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Birgit Kosjek

Merck & Co., Inc.

27H指数
53论文数
2.3K被引数
收录论文 28
发表时间
Biocatalytic cascades enable manufacture of the macrocyclic peptide enlicitide生物催化级联实现大环肽enlicitide的制造
errScience
IF45.8
err2026-05-07
err0
PREAI
errArtis Klapars; Anna Fryszkowska; Stephanie Galanie; Omer Ad; Ellen Y. Aguilera; Nnamdi Akporji; Chihui An; Stephanus Axnanda; Tewoderos M. Ayele; Richard S. Ayikpoe; Rodell C. Barrientos; Matthew R. Bauerle; Marc R. Becker; Kevin M. Belyk; Lisa Bereznitski; Jackson K. B. Cahn; Karla Camacho Soto; Louis-Charles Campeau; Kevin R. Campos; Anagha Chandra; Hsieh Yao Darryl Chang; Mengbin Chen; Zhiwei Chen; Wai Ling Cheung-Lee; Cheol K. Chung; Stephanie W. Chun; Sarah S. Co; Ryan D. Cohen; Stephen M. Dalby; Guilherme Dal Poggetto; Truc Do; Spencer D. Dreher; Riki J. Drout; Noah P. Dunham; Yi Fan; Ryan M. Flessner; Jacob H. Forstater; Scott P. France; Janaka C. Gamekkanda; Donald R. Gauthier; Agnieszka A. Gil; Jacob W. Greenwood; Noel Ha; Holst M. Halsey; Xinxin Han; Michael Hartmann; Clara Hartmanshenn; Yu He; Edgar Hernandez; Kaori Hiraga; Hsing-I Ho; Cynthia M. Hong; Alan Hruza; Hang Hu; Kari Hullen; Alan M. Hyde; Tetsuji Itoh; Chey M. Jones; Woo-Ok Jung; Kanan Kanuga; James Levi Knippel; Joshua N. Kolev; Jongrock Kong; Birgit Kosjek; Sara Koynov; Michael H. Kress; Bharath Krishnamurthi; Jeffrey T. Kuethe; Thomas T. Kwok; Alfred Y. Lee; Joshua Lee; Qiuhan Li; Shasha Li; Jing Liao; Wenjun Liu; Gurpreet Longia; Emma Madrigal; Peter E. Maligres; Kevin M. Maloney; Erin L. McCarthy; John A. McIntosh; Samaneh Mesbahi-Vasey; Margaret Miller; Mansi Modi; Jeffrey C. Moore; Debopreeti Mukherjee; Grant S. Murphy; Jennifer Victoriano Obligacion; Weilan Pan; Julia Parzecki; Anisha Patel; Teng Peng; Byron K. Peters; Tiffany Piou; Carlos A. Pons Siepermann; Christopher K. Prier; Akasha K. Purohit; Yangzhong Qin; Erik L. Regalado; Mikhail Reibarkh; Nelo R. Rivera; Sandra A. Robaire; Lee Robison; Syamantak Roy; Rebecca T. Ruck; Katie A. Rykaczewski; Christopher H. Schuster; Erica L. Schwalm; Andrew N. Singh; Eric Sirota; Alexandra C. Sun; Weijuan Tang; David A. Thaisrivongs; Nimisha Thakur; Weidong Tong; Van Truong; Ryan Tsoi; Qiang Tu; Ben W. H. Turnbull; Ophelia Ukaegbu; David A. Vargas; Juan E. Velasquez; Deeptak Verma; Heather Wang; Tao Wang; Xiao Wang; Ying Wang; Zhixun Wang; Matthew S. Winston; Chunyu Wu; Brian M. Wyvratt; Kai-Jiong Xiao; Yingju Xu; Jia-Xuan Yan; Hao Yang; Victoria Zhang; Yongqian Zhang; Michelle Zheng; Wendy Zhong
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Biocatalytic Oxidative Desymmetrization of the Substituted Pyrrolidine Intermediate of MK-7845: An Investigational Antiviral Therapy for COVID-19MK-7845的取代吡咯烷中间体的生物催化氧化不对称反应:一种用于COVID-19的探索性抗病毒疗法
err2026-03-11
err0
PREAI
errShorouk O. Badir; Yangzhong Qin; Michelle Zheng; David A. Vargas; Birgit Kosjek; Ajit Vikram; Anna L. Dunn; Michael Whittington; Yining Ji; Keith A. Mattern; Alex M. Confer; Jonathan M. E. Hughes; Reed T. Larson; Justin A. Newman; Nastaran Salehi Marzijarani; Nadine Kuhl; Jamie M. McCabe Dunn
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Ketoreductase Engineering for a Chemoenzymatic Fluorination and Dynamic Kinetic Reduction Cascade酮还原酶工程用于化学酶促氟化和动态动力学还原级联
err2025-07-16
err0
PREAI
errStephanie W. Chun; Birgit Kosjek; Jackson K. B. Cahn; Amanda M. Makarewicz; Wai Ling Cheung-Lee; Deeptak Verma; Chey M. Jones; Alan Hruza; Jacob H. Forstater; Shasha Li; Quinn Gallagher; Grant S. Murphy; Jeffrey C. Moore
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Engineering Hydroxylase Activity, Selectivity, and Stability for a Scalable Concise Synthesis of a Key Intermediate to Belzutifan
err2024-02-19
err19
PREAI
errCheung-Lee, Wai Ling; Kolev, Joshua N.; Mcintosh, John A.; Gil, Agnieszka A.; Pan, Weilan; Xiao, Li; Velasquez, Juan E.; Gangam, Rekha; Winston, Matthew S.; Li, Shasha; Abe, Kotoe; Alwedi, Embarek; Dance, Zachary E. X.; Fan, Haiyang; Hiraga, Kaori; Kim, Jungchul; Kosjek, Birgit; Le, Diane N.; Marzijarani, Nastaran Salehi; Mattern, Keith; Mcmullen, Jonathan P.; Narsimhan, Karthik; Vikram, Ajit; Wang, Wei; Yan, Jia-Xuan; Yang, Rong-Sheng; Zhang, Victoria; Zhong, Wendy; Dirocco, Daniel A.; Morris, William J.; Murphy, Grant S.; Maloney, Kevin M.
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Evolution of a Green and Sustainable Manufacturing Process for Belzutifan: Part 5-Chemoenzymatic Diastereoselective Fluorination/DKR
err2024-02-07
err4
PREAI
errMccann, Scott D.; Dubina, Sean H.; Kosjek, Birgit; Alwedi, Embarek; Behre, Taylor; Burgess, Samantha A.; Dal Poggetto, Guilherme; Dirocco, Daniel A.; Hartmanshenn, Clara; Mcmullen, Jonathan P.; Padivitage, Nilusha; Sun, Alexandra C.
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Evolution of a Green and Sustainable Manufacturing Process for Belzutifan: Part 1-Process History and Development Strategy
err2024-02-05
err6
PREAI
errDiRocco, Daniel A.; Zhong, Yong-Li; Le, Diane N.; McCann, Scott D.; Hethcox, J. Caleb; Kim, Jungchul; Kolev, Joshua N.; Kosjek, Birgit; Dalby, Stephen M.; Mcmullen, Jonathan P.; Gangam, Rekha; Morris, William J.
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Driving Aspirational Process Mass Intensity Using Simple Structure-Based Prediction
err2022-04-18
err11
errOAAI
errSherer, Edward C.; Bagchi, Ansuman; Kosjek, Birgit; Maloney, Kevin M.; Peng, Zhengwei; Robaire, Sandra A.; Sheridan, Robert P.; Metwally, Essam; Campeau, Louis-Charles
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Scalable Asymmetric Synthesis of MK-8998, a T-Type Calcium Channel Antagonist
err2021-09-28
err2
PREAI
errZhong, Yong-Li; Moore, Jeffrey C.; Shevlin, Michael; Shultz, C. Scott; Kosjek, Birgit; Chen, Yonggang; Janey, Jacob M.; Tan, Lushi
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Improved iGAL 2.0 Metric Empowers Pharmaceutical Scientists to Make Meaningful Contributions to United Nations Sustainable Development Goal 12
err2021-08-12
err34
errOAAI
errRoschangar, Frank; Li, Jun; Zhou, Yanyan; Aelterman, Wim; Borovika, Alina; Colberg, Juan; Dickson, David P.; Gallou, Fabrice; Hayler, John D.; Koenig, Stefan G.; Kopach, Michael E.; Kosjek, Birgit; Leahy, David K.; O'Brien, Erin; Smith, Austin G.; Henry, Manuel; Cook, Jutta; Sheldon, Roger A.
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Harnessing the Power of Catalysis for the Synthesis of CRTH2 Antagonist MK-1029
err2021-06-02
err10
PREAI
errRuck, Rebecca T.; Pan, Jun; Vaswani, Rishi G.; Kosjek, Birgit; Strotman, Neil A.; Cai, Chaoxian; Humphrey, Guy R.
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Recent preparative applications of redox enzymes
err2019-04-01
err44
PREAI
errPrier, Christopher K.; Kosjek, Birgit
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Practical Asymmetric Synthesis of a Calcitonin Gene-Related Peptide (CGRP) Receptor Antagonist Ubrogepant
err2017-11-02
err29
PREAI
errYasuda, Nobuyoshi; Cleator, Ed; Kosjek, Birgit; Yin, Jianguo; Xiang, Bangping; Chen, Frank; Kuo, Shen-Chun; Belyk, Kevin; Mullens, Peter R.; Goodyear, Adrian; Edwards, John S.; Bishop, Brian; Ceglia, Scott; Belardi, Justin; Tan, Lushi; Song, Zhiguo J.; DiMichele, Lisa; Reamer, Robert; Cabiro, Fabien L.; Tang, Weng Lin; Liu, Guiquan
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Synthesis of the GPR40 Partial Agonist MK-8666 through a Kinetically Controlled Dynamic Enzymatic Ketone Reduction
err2016-11-01
err26
PREAI
errHyde, Alan M.; Liu, Zhijian; Kosjek, Birgit; Tan, Lushi; Klapars, Artis; Ashley, Eric It; Zhong, Yong-Li; Alvizo, Oscar; Agard, Nicholas J.; Liu, Guiquan; Gu, Xiuyan; Yasuda, Nobuyoshi; Limanto, John; Huffman, Mark K.; Tschaen, David M.
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Ene Reductase Enzymes for the Aromatisation of Tetralones and Cyclohexenones to Naphthols and Phenols
err2016-02-17
err7
PREAI
errKelly, Paul P.; Lipscom, David; Quinn, Derek J.; Lemon, Ken; Caswell, Jill; Spratt, Jenny; Kosjek, Birgit; Truppo, Matthew; Moody, Thomas S.
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Synthesis of Bis-Macrocyclic HCV Protease Inhibitor MK-6325 via Intramolecular sp2-sp3 Suzuki-Miyaura Coupling and Ring Closing Metathesis
err2015-03-10
err18
PREAI
errLi, Hongmei; Scott, Jeremy P.; Chen, Cheng-yi; Journet, Michel; Belyk, Kevin; Balsells, Jaume; Kosjek, Birgit; Baxter, Carl A.; Stewart, Gavin W.; Wise, Christopher; Alam, Mahbub; Song, Zhiguo Jake; Tan, Lushi
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Process Development of C-N Cross-Coupling and Enantioselective Biocatalytic Reactions for the Asymmetric Synthesis of Niraparib
err2013-10-25
err145
PREAI
errChung, Cheol K.; Bulger, Paul G.; Kosjek, Birgit; Belyk, Kevin M.; Rivera, Nelo; Scott, Mark E.; Humphrey, Guy R.; Limanto, John; Bachert, Donald C.; Emerson, Khateeta M.
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CRTH2 Antagonist MK-7246: A Synthetic Evolution from Discovery through Development
err2012-02-15
err113
PREAI
errMolinaro, Carmela; Bulger, Paul G.; Lee, Ernest E.; Kosjek, Birgit; Lau, Stephen; Gauvreau, Danny; Howard, Melissa E.; Wallace, Debra J.; O'Shea, Paul D.
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Resolution of 2,2-Disubstituted Epoxides via Biocatalytic Azidolysis
err2010-08-03
err58
PREAI
errMolinaro, Carmela; Guilbault, Audrey-Anne; Kosjek, Birgit
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