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Different in vitro and in vivo profiles of substituted 3-aminopropylphosphinate and 3-aminopropyl(methyl)phosphinate GABAB receptor agonists as inhibitors of transient lower oesophageal sphincter relaxation Lehmann, A.; Antonsson, M.; Aurell-Holmberg, A.; Blackshaw, L. A.; Branden, L.; Elebring, T.; Jensen, J.; Karrberg, L.; Mattsson, J. P.; Nilsson, K.; Oja, S. S.; Saransaari, P.; von Unge, S. 分享 收藏
(R)-(3-Amino-2-fluoropropyl) Phosphinic Acid (AZD3355), a Novel GABAB Receptor Agonist, Inhibits Transient Lower Esophageal Sphincter Relaxation through a Peripheral Mode of Action Lehmann, Anders; Antonsson, Madeleine; Holmberg, Ann Aurell; Blackshaw, L. Ashley; Branden, Lena; Braeuner-Osborne, Hans; Christiansen, Bolette; Dent, John; Elebring, Thomas; Jacobson, Britt-Marie; Jensen, Jorgen; Mattsson, Jan P.; Nilsson, Karolina; Oja, Simo S.; Page, Amanda J.; Saransaari, Pirjo; von Unge, Sverker 分享 收藏
Making medicinal chemistry more effective-application of Lean Sigma to improve processes, speed and quality Andersson, Shalini; Armstrong, Alan; Bjore, Annika; Bowker, Sue; Chapman, Steve; Davies, Rob; Donald, Craig; Egner, Bryan; Elebring, Thomas; Holmqvist, Sara; Inghardt, Tord; Johannesson, Petra; Johansson, Magnus; Johnstone, Craig; Kemmitt, Paul; Kihlberg, Jan; Korsgren, Pernilla; Lemurell, Malin; Moore, Jane; Pettersson, Jonas A.; Pointon, Helen; Ponten, Fritiof; Schofield, Paul; Selmi, Nidhal; Whittamore, Paul 分享 收藏
The orphan receptor GPR55 is a novel cannabinoid receptor 孤儿受体GPR55是一种新型大麻素受体 Ryberg, E.; Larsson, N.; Sjoegren, S.; Hjorth, S.; Hermansson, N-O; Leonova, J.; Elebring, T.; Nilsson, K.; Drmota, T.; Geasley, P. J. 分享 收藏
Effects of (2R)-(3-amino-2-fluoropropyl)sulphinic acid (AFPSiA) on transient lower oesophageal sphincter relaxation in dogs and mechanism of hypothermic effects in mice Lehmann, A; Holmberg, AA; Bhatt, U; Bremner-Danielsen, M; Brändén, L; Elg, S; Elebring, T; Fitzpatrick, K; Geiss, WB; Guzzo, P; Jensen, J; Jerndal, G; Mattsson, JP; Nilsson, K; Olsson, BM 分享 收藏
Synthesis and pharmacological evaluation of novel γ-aminobutyric acid type B (GABAB) receptor agonists as gastroesophageal reflux inhibitors Alstermark, Christer; Amin, Kosrat; Dinn, Sean R.; Elebring, Thomas; Fjellstroem, Ola; Fitzpatrick, Kevin; Geiss, William B.; Gottfries, Johan; Guzzo, Peter R.; Harding, James P.; Holmen, Anders; Kothare, Mohit; Lehmann, Anders; Mattsson, P.; Nilsson, Karolina; Sunden, Gunnel; Swanson, Marianne; von Unge, Sverker; Woo, Alex M.; Wyle, Michael J.; Zheng, Xiaozhang 分享 收藏
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Novel structures derived from 2-[[(2-Pyridyl)methyl]thio]-1H-benzimidazole as anti-Helicobacter pylori agents, part 1 Kühler, TC; Swanson, M; Christenson, B; Klintenberg, AC; Lamm, B; Fägerhag, J; Gatti, R; Ölwegård-Halvarsson, M; Shcherbuchin, V; Elebring, T; Sjöström, JE 分享 收藏
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6-HYDROXY-3-N-PROPYL-2,3,4,5-TETRAHYDRO-1H-3-BENZAZEPINE AND ANALOGS - NEW CENTRALLY ACTING 5-HT1A RECEPTOR AGONISTS WIKSTROM, H; ANDERSSON, B; ELEBRING, T; LAGERKVIST, S; HALLNEMO, G; PETTERSSON, I; JOVALL, PA; SVENSSON, K; EKMAN, A; CARLSSON, A 分享 收藏
6,7,8,9-TETRAHYDRO-N,N-DI-N-PROPYL-3H-BENZINDOL-8-AMINES - DERIVATIVES AS POTENT AND ORALLY-ACTIVE SEROTONIN 5-HT1A RECEPTOR AGONISTS STJERNLOF, P; ELEBRING, T; NILSSON, J; ANDERSSON, B; LAGERKVIST, S; SVENSSON, K; EKMAN, A; CARLSSON, A; WIKSTROM, H 分享 收藏