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Hans Bräuner‐Osborne

university of copenhagen

56H指数
280论文数
1.2W被引数
收录论文 163
发表时间
Ultra-large virtual screening unveils potent agonists of the neuromodulatory orphan receptor GPR139超大规模虚拟筛选揭示了神经调节孤核受体GPR139的强效激动剂
err2025-12-09
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errIsrael Cabeza de Vaca; Boris Trapkov; Ling Shen; Duy Duc Vo; Xiaoqun Zhang; Yunting Yang; Mitra Pezeshki; Xuehan Zhang; Frida Bällgren; Aljona Saleh; Andrii V. Tarnovskiy; Dmytro S. Radchenko; Yurii S. Moroz; Hans Bräuner-Osborne; Per Svenningsson; Jan Kihlberg; Zhi-Jie Liu; Alexander Sebastian Hauser; Jens Carlsson
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The Concise Guide to PHARMACOLOGY 2025/26: G protein-coupled receptors《简明药理学指南2025/26:G蛋白偶联受体》
err2025-12-01
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errAlexander, Stephen P. H.; Davenport, Anthony P.; Kelly, Eamonn; Gibb, Alasdair J.; Mathie, Alistair A.; Peach, Chloe J.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Southan, Christopher; Davies, Jamie A.; Abbracchio, Maria Pia; Abraham, George R.; Agoulnik, Alexander; Alexander, Wayne; Al-hosaini, Khaled; Back, Magnus; Baker, Jillian G.; Barnes, Nicholas M.; Bathgate, Ross; Beaulieu, Jean-Martin; Beck-Sickinger, Annette G.; Behrens, Maik; Bennett, Kirstie A.; Bernstein, Kenneth E.; Bettler, Bernhard; Birdsall, Nigel J. M.; Blaho, Victoria A.; Bonaventure, Pascal; Boulay, Francois; Bousquet, Corinne; Brauner-Osborne, Hans; Brown, Andrew J.; Burnstock, Geoffrey; Busnelli, Marta; Calo, Girolamo; Caruso, Vanni; Castano, Justo P.; Catt, Kevin J.; Ceruti, Stefania; Chazot, Paul; Chiang, Nan; Chini, Bice; Christopoulos, Arthur; Chun, Jerold; Cianciulli, Antonia; Civelli, Olivier; Clapp, Lucie H.; Couture, Rejean; Cox, Helen M.; Csaba, Zsolt; Dahlgren, Claes; Dautzenberg, Frank M.; Dent, Gordon; Douglas, Steven D.; Dournaud, Pascal; Dubocovich, Margarita L.; Eguchi, Satoru; Escher, Emanuel; Filardo, Edward J.; Fong, Tung; Forsman, Huamei Fu; Fumagalli, Marta; Gainetdinov, Raul R.; Garelja, Michael L.; de Gasparo, Marc; Gbahou, Florence; Gerard, Craig; Gershengorn, Marvin; Glass, Michelle; Gloriam, David E.; Gobeil, Fernand; Goodfriend, Theodore L.; Goudet, Cyril; Gratz, Lukas; Gregory, Karen J.; Gruber, Christian; Gundlach, Andrew L.; Hamann, Jorg; Hanson, Julien; Hartman, Deborah S.; Hauger, Richard L.; Hay, Debbie L.; Heinemann, Akos; Heitman, Laura; Herr, Deron R.; Hollenberg, Morley D.; Holliday, Nicholas D.; Holst, Birgitte; Horiuchi, Mastgugu; Hoyer, Daniel; Hunyady, Laszlo; Husain, Ahsan; IJzerman, Adriaan P.; Inagami, Tadashi; Insel, Paul A.; Jacobson, Kenneth A.; Jacobson, Laura H.; Jensen, Robert T.; Jockers, Ralf; Jonnalagadda, Deepa; Karnik, Sadashiva; Kaupmann, Klemens; Kemp, Jacqueline; Kennedy, Charles; Kihara, Yasuyuki; Kinsolving, Julia; Kitazawa, Takio; Kozielewicz, Pawel; Kreienkamp, Hans-Juergen; Kukkonen, Jyrki P.; Laishram, Luxmichan; Langenhan, Tobias; Langmead, Christopher J.; Larhammar, Dan; Leach, Katie; Lecca, Davide; Lee, John D.; Leeman, Susan E.; Leprince, Jerome; Leurs, Rob; Li, Xaria X.; Liebscher, Ines; Lolait, Stephen J.; Lupp, Amelie; Macrae, Robyn; Maguire, Janet J.; Malfacini, Davide; Manning, Maurice; Marangon, Davide; Martemyanov, Kirill; Mazella, Jean; McArdle, Craig A.; Melmed, Shlomo; Michel, Martin C.; Miller, Laurence J.; Mitolo, Vincenzo; Mouillac, Bernard; Mueller, Christa E.; Murphy, Philip M.; Nahon, Jean-Louis; Neubig, Richard R.; Ngo, Tony; Norel, Xavier; Nyimanu, Duuamene; O'Carroll, Anne-Marie; Offermanns, Stefan; Panaro, Maria Antonietta; Parmentier, Marc; Perry-Hauser, Nicole; Pertwee, Roger G.; Pin, Jean-Philippe; Prossnitz, Eric R.; Qin, Helena Chengxue; Quinn, Mark; Raffaele, Stefano; Ramachandran, Rithwik; Ray, Manisha; Reinscheid, Rainer K.; Buzon, Alejandro Romeral; Rondard, Philippe; Rosenkilde, Mette M.; Rovati, G. Enrico; Ruzza, Chiara; Sanger, Gareth J.; Scholz, Nicole; Schoeneberg, Torsten; Schulte, Gunnar; Schulz, Stefan; Segaloff, Deborah L.; Serhan, Charles N.; Shukla, Arun K.; Singh, Khuraijam Dhanachandra; Smith, Craig M.; Smith, Nicola J.; Staeubert, Claudia; Stoddart, Leigh A.; Sugimoto, Yukihiko; Summers, Roger; Tan, Valerie P.; Thal, David M.; Thomas, Walter (Wally); Timmermans, Pieter B. M. W. M.; Tirupula, Kalyan; Toll, Lawrence; Tulipano, Giovanni; Unal, Hamiyet; Unger, Thomas; Valant, Celine; Vanderheyden, Patrick; Vaudry, David; Vaudry, Hubert; Verbalis, Joseph G.; Vilardaga, Jean-Pierre; Walker, Christopher S.; Wang, Ji Ming; Ward, Donald T.; Wester, Hans-Juergen; Willars, Gary B.; Williams, Tom Lloyd; Woodruff, Trent M.; Wu, Huixian; Yang, Cheng; Yao, Chengcan; Ye, Richard D.; Zaidman, Nathan
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Arrestin-independent internalization of the GLP-1 receptor is facilitated by a GRK, clathrin, and caveolae-dependent mechanism
err2025-01-05
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errVon Moo, Ee; Moller, Thor Christian; Sorensen, Frederikke Astrid; Inoue, Asuka; Brauner-Osborne, Hans
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Detailed functional characterization of four nanobodies as positive allosteric modulators of the human calcium-sensing receptor
err2025-01-01
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errDu, Wei; Rahman, Sabrina N.; Barker, Eleanor; Brauner-Osborne, Hans; Mathiesen, Jesper M.; Ward, Donald T.; Jensen, Anders A.
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Heterogeneous Origins of Calcium Homeostasis Disorders Arising From 5 Heterozygous Calcium-Sensing Receptor Variants
err2024-10-16
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errDu, Wei; Boisen, Ida Marie; Rahman, Sabrina N.; Poulsen, Nadia Nicholine; Mathiesen, Jesper M.; Jensen, Martin Blomberg; Brauner-Osborne, Hans; Jensen, Anders A.
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Fish-hunting cone snail disrupts prey's glucose homeostasis with weaponized mimetics of somatostatin and insulin
err2024-08-20
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errYeung, Ho Yan; Ramiro, Iris Bea L.; Andersen, Daniel B.; Koch, Thomas Lund; Hamilton, Alexander; Bjorn-Yoshimoto, Walden E.; Espino, Samuel; Vakhrushev, Sergey Y.; Pedersen, Kasper B.; de Haan, Noortje; Ederveen, Agnes L. Hipgrave; Olivera, Baldomero M.; Knudsen, Jakob G.; Brauner-Osborne, Hans; Schjoldager, Katrine T.; Holst, Jens Juul; Safavi-Hemami, Helena
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Loss-of-function Thr347Ala Variant in the G Protein Subunit-Α11 Causes Familial Hypocalciuric Hypercalcemia 2
err2024-06-26
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errBoisen, Ida Marie; Du, Wei; Juul, Anders; Brauner-Osborne, Hans; Jensen, Anders A.; Jensen, Martin Blomberg
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Differential G protein activation by the long and short isoforms of the dopamine D2 receptor多巴胺D2受体的长短同工型的差异g蛋白激活
err2024-05-09
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errReiner-Link, David; Madsen, Jakob Sture; Gloriam, David E.; Brauner-Osborne, Hans; Hauser, Alexander S.
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Structure-Activity Relationship Studies and Optimization of 4-Hydroxypyridones as GPR84 Agonists4-羟基吡啶酮作为GPR84激动剂的构效关系研究和优化
err2024-02-21
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PREAI
errIeremias, Loukas; Kaspersen, Mads H.; Manandhar, Asmita; Schultz-Knudsen, Katrine; Vrettou, Christina Ioanna; Pokhrel, Rina; Heidtmann, Christoffer V.; Jenkins, Laura; Kanellou, Christina; Marsango, Sara; Li, Yueming; Brauner-Osborne, Hans; Ulven, Elisabeth Rexen; Milligan, Graeme; Ulven, Trond
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The Concise Guide to PHARMACOLOGY 2023/24: G protein-coupled receptors药理学2023/24简明指南: g蛋白偶联受体
err2023-12-20
err149
errOAAI
errAlexander, Stephen P. H.; Christopoulos, Arthur; Davenport, Anthony P.; Kelly, Eamonn; Mathie, Alistair A.; Peters, John A.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Davies, Jamie A.; Abbracchio, Maria Pia; Abraham, George; Agoulnik, Alexander; Alexander, Wayne; Al-hosaini, Khaled; Back, Magnus; Baker, Jillian G.; Barnes, Nicholas M.; Bathgate, Ross; Beaulieu, Jean-Martin; Beck-Sickinger, Annette G.; Behrens, Maik; Bernstein, Kenneth E.; Bettler, Bernhard; Birdsall, Nigel J. M.; Blaho, Victoria; Boulay, Francois; Bousquet, Corinne; Brauner-Osborne, Hans; Burnstock, Geoffrey; Calo, Girolamo; Castano, Justo P.; Catt, Kevin J.; Ceruti, Stefania; Chazot, Paul; Chiang, Nan; Chini, Bice; Chun, Jerold; Cianciulli, Antonia; Civelli, Olivier; Clapp, Lucie H.; Couture, Rejean; Cox, Helen M.; Csaba, Zsolt; Dahlgren, Claes; Dent, Gordon; Douglas, Steven D.; Dournaud, Pascal; Eguchi, Satoru; Escher, Emanuel; Filardo, Edward J.; Fong, Tung; Fumagalli, Marta; Gainetdinov, Raul R.; Garelja, Michael L.; de Gasparo, Marc; Gerard, Craig; Gershengorn, Marvin; Gobeil, Fernand; Goodfriend, Theodore L.; Goudet, Cyril; Gratz, Lukas; Gregory, Karen J.; Gundlach, Andrew L.; Hamann, Jorg; Hanson, Julien; Hauger, Richard L.; Hay, Debbie L.; Heinemann, Akos; Herr, Deron; Hollenberg, Morley D.; Holliday, Nicholas D.; Horiuchi, Mastgugu; Hoyer, Daniel; Hunyady, Laszlo; Husain, Ahsan; Ijzerman, Adriaan P.; Inagami, Tadashi; Jacobson, Kenneth A.; Jensen, Robert T.; Jockers, Ralf; Jonnalagadda, Deepa; Karnik, Sadashiva; Kaupmann, Klemens; Kemp, Jacqueline; Kennedy, Charles; Kihara, Yasuyuki; Kitazawa, Takio; Kozielewicz, Pawel; Kreienkamp, Hans-Juergen; Kukkonen, Jyrki P.; Langenhan, Tobias; Larhammar, Dan; Leach, Katie; Lecca, Davide; Lee, John D.; Leeman, Susan E.; Leprince, Jerome; Li, Xaria X.; Lolait, Stephen J.; Lupp, Amelie; Macrae, Robyn; Maguire, Janet; Malfacini, Davide; Mazella, Jean; McArdle, Craig A.; Melmed, Shlomo; Michel, Martin C.; Miller, Laurence J.; Mitolo, Vincenzo; Mouillac, Bernard; Mueller, Christa E.; Murphy, Philip M.; Nahon, Jean-Louis; Ngo, Tony; Norel, Xavier; Nyimanu, Duuamene; O'Carroll, Anne-Marie; Offermanns, Stefan; Panaro, Maria Antonietta; Parmentier, Marc; Pertwee, Roger G.; Pin, Jean-Philippe; Prossnitz, Eric R.; Quinn, Mark; Ramachandran, Rithwik; Ray, Manisha; Reinscheid, Rainer K.; Rondard, Philippe; Rovati, G. Enrico; Ruzza, Chiara; Sanger, Gareth J.; Schoeneberg, Torsten; Schulte, Gunnar; Schulz, Stefan; Segaloff, Deborah L.; Serhan, Charles N.; Singh, Khuraijam Dhanachandra; Smith, Craig M.; Stoddart, Leigh A.; Sugimoto, Yukihiko; Summers, Roger; Tan, Valerie P.; Thal, David; Thomas, Walter (Wally); Timmermans, Pieter B. M. W. M.; Tirupula, Kalyan; Toll, Lawrence; Tulipano, Giovanni; Unal, Hamiyet; Unger, Thomas; Valant, Celine; Vanderheyden, Patrick; Vaudry, David; Vaudry, Hubert; Vilardaga, Jean-Pierre; Walker, Christopher S.; Wang, Ji Ming; Ward, Donald T.; Wester, Hans-Juergen; Willars, Gary B.; Williams, Tom Lloyd; Woodruff, Trent M.; Yao, Chengcan; Ye, Richard D.
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Endocytic proteins mediating GPR15 receptor internalization provide insight into the underlying mechanisms
err2023-05-01
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errDeng, Yufang; Von Moo, Ee; Inoue, Asuka; Braeuner-Osborne, Hans
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Pharmacological characterization of novel small molecule agonists and antagonists for the orphan receptor GPR139
err2023-03-01
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errPallareti, Lisa; Rath, Tine F.; Trapkov, Boris; Tsonkov, Tsonko; Nielsen, Anders Thorup; Harpsoe, Kasper; Gentry, Patrick R.; Brauner-Osborne, Hans; Gloriam, David E.; Foster, Simon R.
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Somatostatin venom analogs evolved by fish-hunting cone snails: From prey capture behavior to identifying drug leads
err2022-03-25
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errRamiro, Iris Bea L.; Bjorn-Yoshimoto, Walden E.; Imperial, Julita S.; Gajewiak, Joanna; Salcedo, Paula Florez; Watkins, Maren; Taylor, Dylan; Resager, William; Ueberheide, Beatrix; Brauner-Osborne, Hans; Whitby, Frank G.; Hill, Christopher P.; Martin, Laurent F.; Patwardhan, Amol; Concepcion, Gisela P.; Olivera, Baldomero M.; Safavi-Hemami, Helena
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Ligand-directed bias of G protein signaling at the dopamine D2 receptor
err2022-02-01
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errVon Moo, Ee; Harpsoe, Kasper; Hauser, Alexander S.; Masuho, Ikuo; Brauner-Osborne, Hans; Gloriam, David E.; Martemyanov, Kirill A.
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Molecular insights into ligand recognition and G protein coupling of the neuromodulatory orphan receptor GPR139
err2021-12-17
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errZhou, Yali; Daver, Henrik; Trapkov, Boris; Wu, Lijie; Wu, Meng; Harpsoe, Kasper; Gentry, Patrick R.; Liu, Kaiwen; Larionova, Marina; Liu, Junlin; Chen, Na; Brauner-Osborne, Hans; Gloriam, David E.; Hua, Tian; Liu, Zhi-Jie
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THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: G protein-coupled receptors药理学2021/22简明指南: g蛋白偶联受体
err2021-09-16
err359
errOAAI
errAlexander, Stephen P. H.; Christopoulos, Arthur; Davenport, Anthony P.; Kelly, Eamonn; Mathie, Alistair; Peters, John A.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Pawson, Adam J.; Southan, Christopher; Davies, Jamie A.; Abbracchio, Maria Pia; Alexander, Wayne; Al-hosaini, Khaled; Baeck, Magnus; Barnes, Nicholas M.; Bathgate, Ross; Beaulieu, Jean-Martin; Bernstein, Kenneth E.; Bettler, Bernhard; Birdsall, Nigel J. M.; Blaho, Victoria; Boulay, Francois; Bousquet, Corinne; Braeuner-Osborne, Hans; Burnstock, Geoffrey; Calo, Girolamo; Castano, Justo P.; Catt, KevinJ; Ceruti, Stefania; Chazot, Paul; Chiang, Nan; Chini, Bice; Chun, Jerold; Cianciulli, Antonia; Civelli, Olivier; Clapp, Lucie H.; Couture, Rejean; Csaba, Zsolt; Dahlgren, Claes; Dent, Gordon; Singh, Khuraijam Dhanachandra; Douglas, Steven D.; Dournaud, Pascal; Eguchi, Satoru; Escher, Emanuel; Filardo, Edward J.; Fong, Tung; Fumagalli, Marta; Gainetdinov, Raul R.; de Gasparo, Marc; Gerard, Craig; Gershengorn, Marvin; Gobeil, Fernand; Goodfriend, Theodore L.; Goudet, Cyril; Gregory, Karen J.; Gundlach, Andrew L.; Hamann, Joerg; Hanson, Julien; Hauger, Richard L.; Hay, Debbie L.; Heinemann, Akos; Hollenberg, Morley D.; Holliday, Nicholas D.; Horiuchi, Mastgugu; Hoyer, Daniel; Hunyady, Laszlo; Husain, Ahsan; IJzerman, Adriaan P.; Inagami, Tadashi; Jacobson, Kenneth A.; Jensen, Robert T.; Jockers, Ralf; Jonnalagadda, Deepa; Karnik, Sadashiva; Kaupmann, Klemens; Kemp, Jacqueline; Kennedy, Charles; Kihara, Yasuyuki; Kitazawa, Takio; Kozielewicz, Pawel; Kreienkamp, Hans-Juergen; Kukkonen, Jyrki P.; Langenhan, Tobias; Leach, Katie; Lecca, Davide; Lee, John D.; Leeman, Susan E.; Leprince, Jerome; Li, Xaria X.; Williams, Tom Lloyd; Lolait, Stephen J.; Lupp, Amelie; Macrae, Robyn; Maguire, Janet; Mazella, Jean; McArdle, Craig A.; Melmed, Shlomo; Michel, Martin C.; Miller, Laurence J.; Mitolo, Vincenzo; Mouillac, Bernard; Mueller, Christa E.; Murphy, Philip; Nahon, Jean-Louis; Ngo, Tony; Norel, Xavier; Nyimanu, Duuamene; Ocarroll, Anne-Marie; Offermanns, Stefan; Panaro, Maria Antonietta; Parmentier, Marc; Pertwee, Roger G.; Pin, Jean-Philippe; Prossnitz, Eric R.; Quinn, Mark; Ramachandran, Rithwik; Ray, Manisha; Reinscheid, Rainer K.; Rondard, Philippe; Rovati, G. Enrico; Ruzza, Chiara; Sanger, Gareth J.; Schoeneberg, Torsten; Schulte, Gunnar; Schulz, Stefan; Segaloff, Deborah L.; Serhan, Charles N.; Stoddart, Leigh A.; Sugimoto, Yukihiko; Summers, Roger; Tan, Valerie P.; Thal, David; Thomas, Walter (Wally); Timmermans, PieterB M. W. M.; Tirupula, Kalyan; Tulipano, Giovanni; Unal, Hamiyet; Unger, Thomas; Valant, Celine; Vanderheyden, Patrick; Vaudry, David; Vaudry, Hubert; Vilardaga, Jean-Pierre; Walker, Christopher S.; Wang, Ji Ming; Ward, Donald T.; Wester, Hans-Juergen; Willars, Gary B.; Woodruff, Trent M.; Yao, Chengcan; Ye, Richard D.
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Mutational Landscape of the Proglucagon-Derived Peptides
err2021-06-17
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errOAAI
errLindquist, Peter; Madsen, Jakob S.; Brauner-Osborne, Hans; Rosenkilde, Mette M.; Hauser, Alexander S.
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Positive Allosteric Modulators of Metabotropic Glutamate Receptor 5 as Tool Compounds to Study Signaling Bias
err2021-05-01
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errArsova, Angela; Moller, Thor C.; Hellyer, Shane D.; Vedel, Line; Foster, Simon R.; Hansen, Jakob L.; Brauner-Osborne, Hans; Gregory, Karen J.
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