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Design, synthesis, docking studies and bioactivity evaluation of 1,2,3-triazole eugenol derivatives Cutrim, Thiago Antonio de Sousa; Barcelos, Fernando Fontes; Meireles, Leandra Martins; Gazolla, Poliana Aparecida Rodrigues; Lima, angela Maria Almeida; Teixeira, Robson Ricardo; Moreira, Luiza Carvalheira; de Queiroz, Vagner Tebaldi; Barbosa, Luiz Claudio Almeida; Morais, Pedro Alves Bezerra; do Nascimento, Claudia Jorge; Junker, Jochen; Costa, Adilson Vidal; Fronza, Marcio; Scherer, Rodrigo 分享 收藏
NMR analysis, cytotoxic activity and theoretical study of a complex between SRPIN340 and p-sulfonic acid calix[6]arene Viol, Livia Cristina de Souza; Silva, Natalia Aparecida Liberto; Cerceau, Cristiane Isaac; Barros, Marcus Vinicius de Andrade; Siqueira, Raoni Pais; Goncalves, Victor Hugo Sousa; Bressan, Gustavo Costa; Fernandes, Sergio Antonio; Alvarenga, Elson Santiago; Teixeira, Robson Ricardo 分享 收藏
Design and Synthesis of Eugenol Derivatives Bearing a 1,2,3-Triazole Moiety for Papaya Protection against Colletotrichum gloeosporioides Lima, Angela Maria Almeida; Moreira, Luiza Carvalheira; Gazolla, Poliana Rodrigues; Oliveira, Mariana Belizario; Teixeira, Robson Ricardo; Queiroz, Vagner Tebaldi; Rocha, Matheus Ricardo; Moraes, Willian Bucker; dos Santos, Nayara Araujo; Romao, Wanderson; Lacerda Jr, Valdemar; Morais, Pedro Alves Bezerra; de Oliveira, Osmair Vital; de Jesus Junior, Waldir Cintra; Barbosa, Luiz C. A.; Nascimento, Claudia Jorge; Junker, Jochen; Costa, Adilson Vidal 分享 收藏
New synthetic molecules incorporated into polymeric micelles used for treatment against visceral leishmaniasis Freitas, Camila S.; Pereira, Isabela A. G.; Lage, Daniela P.; Vale, Danniele L.; Pimenta, Breno L.; Soares, Nicia P.; Santiago, Samira S.; Martins, Vivian T.; Camara, Raquel S. B.; Jesus, Marcelo M.; Tavares, Grasiele S. V.; Ramos, Fernanda F.; Ludolf, Fernanda; Magalhaes, Licia N. D.; Oliveira, Fabricio M.; Duarte, Mariana C.; Chavez-Fumagalli, Miguel A.; Costa, Adilson V.; Roatt, Bruno M.; Teixeira, Robson R.; Coelho, Eduardo A. F. 分享 收藏
Leishmanicidal activity and 4D quantitative structure-activity relationship and molecular docking studies of vanillin-containing 1,2,3-triazole derivatives Gazolla, Poliana Aparecida Rodrigues; Lima, Wallace Pacienza; de Aguiar, Alex Ramos; Borsodi, Maria Paula Goncalves; Costa, Adilson Vidal; de Oliveira, Fabricio Marques; de Oliveira, Osmair Vital; Costa, Maria Cristina Andreazza; Ferreira, Marcia Miguel Castro; do Nascimento, Claudia Jorge; Junker, Jochen; Vaz, Boniek Gontijo; Teixeira, Robson Ricardo 分享 收藏
Novel diamides inspired by protein kinase inhibitors as anti-Trypanosoma cruzi agents: in vitro and in vivo evaluations Torchelsen, Fernanda Karoline Vieira da Silva; Pedrosa, Tamiles Caroline Fernandes; Rodrigues, Michelle Peixoto; de Aguiar, Alex Ramos; de Oliveira, Fabricio Marques; Amarante, Giovanni Wilson; Sales-Junior, Policarpo Ademar; Branquinho, Renata Tupinamba; da Silva, Sirlaine Pio Gomes; Talvani, Andre; Murta, Silvane Maria Fonseca; Martins, Felipe Terra; Braun, Rodrigo Ligabue; Teixeira, Robson Ricardo; Mosqueira, Vanessa Carla Furtado; de Lana, Marta 分享 收藏
Synthesis of 1,2,3-Triazole-Containing Methoxylated Cinnamides and Their Antileishmanial Activity against the Leishmania braziliensis Species dos Santos, Fabiola Suelen; de Freitas, Rossimiriam Pereira; de Freitas, Camila Simoes; Mendonca, Debora Vasconcelos Costa; Lage, Daniela Pagliara; Tavares, Grasiele de Sousa Vieira; Machado, Amanda Sanchez; Martins, Vivian Tamieti; Costa, Adilson Vidal; de Queiroz, Vagner Tebaldi; de Oliveira, Mariana Belizario; de Oliveira, Fabricio Marques; Antinarelli, Luciana Maria Ribeiro; Coimbra, Elaine Soares; Pilau, Eduardo Jorge; da Silva, Geovane Perez; Coelho, Eduardo Antonio Ferraz; Teixeira, Robson Ricardo 分享 收藏
Herbicide and Cytogenotoxic Activity of Inclusion Complexes of Psidium gaudichaudianum Leaf Essential Oil and β-Caryophyllene on 2-Hydroxypropyl-β-cyclodextrin Mendes, Luiza Alves; Vasconcelos, Loren Cristina; Fontes, Milene Miranda Praca; Martins, Geisiele Silva; Bergamin, Aline dos Santos; Silva, Matheus Alves; Silva, Rafael Resende Assis; de Oliveira, Taila Veloso; Souza, Victor Gomes Lauriano; Ferreira, Marcia Flores da Silva; Teixeira, Robson Ricardo; Lopes, Renata Pereira 分享 收藏
Structure-based discovery of thiosemicarbazones as SARS-CoV-2 main protease inhibitors 氨基硫脲作为SARS-CoV-2主要蛋白酶抑制剂的基于结构的发现 Maltarollo, Vinicius Goncalves; da Silva, Elany Barbosa; Kronenberger, Thales; Andrade, Marina Mol Sena; Marques, Gabriel V. de Lima; Oliveira, Nereu J. Candido; Santos, Lucianna H.; Rezende Junior, Celso de Oliveira; Martinho, Ana C. Cassiano; Skinner, Danielle; Fajtova, Pavla; Fernandes, Thais H.; dos Santos, Eduardo da Silveira; Gazolla, Poliana A. Rodrigues; de Souza, Ana P. Martins; da Silva, Milene Lopes; dos Santos, Fabiola S.; Lavorato, Stefania N.; Bretas, Ana C. Oliveira; Carvalho, Diogo Teixeira; Franco, Lucas Lopardi; Luedtke, Stephanie; Giardini, Miriam A.; Poso, Antti; Dias, Luiz C.; Podust, Larissa M.; Alves, Ricardo J.; McKerrow, James; Andrade, Saulo F.; Teixeira, Robson R.; Siqueira-Neto, Jair L.; O'Donoghue, Anthony; de Oliveira, Renata B.; Ferreira, Rafaela S. 分享 收藏
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Synthesis and Fungicide Activity on Asperisporium caricae of Glycerol Derivatives Bearing 1,2,3-Triazole Fragments Lima, Angela Maria Almeida; Teixeira, Robson Ricardo; Moraes, Willian Bucker; Rocha, Matheus Ricardo; Moraes, Arlan Figueiredo Carvalho; Gomes, Samela Cansi; Gazolla, Poliana Rodrigues; Silva, Silma Francielle; Queiroz, Vagner Tebaldi; Fonseca, Victor Rocha; Romao, Wanderson; Morais, Pedro Alves Bezerra; Lacerda, Valdemar; de Abreu, Lucas Magalha; Oliveira, Fabricio Marques; de Oliveira, Osmair Vital; Costa, Adilson Vidal 分享 收藏
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Immunomodulatory activity of trifluoromethyl arylamides derived from the SRPK inhibitor SRPIN340 and their potential use as vaccine adjuvant Mendes, Flavia Carneiro; de Paiva, Janine Cerqueira; Goncalves da Silva, Eloi Quintas; Santos, Marcus Reboucas; de Almeida Lima, Graziela Domingues; Moreira, Gabriela Alves; Silva, Lucas Viana Gomes; Agripino, Joice de Melo; de Souza, Ana Paula Martins; Mendes, Tiago Antonio de Oliveira; Machado-Neves, Mariana; Ricardo Teixeira, Robson; Silva-Junior, Abelardo; Rangel Fietto, Juliana Lopes; de Oliveira, Leandro Licursi; Bressan, Gustavo Costa 分享 收藏
The SRPK inhibitor N-(2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl) isonicotinamide (SRPIN340) increases the immune response against metastatic melanoma in mice Moreira, Gabriela Alves; Magalhaes Caetano, Monica Maria; do Vale, Juliana Alves; de Paiva, Janine Cerqueira; Sousa Goncalves, Victor Hugo; Almeida, Alisson Andrade; Gomes Silva, Lucas Viana; Giordano Martim, Fernanda Rebellato; de Andrade Barros, Marcus Vinicius; Guimaraes, Gabriela Rapozo; Santos, Leandro de Oliveira; Martins de Souza, Ana Paula; Machado-Neves, Mariana; Teixeira, Robson Ricardo; Silva-Junior, Abelardo; Rangel Fietto, Juliana Lopes; Boroni, Mariana; de Oliveira, Leandro Licursi; Bressan, Gustavo Costa 分享 收藏
Synthesis of cinnamic acid ester derivatives with antiproliferative and antimetastatic activities on murine melanoma cells 对小鼠黑色素瘤细胞具有抗增殖和抗转移活性的肉桂酸酯衍生物的合成 do Vale, Juliana Alves; Rodrigues, Michelle Peixoto; Lima, Angela Maria Almeida; Santiago, Samira Soares; de Almeida Lima, Graziela Domingues; Almeida, Alisson Andrade; de Oliveira, Leandro Licursi; Bressan, Gustavo Costa; Teixeira, Robson Ricardo; Machado-Neves, Mariana 分享 收藏
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