P.A. Elkins - Publications, H-index & Citations

P.A. Elkins

University of Michigan

13H指数

38论文数

1.6K被引数

收录论文 8

发表时间

The exploration of aza-quinolines as hematopoietic prostaglandin D synthase (H-PGDS) inhibitors with low brain exposure

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2020-12-01

PREAI

Cadilla, Rodolfo; Deaton, David N.; Do, Young; Elkins, Patricia A.; Ennulat, Daniela; Guss, Jeffrey H.; Holt, Jason; Jeune, Michael R.; King, Andrew G.; Klapwijk, Jan C.; Kramer, H. Fritz; Kramer, Nicholas J.; Laffan, Susan B.; Masuria, Paresh, I; McDougal, Alan, V; Mortenson, Paul N.; Musetti, Caterina; Peckham, Gregory E.; Pietrak, Beth L.; Poole, Chuck; Price, Daniel J.; Rendina, Alan R.; Sati, Girish; Saxty, Gordon; Shearer, Barry G.; Shewchuk, Lisa M.; Sneddon, Helen F.; Stewart, Eugene L.; Stuart, J. Darren; Thomas, Dean N.; Thomson, Stephen A.; Ward, Paris; Wilson, Joseph W.; Xu, Tiahshun; Youngman, Mark A.

Discovery of Isoxazole Amides as Potent and Selective SMYD3 Inhibitors

ACS MEDICINAL CHEMISTRY LETTERS

IF4

2019-12-27

OAAI

Su, Dai-Shi; Qu, Junya; Schulz, Mark; Blackledge, Chuck W.; Yu, Hongyi; Zeng, Jenny; Burgess, Joelle; Reif, Alexander; Stern, Melissa; Nagarajan, Raman; Pappalardi, Melissa Baker; Wong, Kristen; Graves, Alan P.; Bonnette, William; Wang, Liping; Elkins, Patricia; Knapp-Reed, Beth; Carson, Jeffrey D.; McHugh, Charles; Mohammad, Helai; Kruger, Ryan; Luengo, Juan; Heerding, Dirk A.; Creasy, Caretha L.

CSAR 2014: A Benchmark Exercise Using Unpublished Data from Pharma

JOURNAL OF CHEMICAL INFORMATION AND MODELING

IF5.3

2016-05-17

OAAI

Carlson, Heather A.; Smith, Richard D.; Damm-Ganamet, Kelly L.; Stuckey, Jeanne A.; Ahmed, Aqeel; Convery, Maire A.; Somers, Donald O.; Kranz, Michael; Elkins, Patricia A.; Cui, Guanglei; Peishoff, Catherine E.; Lambert, Millard H.; Dunbar, James B., Jr.

Discovery of a Potent Class of PI3Kα Inhibitors with Unique Binding Mode via Encoded Library Technology (ELT)

ACS MEDICINAL CHEMISTRY LETTERS

IF4

2015-04-08

OAAI

Yang, Hongfang; Medeiros, Patricia F.; Raha, Kaushik; Elkins, Patricia; Lind, Kenneth E.; Lehr, Ruth; Adams, Nicholas D.; Burgess, Joelle L.; Schmidt, Stanley J.; Knight, Steven D.; Auger, Kurt R.; Schaber, Michael D.; Franklin, G. Joseph; Ding, Yun; DeLorey, Jennifer L.; Centrella, Paolo A.; Mataruse, Sibongile; Skinner, Steven R.; Clark, Matthew A.; Cuozzo, John W.; Evindar, Ghotas

Discovery of GSK2126458, a Highly Potent Inhibitor of PI3K and the Mammalian Target of Rapamycin

ACS MEDICINAL CHEMISTRY LETTERS

IF4

2010-01-19

367

OAAI

Knight, Steven D.; Adams, Nicholas D.; Burgess, JoeIle L.; Chaudhari, Amita M.; Darcy, Michael G.; Donatelli, Carla A.; Luengo, Juan I.; Newlander, Ken A.; Parrish, Cynthia A.; Ridgers, Lance H.; Sarpong, Martha A.; Schmidt, Stanley J.; Van Aller, Glenn S.; Carson, Jeffrey D.; Diamond, Melody A.; Elkins, Patricia A.; Gardiner, Christine M.; Garver, Eric; Gilbert, Seth A.; Gontarek, Richard R.; Jackson, Jeffrey R.; Kershner, Kevin L.; Luo, Lusong; Raha, Kaushik; Sherk, Christian S.; Sung, Chiu-Mei; Sutton, David; Tummino, Peter J.; Wegrzyn, Ronald J.; Auger, Kurt R.; Dhanak, Dashyant

Potent, Selective and Orally Bioavailable Dihydropyrimidine Inhibitors of Rho Kinase (ROCK1) as Potential Therapeutic Agents for Cardiovascular Diseases

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2008-10-09

PREAI

Sehon, Clark A.; Wang, Gren Z.; Viet, Andrew Q.; Goodman, Krista B.; Dowdell, Sarah E.; Elkins, Patricia A.; Semus, Simon F.; Evans, Christopher; Jolivette, Larry J.; Kirkpatrick, Robert B.; Dul, Edward; Khandekar, Sanjay S.; Yi, Tracey; Wright, Lois L.; Srnith, Gary K.; Behm, David J.; Bentley, Ross; Doe, Christopher P.; Hu, Erding; Lee, Dennis

Discovery of aminofurazan-azabenzimidazoles as inhibitors of Rho-kinase with high kinase selectivity and antihypertensive activity

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2006-12-15

PREAI

Stavenger, Robert A.; Cui, Haifeng; Dowdell, Sarah E.; Franz, Robert G.; Gaitanopoulos, Dimitri E.; Goodman, Krista B.; Hilfiker, Mark A.; Ivy, Robert L.; Leber, Jack D.; Marino, Joseph P., Jr.; Oh, Hye-Ja; Viet, Andrew Q.; Xu, Weiwei; Ye, Guosen; Zhang, Daohua; Zhao, Yongdong; Jolivette, Larry J.; Head, Martha S.; Semus, Simon F.; Elkins, Patricia A.; Kirkpatrick, Robert B.; Dul, Edward; Khandekar, Sanjay S.; Yi, Tracey; Jung, David K.; Wright, Lois L.; Smith, Gary K.; Behm, David J.; Doe, Christopher P.; Bentley, Ross; Chen, Zunxuan X.; Hu, Erding; Lee, Dennis

Indole naphthyridinones as inhibitors of bacterial enoyl-ACP reductases FabI and FabK

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2003-03-25

177

PREAI

Seefeld, MA; Miller, WH; Newlander, KA; Burgess, WJ; DeWolf, WE; Elkins, PA; Head, MS; Jakas, DR; Janson, CA; Keller, PM; Manley, PJ; Moore, TD; Payne, DJ; Pearson, S; Polizzi, BJ; Qiu, XY; Rittenhouse, SF; Uzinskas, IN; Wallis, NG; Huffmann, WF

研究方向