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J

John J. Renger

merck & company

56H指数
178论文数
9.2K被引数
收录论文 54
发表时间
PET imaging of M4 muscarinic acetylcholine receptors in rhesus macaques using [11C]MK-6884: Quantification with kinetic modeling and receptor occupancy by CVL-231 (emraclidine), a novel positive allosteric modulator
err2024-03-13
err3
PREAI
errBelov, Vasily; Guehl, Nicolas J.; Duvvuri, Sridhar; Iredale, Philip; Moon, Sung-Hyun; Dhaynaut, Maeva; Chakilam, Srinivas; MacDonagh, Alexander C.; Rice, Peter A.; Yokell, Daniel L.; Renger, John J.; El Fakhri, Georges; Normandin, Marc D.
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Phase 1 Trial of Darigabat for the Reduction of Acute Psychological and Physiological Panic and Fear Symptoms Following CO2 Inhalation in Healthy Participants
err2023-04-25
err1
PREAI
errGurrell, Rachel; Chang, Ih; Dandurand, Ann; Duvvuri, Sridhard; Guigliano, Amy; Pastino, Gina; Pham, Theresa; Versavel, Stacey; Jacobs, Gabriel; Pour, Koshar Safai; Zuiker, Rob; Sanchez, Raymond; Renger, John
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Parkinson disease among patients treated for benign prostatic hyperplasia with α1 adrenergic receptor antagonists
err2021-06-01
err21
errOAAI
errSasane, Rahul; Bartels, Amy; Field, Michelle; Sierra, Maria I.; Duvvuri, Sridhar; Gray, David L.; Pin, Sokhom S.; Renger, John J.; Stone, David J.
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Cross-species systems analysis identifies gene networks differentially altered by sleep loss and depression
err2018-07-06
err21
errOAAI
errScarpa, Joseph R.; Jiang, Peng; Gao, Vance D.; Fitzpatrick, Karrie; Millstein, Joshua; Olker, Christopher; Gotter, Anthony; Winrow, Christopher J.; Renger, John J.; Kasarskis, Andrew; Turek, Fred W.; Vitaterna, Martha H.
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Aging African green monkeys manifest transcriptional, pathological, and cognitive hallmarks of human Alzheimer's disease
err2018-04-01
err45
PREAI
errCramer, Paige E.; Gentzel, Renee C.; Tanis, Keith Q.; Vardigan, Joshua; Wang, Yi; Connolly, Brett; Manfre, Philip; Lodge, Kenneth; Renger, John J.; Zerbinatti, Celina; Uslaner, Jason M.
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Transcriptional Profiling of Cholinergic Neurons From Basal Forebrain Identifies Changes in Expression of Genes Between Sleep and Wake来自基底前脑的胆碱能神经元的转录谱分析确定睡眠和觉醒之间基因表达的变化
errSLEEP
IF4.9
err2017-04-18
err11
errOAAI
errNikonova, Elena V.; Gilliland, Jason D. A.; Tanis, Keith Q.; Podtelezhnikov, Alexei A.; Rigby, Alison M.; Galante, Raymond J.; Finney, Eva M.; Stone, David J.; Renger, John J.; Pack, Allan I.; Winrow, Christopher J.
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Discovery of a 3-(4-Pyrimidinyl) Indazole (MLi-2), an Orally Available and Selective Leucine-Rich Repeat Kinase 2 (LRRK2) Inhibitor that Reduces Brain Kinase Activity
err2017-03-16
err113
PREAI
errScott, Jack D.; DeMong, Duane E.; Greshock, Thomas J.; Basu, Kallol; Dai, Xing; Harris, Joel; Hruza, Alan; Li, Sarah W.; Lin, Sue-Ing; Liu, Hong; Macala, Megan K.; Hu, Zhiyong; Mei, Hong; Zhang, Honglu; Walsh, Paul; Poirier, Marc; Shi, Zhi-Cai; Xiao, Li; Agnihotri, Gautam; Baptista, Marco A. S.; Columbus, John; Fell, Matthew J.; Hyde, Lynn A.; Kuvelkar, Reshma; Lin, Yinghui; Mirescu, Christian; Morrow, John A.; Yin, Zhizhang; Zhang, Xiaoping; Zhou, Xiaoping; Chang, Ronald K.; Embrey, Mark W.; Sanders, John M.; Tiscia, Heather E.; Drolet, Robert E.; Kern, Jonathan T.; Sur, Sylvie M.; Renger, John J.; Bilodeau, Mark T.; Kennedy, Matthew E.; Parker, Eric M.; Stamford, Andrew W.; Nargund, Ravi; McCauley, John A.; Miller, Michael W.
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The Discovery of Suvorexant, the First Orexin Receptor Drug for Insomnia
err2017-01-06
err100
PREAI
errColeman, Paul J.; Gotter, Anthony L.; Herring, W. Joseph; Winrow, Christopher J.; Renger, John J.
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Orexin 2 Receptor Antagonism is Sufficient to Promote NREM and REM Sleep from Mouse to Man
err2016-06-03
err70
errOAAI
errGotter, Anthony L.; Forman, Mark S.; Harrell, Charles M.; Stevens, Joanne; Svetnik, Vladimir; Yee, Ka Lai; Li, Xiaodong; Roecker, Anthony J.; Fox, Steven V.; Tannenbaum, Pamela L.; Garson, Susan L.; De Lepeleire, Inge; Calder, Nicole; Rosen, Laura; Struyk, Arie; Coleman, Paul J.; Herring, W. Joseph; Renger, John J.; Winrow, Christopher J.
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Identification and in Vivo Evaluation of Liver X Receptor β-Selective Agonists for the Potential Treatment of Alzheimer's Disease
err2016-04-01
err41
errOAAI
errStachel, Shawn J.; Zerbinatti, Celina; Rudd, Michael T.; Cosden, Mali; Suon, Sokreine; Nanda, Kausik K.; Wessner, Keith; DiMuzio, Jillian; Maxwell, Jill; Wu, Zhenhua; Uslaner, Jason M.; Michener, Maria S.; Szczerba, Peter; Brnardic, Edward; Rada, Vanessa; Kim, Yuntae; Meissner, Robert; Wuelfing, Peter; Yuan, Yang; Ballard, Jeanine; Holahan, Marie; Klein, Daniel J.; Lu, Jun; Fradera, Xavier; Parthasarathy, Gopal; Uebele, Victor N.; Chen, Zhongguo; Li, Yingjie; Li, Jian; Cooke, Andrew J.; Bennett, D. Jonathan; Bilodeau, Mark T.; Renger, John
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Structure and ligand-binding mechanism of the human OX1 and OX2 orexin receptors
err2016-03-07
err117
PREAI
errYin, Jie; Babaoglu, Kerim; Brautigam, Chad A.; Clark, Lindsay; Shao, Zhenhua; Scheuermann, Thomas H.; Harrell, Charles M.; Gotter, Anthony L.; Roecker, Anthony J.; Winrow, Christopher J.; Renger, John J.; Coleman, Paul J.; Rosenbaum, Daniel M.
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Inhibition of Orexin Signaling Promotes Sleep Yet Preserves Salient Arousability in Monkeys
errSLEEP
IF4.9
err2016-03-01
err40
errOAAI
errTannenbaum, Pamela L.; Tye, Spencer J.; Stevens, Joanne; Gotter, Anthony L.; Fox, Steven V.; Savitz, Alan T.; Coleman, Paul J.; Uslaner, Jason M.; Kuduk, Scott D.; Hargreaves, Richard; Winrow, Christopher J.; Renger, John J.
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New approach for analyzing self-reporting of insomnia symptoms reveals a high rate of comorbid insomnia across a wide spectrum of chronic diseases
err2015-11-01
err19
errOAAI
errKatic, Bozena; Heywood, James; Turek, Fred; Chiauzzi, Emil; Vaughan, Timothy E.; Simacek, Kristina; Wicks, Paul; Jain, Sachin; Winrow, Christopher; Renger, John J.
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Discovery and Optimization of a Series of Pyrimidine-Based Phosphodiesterase 10A (PDE10A) Inhibitors through Fragment Screening, Structure-Based Design, and Parallel Synthesis
err2015-09-25
err52
PREAI
errShipe, William D.; Sharik, Steven S.; Barrow, James C.; McGaughey, Georgia B.; Theberge, Cory R.; Uslaner, Jason M.; Yan, Youwei; Renger, John J.; Smith, Sean M.; Coleman, Paul J.; Cox, Christopher D.
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Evidence for orexinergic mechanisms in migraine
err2015-02-01
err76
PREAI
errHoffmann, Jan; Supronsinchai, Weera; Akerman, Simon; Andreou, Anna P.; Winrow, Christopher J.; Renger, John; Hargreaves, Richard; Goadsby, Peter J.
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Improved cognition without adverse effects: novel M1 muscarinic potentiator compares favorably to donepezil and xanomeline in rhesus monkey
err2014-12-10
err57
PREAI
errVardigan, Joshua D.; Cannon, Christopher E.; Puri, Vanita; Dancho, Mandy; Koser, AmyJo; Wittmann, Marion; Kuduk, Scott D.; Renger, John J.; Uslaner, Jason M.
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Orexin receptor antagonists and insomnia treatment: state of the art
err2014-10-01
err0
PREAI
errGotter, A. L.; Coleman, P. J.; Kuduk, S. D.; Tannenbaum, P. L.; Struyk, A.; Wrishko, R. E.; Connor, K. M.; Herring, W. J.; Renger, J. J.; Winrow, C. J.
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Blood-Gene Expression Reveals Reduced Circadian Rhythmicity in Individuals Resistant to Sleep Deprivation
errSLEEP
IF4.9
err2014-10-01
err59
errOAAI
errArnardottir, Erna S.; Nikonova, Elena V.; Shockley, Keith R.; Podtelezhnikov, Alexei A.; Anafi, Ron C.; Tanis, Keith Q.; Maislin, Greg; Stone, David J.; Renger, John J.; Winrow, Christopher J.; Pack, Allan I.
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Cross-Modulation and Molecular Interaction at the Cav3.3 Protein between the Endogenous Lipids and the T-Type Calcium Channel Antagonist TTA-A2.
err2014-02-01
err18
errOAAI
errCazade, Magali; Nuss, Cindy E.; Bidaud, Isabelle; Renger, John J.; Uebele, Victor N.; Lory, Philippe; Chemin, Jean
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Discovery of 5-Chloro-N-[( 5,6-dimethoxypyridin-2-yl)methyl]-2,2′:5′,3-terpyridine-3′-carboxamide (MK-1064): A Selective Orexin 2 Receptor Antagonist (2-SORA) for the Treatment of Insomnia
err2013-12-27
err78
PREAI
errRoecker, Anthony J.; Mercer, Swati P.; Schreier, John D.; Cox, Christopher D.; Fraley, Mark E.; Steen, Justin T.; Lemaire, Wei; Bruno, Joseph G.; Harrell, C. Meacham; Garson, Susan L.; Gotter, Anthony L.; Fox, Steven V.; Stevens, Joanne; Tannenbaum, Pamela L.; Prueksaritanont, Thomayant; Cabalu, Tamara D.; Cui, Donghui; Stellabott, Joyce; Hartman, George D.; Young, Steven D.; Winrow, Christopher J.; Renger, John J.; Coleman, Paul J.
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