xu, Li-Li; Yang, Ting-Ting; Xi, Mei-Yang; Xu, Xiao-Li; Guo, Xiao-Ke; Zhang, Xiao-Jin; You, Qi-Dong; Sun, Hao-Peng
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收藏Discovery of Potent Keap1-Nrf2 Protein-Protein Interaction Inhibitor Based on Molecular Binding Determinants Analysis
Jiang, Zheng-Yu; Lu, Meng-Chen; Xu, Li-Li; Yang, Ting-Ting; Xi, Mei-Yang; Xu, Xiao-Li; Guo, Xiao-Ke; Zhang, Xiao-Jin; You, Qi-Dong; Sun, Hao-Peng
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收藏3-Aroylmethylene-2,3,6,7-tetrahydro-1H-pyrazino[2,1-a]isoquinolin-4(11bH)-ones as Potent Nrf2/ARE Inducers in Human Cancer Cells and AOM-DSS Treated Mice
Xi, Mei-yang; Jia, Jian-min; Sun, Hao-peng; Sun, Zhong-ying; Jiang, Jie-wei; Wang, Ya-jing; Zhang, Min-ye; Zhu, Jun-feng; Xu, Li-li; Jiang, Zheng-yu; Xue, Xin; Ye, Ming; Yang, Xi; Gao, Yuan; Tao, Lei; Guo, Xiao-ke; Xu, Xiao-li; Guo, Qing-long; Zhang, Xiao-jin; Hu, Rong; You, Qi-dong
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收藏Effective Screening Strategy Using Ensembled Pharmacophore Models Combined with Cascade Docking: Application to p53-MDM2 Interaction Inhibitors
Xue, Xin; Wei, Jin-Lian; Xu, Li-Li; Xi, Mei-Yang; Xu, Xiao-Li; Liu, Fang; Guo, Xiao-Ke; Wang, Lei; Zhang, Xiao-Jin; Zhang, Ming-Ye; Lu, Meng-Chen; Sun, Hao-Peng; You, Qi-Dong
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收藏Synthesis and bioevaluation of a series of α-pyrone derivatives as potent activators of Nrf2/ARE pathway (part I)作为Nrf2/ARE途径有效激活剂的一系列 α-吡喃酮衍生物的合成和生物评价 (第一部分)
Xi, Mei-yang; Sun, Zhong-ying; Sun, Hao-peng; Jia, Jian-min; Jiang, Zheng-yu; Tao, Lei; Ye, Ming; Yang, Xi; Wang, Ya-jing; Xue, Xin; Huang, Jing-jie; Gao, Yuan; Guo, Xiao-ke; Zhang, Sheng-lie; Yang, Ying-rui; Guo, Qing-long; Hu, Rong; You, Qi-dong
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收藏Studies on chemical modification and biology of a natural product, gambogic acid (III): Determination of the essential pharmacophore for biological activity
Wang, Xiaojian; Lu, Na; Yang, Qian; Gong, Dandan; Lin, Changjun; Zhang, Shenglie; Xi, Meiyang; Gao, Yuan; Wei, Libing; Guo, Qinglong; You, Qidong
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