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收藏Potent and Selective Human 5-HT2B Serotonin Receptor Antagonists: 4′-Cyano-(N)-methanocarba-adenosines by Synthetic Serendipity
Tosh, Dilip K.; Pavan, Matteo; Clark, Allison A.; Lammers, Josie; Villano, Serafina; Marri, Silvia; Sgambellone, Silvia; Choi, Suebin; Lee, Jihyun; Ivancich, Marko S.; Bock, Hailey A.; Campbell, Ryan G.; Lewicki, Sarah A.; Levitan, Ian M.; Chen, Eric; Liu, Naili; Demby, Tamar; Gavrilova, Oksana; Gao, Zhan-Guo; Lucarini, Laura; Mccorvy, John D.; Jacobson, Kenneth A.
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收藏Lipodystrophy in methylmalonic acidemia associated with elevated FGF21 and abnormal methylmalonylation
Manoli, Irini; Sysol, Justin R.; Head, PamelaSara E.; Epping, Madeline W.; Gavrilova, Oksana; Crocker, Melissa K.; Sloan, Jennifer L.; Koutsoukos, Stefanos A.; Wang, Cindy; Ktena, Yiouli P.; Mendelson, Sophia; Pass, Alexandra R.; Zerfas, Patricia M.; Hoffmann, Victoria; Vernon, Hilary J.; Fletcher, Laura A.; Reynolds, James C.; Tsokos, Maria G.; Stratakis, Constantine A.; Voss, Stephan D.; Chen, Kong Y.; Brown, Rebecca J.; Hamosh, Ada; Berry, Gerard T.; Chen, Xiaoyuan Shawn; Yanovski, Jack A.; Venditti, Charles P.
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收藏A human obesity-associated MC4R mutation with defective Gq/11α signaling leads to hyperphagia in mice
Metzger, Peter J.; Zhang, Aileen; Carlson, Bradley A.; Sun, Hui; Cui, Zhenzhong; Li, Yongqi; Jahnke, Marshal T.; Layton, Daniel R.; Gupta, Meenakshi B.; Liu, Naili; Kostenis, Evi; Gavrilova, Oksana; Chen, Min; Weinstein, Lee S.
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收藏2-Amino-5-arylethynyl-thiophen-3-yl-(phenyl)methanones as A1 Adenosine Receptor Positive Allosteric Modulators
Oliva, Paola; Suresh, R. Rama; Pasquini, Silvia; Salmaso, Veronica; Will, Edward J.; Tosh, Dilip K.; Gao, Zhan-Guo; Liu, Naili; Gavrilova, Oksana; Vincenzi, Fabrizio; Varani, Katia; Jacobson, Kenneth A.
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收藏CDK4-E2F3 signals enhance oxidative skeletal muscle fiber numbers and function to affect myogenesis and metabolismCDK4-E2F3信号增强氧化骨骼肌纤维数量和功能以影响肌生成和代谢
Bahn, Young Jae; Yadav, Hariom; Piaggi, Paolo; Abel, Brent S.; Gavrilova, Oksana; Springer, Danielle A.; Papazoglou, Ioannis; Zerfas, Patricia M.; Skarulis, Monica C.; McPherron, Alexandra C.; Rane, Sushil G.
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收藏Constitutive and conditional deletion reveals distinct phenotypes driven by developmental versus neurotransmitter actions of the neuropeptide PACAP
Bakalar, Dana; Gavrilova, Oksana; Jiang, Sunny Z.; Zhang, Hai-ying; Roy, Snehashis; Williams, Sarah K.; Liu, Naili; Wisser, Stephen; Usdin, Ted B.; Eiden, Lee E.
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收藏Radiolabeled αvβ3 analog 177Lu-EB-RGD is an effective therapeutic agent in thyroid cancer xenograft mouse model
Kumari, Sonam; Wang, Zhantong; Thakur, Shilpa; Abaandou, Laura; Gavrilova, Oksana; Lu, Huiyan; Lang, Lixin; Kiesewetter, Dale; Vasko, Vasyl; Klubo-Gwiezdzinska, Joanna
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收藏Growth, adipose, brain, and skin alterations resulting from targeted disruption of the mouse peroxisome proliferator-activated receptor β(δ)
Peters, JM; Lee, SST; Li, W; Ward, JM; Gavrilova, O; Everett, C; Reitman, ML; Hudson, LD; Gonzalez, FJ
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收藏The Winged Helix Transcription Factor Foxa3 Regulates Adipocyte Differentiation and Depot-Selective Fat Tissue Expansion
Xu, Lingyan; Panel, Valentine; Ma, Xinran; Du, Chen; Hugendubler, Lynne; Gavrilova, Oksana; Liu, Alice; McLaughlin, Tracey; Kaestner, Klaus H.; Muellera, Elisabetta
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收藏Epigenetic regulation of white adipose tissue plasticity and energy metabolism by nucleosome binding HMGN proteins
Nanduri, Ravikanth; Furusawa, Takashi; Lobanov, Alexei; He, Bing; Xie, Carol; Dadkhah, Kimia; Kelly, Michael C.; Gavrilova, Oksana; Gonzalez, Frank J.; Bustin, Michael
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收藏Intestinal peroxisome proliferator-activated receptor α-fatty acid-binding protein 1 axis modulates nonalcoholic steatohepatitis肠过氧化物酶体增殖物激活受体 α-脂肪酸结合蛋白1轴调节非酒精性脂肪性肝炎
Yan, Tingting; Luo, Yuhong; Yan, Nana; Hamada, Keisuke; Zhao, Nan; Xia, Yangliu; Wang, Ping; Zhao, Changdong; Qi, Dan; Yang, Shoumei; Sun, Lulu; Cai, Jie; Wang, Qiong; Jiang, Changtao; Gavrilova, Oksana; Krausz, Kristopher W.; Patel, Daxesh P.; Yu, Xiaoting; Wu, Xuan; Hao, Haiping; Liu, Weiwei; Qu, Aijuan; Gonzalez, Frank J.
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收藏Adipocyte Gq signaling is a regulator of glucose and lipid homeostasis in mice脂肪细胞Gq信号是小鼠葡萄糖和脂质稳态的调节剂
Kimura, Takefumi; Pydi, Sai P.; Wang, Lei; Haspula, Dhanush; Cui, Yinghong; Lu, Huiyan; Koenig, Gabriele M.; Kostenis, Evi; Steinberg, Gregory R.; Gavrilova, Oksana; Wess, Juergen
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收藏Clenbuterol exerts antidiabetic activity through metabolic reprogramming of skeletal muscle cells克伦特罗通过骨骼肌细胞的代谢重编程发挥抗糖尿病活性
Meister, Jaroslawna; Bone, Derek B. J.; Knudsen, Jonas R.; Barella, Luiz F.; Velenosi, Thomas J.; Akhmedov, Dmitry; Lee, Regina J.; Cohen, Amanda H.; Gavrilova, Oksana; Cui, Yinghong; Karsenty, Gerard; Chen, Min; Weinstein, Lee S.; Kleinert, Maximilian; Berdeaux, Rebecca; Jensen, Thomas E.; Richter, Erik A.; Wess, Jurgen
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收藏A3 adenosine receptor agonists containing dopamine moieties for enhanced interspecies affinity
Tosh, Dilip K.; Salmaso, Veronica; Campbell, Ryan G.; Rao, Harsha; Bitant, Amelia; Pottie, Eline; Stove, Christophe P.; Liu, Naili; Gavrilova, Oksana; Gao, Zhan-Guo; Auchampach, John A.; Jacobson, Kenneth A.
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收藏In vivo metabolic effects after acute activation of skeletal muscle Gs signaling
Meister, Jaroslawna; Bone, Derek B. J.; Knudsen, Jonas R.; Barella, Luiz F.; Liu, Liu; Lee, Regina; Gavrilova, Oksana; Chen, Min; Weinstein, Lee S.; Kleinert, Maximilian; Jensen, Thomas E.; Wess, Juergen
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